JP2013533267A5 - - Google Patents
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- Publication number
- JP2013533267A5 JP2013533267A5 JP2013520191A JP2013520191A JP2013533267A5 JP 2013533267 A5 JP2013533267 A5 JP 2013533267A5 JP 2013520191 A JP2013520191 A JP 2013520191A JP 2013520191 A JP2013520191 A JP 2013520191A JP 2013533267 A5 JP2013533267 A5 JP 2013533267A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- group
- compound
- alkyl group
- branched
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 0 *c(cc1)ccc1N=O Chemical compound *c(cc1)ccc1N=O 0.000 description 2
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR1055951 | 2010-07-21 | ||
| FR1055951A FR2963006B1 (fr) | 2010-07-21 | 2010-07-21 | Procede de preparation de derives de nitro-benzofurane |
| PCT/FR2011/051751 WO2012010802A1 (fr) | 2010-07-21 | 2011-07-20 | Procede de preparation de derives de benzofurane substitues en position 5 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013533267A JP2013533267A (ja) | 2013-08-22 |
| JP2013533267A5 true JP2013533267A5 (enExample) | 2014-07-10 |
Family
ID=42790926
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013520191A Pending JP2013533267A (ja) | 2010-07-21 | 2011-07-20 | ５位で置換されたべンゾフラン誘導体の調製方法 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US8748636B2 (enExample) |
| EP (1) | EP2595977A1 (enExample) |
| JP (1) | JP2013533267A (enExample) |
| KR (1) | KR20130094305A (enExample) |
| CN (1) | CN103221401A (enExample) |
| AU (1) | AU2011281435A1 (enExample) |
| BR (1) | BR112013001365A2 (enExample) |
| CA (1) | CA2805868A1 (enExample) |
| FR (1) | FR2963006B1 (enExample) |
| MX (1) | MX2013000845A (enExample) |
| RU (1) | RU2013107600A (enExample) |
| SG (1) | SG187565A1 (enExample) |
| WO (1) | WO2012010802A1 (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HUP0900759A2 (en) | 2009-12-08 | 2011-11-28 | Sanofi Aventis | Novel process for producing dronedarone |
| HUP1000010A2 (en) | 2010-01-08 | 2011-11-28 | Sanofi Sa | Process for producing dronedarone |
| FR2958290B1 (fr) | 2010-03-30 | 2012-10-19 | Sanofi Aventis | Procede de preparation de derives de sulfonamido-benzofurane |
| HUP1000330A2 (en) | 2010-06-18 | 2011-12-28 | Sanofi Sa | Process for the preparation of dronedarone and the novel intermediates |
| FR2962731B1 (fr) | 2010-07-19 | 2012-08-17 | Sanofi Aventis | Procede de preparation de derives d'amino-benzoyl-benzofurane |
| HUP1100167A2 (en) | 2011-03-29 | 2012-11-28 | Sanofi Sa | Process for preparation of dronedarone by mesylation |
| HUP1100165A2 (en) | 2011-03-29 | 2012-12-28 | Sanofi Sa | Process for preparation of dronedarone by n-butylation |
| FR2983198B1 (fr) | 2011-11-29 | 2013-11-15 | Sanofi Sa | Procede de preparation de derives de 5-amino-benzoyl-benzofurane |
| EP2617718A1 (en) | 2012-01-20 | 2013-07-24 | Sanofi | Process for preparation of dronedarone by the use of dibutylaminopropanol reagent |
| WO2013121235A2 (en) | 2012-02-13 | 2013-08-22 | Sanofi | Process for preparation of dronedarone by removal of hydroxyl group |
| US9249119B2 (en) | 2012-02-14 | 2016-02-02 | Sanofi | Process for the preparation of dronedarone by oxidation of a sulphenyl group |
| WO2013124745A1 (en) | 2012-02-22 | 2013-08-29 | Sanofi | Process for preparation of dronedarone by oxidation of a hydroxyl group |
| WO2013178337A1 (en) | 2012-05-31 | 2013-12-05 | Sanofi | Process for preparation of dronedarone by grignard reaction |
| CN109384754B (zh) * | 2017-08-14 | 2020-06-09 | 新发药业有限公司 | 一种盐酸决奈达隆的制备方法 |
Family Cites Families (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2337396A1 (de) * | 1973-07-23 | 1975-02-13 | Hoechst Ag | Verfahren zur herstellung aromatischer 1,3-diketone |
| FR2665444B1 (fr) | 1990-08-06 | 1992-11-27 | Sanofi Sa | Derives d'amino-benzofuranne, benzothiophene ou indole, leur procede de preparation ainsi que les compositions les contenant. |
| IT1275997B1 (it) * | 1995-03-31 | 1997-10-24 | Great Lakes Chemical Italia | Enammine come accelleranti di vulcanizzazione per gomme naturali o sintetiche |
| FR2813306B1 (fr) | 2000-08-23 | 2005-10-21 | Sanofi Synthelabo | Aminoalkybenzoyl-benzofurannes ou benzothiophenes, leur procede de preparation et les compositions les contenant |
| FR2813308B1 (fr) * | 2000-08-23 | 2005-07-01 | Sanofi Synthelabo | Aminoalkoxybenzoyl-benzofurannes ou benzothiophenes, leur procede de preparation ainsi que les compositions les contenant |
| FR2817865B1 (fr) | 2000-12-11 | 2005-02-18 | Sanofi Synthelabo | Derive aminoalkoxybenzoyle sous forme de sel, son procede de preparation et son utilisation comme intermediaire de synthese |
| FR2817864B1 (fr) | 2000-12-11 | 2003-02-21 | Sanofi Synthelabo | Derive de methanesulfonamido-benzofurane, son procede de preparation et son utilisation comme intermediaire de synthese |
| DE60319158T2 (de) * | 2003-07-03 | 2009-02-05 | Aventis Pharmaceuticals Inc. | Pyrazoloisochinolinenderivaten als kinase inhibitoren |
| GB0719180D0 (en) * | 2007-10-02 | 2007-11-14 | Cambrex Karlskoga Ab | New process |
| CN102171200B (zh) * | 2008-10-02 | 2015-09-30 | 坎布雷卡尔斯库加公司 | 用于制备二酮类和药物的方法 |
| EP2344467A1 (en) * | 2008-10-10 | 2011-07-20 | Lonza Ltd. | Process for preparing 2-alkyl-3-aroyl-5-nitro-benzofurans |
| TW201111354A (en) | 2009-05-27 | 2011-04-01 | Sanofi Aventis | Process for the production of Dronedarone intermediates |
| TW201107303A (en) | 2009-05-27 | 2011-03-01 | Sanofi Aventis | Process for the production of benzofurans |
| HUP0900759A2 (en) | 2009-12-08 | 2011-11-28 | Sanofi Aventis | Novel process for producing dronedarone |
| HUP1000010A2 (en) | 2010-01-08 | 2011-11-28 | Sanofi Sa | Process for producing dronedarone |
| FR2957079B1 (fr) | 2010-03-02 | 2012-07-27 | Sanofi Aventis | Procede de synthese de derives de cetobenzofurane |
| FR2962731B1 (fr) | 2010-07-19 | 2012-08-17 | Sanofi Aventis | Procede de preparation de derives d'amino-benzoyl-benzofurane |
| FR2973027A1 (fr) | 2011-03-24 | 2012-09-28 | Sanofi Aventis | Procede de synthese de derives de cetobenzofurane |
| HUP1100167A2 (en) | 2011-03-29 | 2012-11-28 | Sanofi Sa | Process for preparation of dronedarone by mesylation |
| HUP1100166A2 (en) | 2011-03-29 | 2012-12-28 | Sanofi Sa | Reductive amination process for preparation of dronedarone using amine intermediary compound |
| HUP1100165A2 (en) | 2011-03-29 | 2012-12-28 | Sanofi Sa | Process for preparation of dronedarone by n-butylation |
-
2010
- 2010-07-21 FR FR1055951A patent/FR2963006B1/fr not_active Expired - Fee Related
-
2011
- 2011-07-20 RU RU2013107600/04A patent/RU2013107600A/ru not_active Application Discontinuation
- 2011-07-20 MX MX2013000845A patent/MX2013000845A/es unknown
- 2011-07-20 WO PCT/FR2011/051751 patent/WO2012010802A1/fr not_active Ceased
- 2011-07-20 BR BR112013001365A patent/BR112013001365A2/pt not_active Application Discontinuation
- 2011-07-20 KR KR1020137004233A patent/KR20130094305A/ko not_active Withdrawn
- 2011-07-20 SG SG2013004338A patent/SG187565A1/en unknown
- 2011-07-20 CN CN2011800454136A patent/CN103221401A/zh active Pending
- 2011-07-20 CA CA2805868A patent/CA2805868A1/fr not_active Abandoned
- 2011-07-20 EP EP11754896.6A patent/EP2595977A1/fr not_active Withdrawn
- 2011-07-20 AU AU2011281435A patent/AU2011281435A1/en not_active Abandoned
- 2011-07-20 JP JP2013520191A patent/JP2013533267A/ja active Pending
-
2013
- 2013-01-16 US US13/742,810 patent/US8748636B2/en active Active
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