JP2013525490A5 - - Google Patents
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- Publication number
- JP2013525490A5 JP2013525490A5 JP2013509201A JP2013509201A JP2013525490A5 JP 2013525490 A5 JP2013525490 A5 JP 2013525490A5 JP 2013509201 A JP2013509201 A JP 2013509201A JP 2013509201 A JP2013509201 A JP 2013509201A JP 2013525490 A5 JP2013525490 A5 JP 2013525490A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- hydroxyl
- optionally substituted
- halo
- het
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US33197410P | 2010-05-06 | 2010-05-06 | |
| US61/331,974 | 2010-05-06 | ||
| PCT/US2011/035091 WO2011140164A1 (en) | 2010-05-06 | 2011-05-04 | Aza-indole derivatives useful as modulators of faah |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013525490A JP2013525490A (ja) | 2013-06-20 |
| JP2013525490A5 true JP2013525490A5 (https=) | 2014-06-05 |
Family
ID=44904047
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013509201A Pending JP2013525490A (ja) | 2010-05-06 | 2011-05-04 | Ｆａａｈのモジュレータとして有用なアザインドール誘導体 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20130059850A1 (https=) |
| EP (1) | EP2566481A4 (https=) |
| JP (1) | JP2013525490A (https=) |
| CN (1) | CN102917707A (https=) |
| AU (1) | AU2011248175A1 (https=) |
| BR (1) | BR112012028055A2 (https=) |
| CA (1) | CA2797281A1 (https=) |
| WO (1) | WO2011140164A1 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201411236D0 (en) | 2014-06-25 | 2014-08-06 | Takeda Pharmaceutical | Novel compounds |
| US10426758B2 (en) | 2015-10-13 | 2019-10-01 | Institut National De La Sante Et De La Recherche Medicale (Inserm) | Sibiriline derivatives for use for preventing and/or treating disorders associated with cellular necroptosis |
| CA3036776A1 (en) * | 2016-09-16 | 2018-03-22 | Sumitomo Chemical Company, Limited | Heterocyclic compound, and harmful-arthropod-controlling agent containing same |
| CN109589325B (zh) * | 2019-02-19 | 2019-11-26 | 牡丹江医学院 | 一种用于治疗肠炎的药物组合物及其制备方法 |
| EP3983384B1 (en) * | 2019-06-17 | 2023-10-11 | UCB Pharma GmbH | N-(phenyl)-indole-3-sulfonamide derivatives and related compounds as gpr17 modulators for treating cns disorders such as multiple sclerosis |
| CN111743864B (zh) * | 2020-08-05 | 2022-04-01 | 牡丹江医学院 | 一种体育外伤喷雾剂及其制备方法 |
| CN112159423A (zh) * | 2020-11-03 | 2021-01-01 | 凯美克(上海)医药科技有限公司 | 1H-吡咯并[2,3-b]吡啶-2-硼酸频哪醇酯的合成方法 |
| JP2024506530A (ja) * | 2021-01-25 | 2024-02-14 | シービーライフ | フェロトーシス制御性細胞死の阻害剤としてのインドール、６－および７－アザインドール誘導体の使用 |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH574441A5 (https=) * | 1973-06-14 | 1976-04-15 | Ciba Geigy Ag | |
| JPS5239672A (en) * | 1975-09-26 | 1977-03-28 | Sankyo Co Ltd | Process for preparing indole-2-allyl-3- thioeter compounds |
| NZ222878A (en) * | 1986-12-17 | 1991-02-26 | Merck Frosst Canada Inc | 3-hetero-substituted-n-benzyl-indole derivatives, and pharmaceutical compositions |
| US5095031A (en) * | 1990-08-20 | 1992-03-10 | Abbott Laboratories | Indole derivatives which inhibit leukotriene biosynthesis |
| US5527819A (en) * | 1991-09-06 | 1996-06-18 | Merck & Co., Inc. | Inhibitors of HIV reverse transcriptase |
| HUT74614A (en) * | 1993-02-24 | 1997-01-28 | Merck & Co Inc | Nindol derivates suitable for treatment of infection by hiv and pharmaceutical compositions containing them |
| FR2705346B1 (fr) * | 1993-05-18 | 1995-08-11 | Union Pharma Scient Appl | Nouveaux dérivés de pipéridinyl thio indole, leurs procédés de préparation, compositions pharmaceutiques les contenant, utiles notamment comme antalgiques . |
| CA2473803A1 (en) * | 2002-02-01 | 2003-08-07 | Robert Greenhouse | Substituted indoles as alpha-1 agonists |
| UA78999C2 (en) * | 2002-06-04 | 2007-05-10 | Wyeth Corp | 1-(aminoalkyl)-3-sulfonylazaindoles as ligands of 5-hydroxytryptamine-6 |
| TW200403243A (en) * | 2002-07-18 | 2004-03-01 | Wyeth Corp | 1-Heterocyclylalkyl-3-sulfonylazaindole or-azaindazole derivatives as 5-hydroxytryptamine-6 ligands |
| US6800655B2 (en) * | 2002-08-20 | 2004-10-05 | Sri International | Analogs of indole-3-carbinol metabolites as chemotherapeutic and chemopreventive agents |
| EP1592690A1 (en) * | 2003-02-14 | 2005-11-09 | Wyeth | Heterocyclyl-3-sulfonylazaindole or -azaindazole derivatives as 5-hydroxytryptamine-6 ligands |
| EP1781654A1 (en) * | 2004-07-27 | 2007-05-09 | SGX Pharmaceuticals, Inc. | Pyrrolo-pyridine kinase modulators |
| BRPI0514397A (pt) * | 2004-08-19 | 2008-06-10 | Aventis Pharma Inc | derivados de 3-ariltioindol-2-carboxamida e análogos destes como inibidores de caseìna cinase iépsilon |
| GB2422831A (en) * | 2005-02-04 | 2006-08-09 | Oxagen Ltd | Pyrrolopyridines and their use in the treatment of diseases mediated by PGD2 at the CRTH2 receptor |
| CN102206216B (zh) * | 2005-06-22 | 2014-11-12 | 普莱希科公司 | 作为蛋白质激酶抑制剂的吡咯并[2,3-b]吡啶衍生物 |
| US7960544B2 (en) * | 2005-12-16 | 2011-06-14 | Ironwood Pharmaceuticals, Inc. | Useful indole compounds |
| TW200914437A (en) * | 2007-06-20 | 2009-04-01 | Ironwood Pharmaceuticals Inc | FAAH inhibitors |
| BRPI0908851A2 (pt) * | 2008-02-22 | 2017-05-30 | Irm Llc | compostos e composições como moduladores da atividades de gpr119 |
| AU2009237657B2 (en) * | 2008-04-16 | 2013-04-04 | Oasmia Pharmaceutical Ab | Novel estrogen receptor ligands |
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2011
- 2011-05-04 AU AU2011248175A patent/AU2011248175A1/en not_active Abandoned
- 2011-05-04 EP EP11778226.8A patent/EP2566481A4/en not_active Withdrawn
- 2011-05-04 JP JP2013509201A patent/JP2013525490A/ja active Pending
- 2011-05-04 CA CA2797281A patent/CA2797281A1/en not_active Abandoned
- 2011-05-04 US US13/696,520 patent/US20130059850A1/en not_active Abandoned
- 2011-05-04 BR BR112012028055A patent/BR112012028055A2/pt not_active IP Right Cessation
- 2011-05-04 WO PCT/US2011/035091 patent/WO2011140164A1/en not_active Ceased
- 2011-05-04 CN CN2011800228440A patent/CN102917707A/zh active Pending