JP2013526523A - メトプロロールを含むアルコール耐性持続放出性経口剤形 - Google Patents
メトプロロールを含むアルコール耐性持続放出性経口剤形 Download PDFInfo
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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| PCT/US2011/035770 WO2011143120A1 (en) | 2010-05-11 | 2011-05-09 | Alcoholres i stant metoprolol - containing extended - release oral dosage forms |
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| CA2784407A1 (en) * | 2009-12-17 | 2011-07-14 | Cima Labs Inc. | Abuse-resistant formulations |
| PT3164117T (pt) | 2014-07-03 | 2023-12-12 | SpecGx LLC | Formulações de libertação imediata de dissuasão de abuso compreendendo polissacáridos não celulósicos |
| ES3008933T3 (en) | 2015-09-29 | 2025-03-25 | Merz Pharmaceuticals Llc | Sustained release compositions of 4-aminopyridine |
| ES3040411T3 (en) | 2018-03-22 | 2025-10-30 | Incarda Therapeutics Inc | A novel method to slow ventricular rate |
| WO2020068510A1 (en) | 2018-09-25 | 2020-04-02 | SpecGx LLC | Abuse deterrent immediate release capsule dosage forms |
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| JPH01128917A (ja) * | 1987-10-08 | 1989-05-22 | Haessle:Ab | 新規な薬学的製剤およびその製法 |
| US20070009589A1 (en) * | 2005-07-07 | 2007-01-11 | Kandarapu Raghupathi | Extended release compositions |
| WO2007048233A1 (en) * | 2005-10-24 | 2007-05-03 | Orbus Pharma Inc. | Stabilized extended release pharmaceutical compositions comprising a beta-adrenoreceptor antagonist |
| WO2008033523A1 (en) * | 2006-09-15 | 2008-03-20 | Cima Labs Inc. | Abuse resistant drug formulation |
| WO2009035474A1 (en) * | 2007-09-13 | 2009-03-19 | Cima Labs Inc. | Abuse resistant drug formulation |
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2011
- 2011-05-09 CA CA2798702A patent/CA2798702A1/en not_active Abandoned
- 2011-05-09 JP JP2013510209A patent/JP2013526523A/ja active Pending
- 2011-05-09 MX MX2012012991A patent/MX2012012991A/es not_active Application Discontinuation
- 2011-05-09 US US13/721,128 patent/US8927025B2/en not_active Expired - Fee Related
- 2011-05-09 WO PCT/US2011/035770 patent/WO2011143120A1/en not_active Ceased
- 2011-05-09 EP EP11720364A patent/EP2568977A1/en not_active Withdrawn
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Also Published As
| Publication number | Publication date |
|---|---|
| US8927025B2 (en) | 2015-01-06 |
| CA2798702A1 (en) | 2011-11-17 |
| US20130266660A1 (en) | 2013-10-10 |
| WO2011143120A1 (en) | 2011-11-17 |
| MX2012012991A (es) | 2012-11-30 |
| EP2568977A1 (en) | 2013-03-20 |
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