JP2012532186A5 - - Google Patents

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Publication number
JP2012532186A5
JP2012532186A5 JP2012519061A JP2012519061A JP2012532186A5 JP 2012532186 A5 JP2012532186 A5 JP 2012532186A5 JP 2012519061 A JP2012519061 A JP 2012519061A JP 2012519061 A JP2012519061 A JP 2012519061A JP 2012532186 A5 JP2012532186 A5 JP 2012532186A5
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JP
Japan
Prior art keywords
formula
acetylating
anhydride
agents
iic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2012519061A
Other languages
English (en)
Japanese (ja)
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JP2012532186A (ja
JP5675800B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/GB2010/051100 external-priority patent/WO2011004182A1/en
Publication of JP2012532186A publication Critical patent/JP2012532186A/ja
Publication of JP2012532186A5 publication Critical patent/JP2012532186A5/ja
Application granted granted Critical
Publication of JP5675800B2 publication Critical patent/JP5675800B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2012519061A 2009-07-06 2010-07-05 4−(アセチルアミノ))−3−[(4−クロロ−フェニル)チオ]−2−メチル−1h−インドール−1−酢酸の製造のための中間体および方法 Expired - Fee Related JP5675800B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US22316309P 2009-07-06 2009-07-06
US61/223,163 2009-07-06
PCT/GB2010/051100 WO2011004182A1 (en) 2009-07-06 2010-07-05 Intermediates and processes for the preparation of 4- (acetylamino) ) -3- [ (4-chloro-phenyl) thio] -2-methyl-1h-indole-1-acetic acid

Publications (3)

Publication Number Publication Date
JP2012532186A JP2012532186A (ja) 2012-12-13
JP2012532186A5 true JP2012532186A5 (enExample) 2013-07-04
JP5675800B2 JP5675800B2 (ja) 2015-02-25

Family

ID=42780497

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012519061A Expired - Fee Related JP5675800B2 (ja) 2009-07-06 2010-07-05 4−(アセチルアミノ))−3−[(4−クロロ−フェニル)チオ]−2−メチル−1h−インドール−1−酢酸の製造のための中間体および方法

Country Status (16)

Country Link
US (1) US8227622B2 (enExample)
EP (1) EP2451780B1 (enExample)
JP (1) JP5675800B2 (enExample)
KR (1) KR101752932B1 (enExample)
CN (1) CN102482214B (enExample)
AR (1) AR077457A1 (enExample)
AU (1) AU2010270050B9 (enExample)
BR (1) BR112012000353B1 (enExample)
CA (1) CA2767132C (enExample)
ES (1) ES2426679T3 (enExample)
IL (1) IL217088A0 (enExample)
MX (1) MX2012000229A (enExample)
RU (1) RU2551852C2 (enExample)
SG (1) SG177286A1 (enExample)
TW (1) TW201118067A (enExample)
WO (1) WO2011004182A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104817544B (zh) * 2015-03-23 2017-05-10 三峡大学 一种四氢吲哚‑4‑酮肟类药物,制备方法及其应用
JP6472419B2 (ja) * 2015-09-30 2019-02-20 富士フイルム株式会社 芳香族化合物の製造方法
JP6452584B2 (ja) * 2015-09-30 2019-01-16 富士フイルム株式会社 芳香族化合物の製造方法

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6916841B2 (en) 1998-02-25 2005-07-12 Genetics Institute, Llc Inhibitors of phospholipase enzymes
WO2001032621A1 (en) 1999-10-29 2001-05-10 Wakunaga Pharmaceutical Co., Ltd. Novel indole derivatives and drugs containing the same as the active ingredient
TWI317634B (en) 2001-12-13 2009-12-01 Nat Health Research Institutes Aroyl indoles compounds
TW200307542A (en) 2002-05-30 2003-12-16 Astrazeneca Ab Novel compounds
SE0202241D0 (sv) 2002-07-17 2002-07-17 Astrazeneca Ab Novel Compounds
SE0301569D0 (sv) 2003-05-27 2003-05-27 Astrazeneca Ab Novel compounds
SE0302232D0 (sv) 2003-08-18 2003-08-18 Astrazeneca Ab Novel Compounds
GB0428100D0 (en) 2004-12-23 2005-01-26 Astrazeneca Ab Chemical processes & intermediates
GB0500604D0 (en) 2005-01-13 2005-02-16 Astrazeneca Ab Novel process
GB0500643D0 (en) 2005-01-13 2005-02-23 Renovo Ltd Medicaments
GB2422831A (en) 2005-02-04 2006-08-09 Oxagen Ltd Pyrrolopyridines and their use in the treatment of diseases mediated by PGD2 at the CRTH2 receptor
JP2009538289A (ja) 2006-05-26 2009-11-05 アストラゼネカ・アクチエボラーグ ビアリールまたはヘテロアリール置換インドール
CA2654026A1 (en) 2006-06-08 2007-12-13 Neurokey A/S Use of cannabinoid receptor agonists as hypothermia inducing drugs for the treatment of ischemia
CA2656150A1 (en) 2006-06-28 2008-01-03 Sanofi-Aventis New cxcr2 inhibitors

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