JP2012531456A5 - - Google Patents

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Publication number
JP2012531456A5
JP2012531456A5 JP2012518092A JP2012518092A JP2012531456A5 JP 2012531456 A5 JP2012531456 A5 JP 2012531456A5 JP 2012518092 A JP2012518092 A JP 2012518092A JP 2012518092 A JP2012518092 A JP 2012518092A JP 2012531456 A5 JP2012531456 A5 JP 2012531456A5
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JP
Japan
Prior art keywords
alkyl
amide
methyl
dicarboxylic acid
pyrrolidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2012518092A
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English (en)
Japanese (ja)
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JP2012531456A (ja
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Publication date
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Priority claimed from PCT/EP2010/059352 external-priority patent/WO2011000905A1/en
Publication of JP2012531456A publication Critical patent/JP2012531456A/ja
Publication of JP2012531456A5 publication Critical patent/JP2012531456A5/ja
Pending legal-status Critical Current

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JP2012518092A 2009-07-02 2010-07-01 置換２−カルボキサミドシクロアミノウレア類 Pending JP2012531456A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US27002909P 2009-07-02 2009-07-02
US61/270,029 2009-07-02
PCT/EP2010/059352 WO2011000905A1 (en) 2009-07-02 2010-07-01 Substituted 2-carboxamide cycloamino ureas

Publications (2)

Publication Number Publication Date
JP2012531456A JP2012531456A (ja) 2012-12-10
JP2012531456A5 true JP2012531456A5 (enExample) 2013-08-01

Family

ID=42727680

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012518092A Pending JP2012531456A (ja) 2009-07-02 2010-07-01 置換２−カルボキサミドシクロアミノウレア類

Country Status (14)

Country Link
US (1) US8293753B2 (enExample)
EP (1) EP2448935B1 (enExample)
JP (1) JP2012531456A (enExample)
KR (1) KR20120092552A (enExample)
CN (1) CN102471332A (enExample)
AR (1) AR077367A1 (enExample)
AU (1) AU2010268019A1 (enExample)
BR (1) BRPI1015909A2 (enExample)
CA (1) CA2766855A1 (enExample)
EA (1) EA201200086A1 (enExample)
MX (1) MX2012000177A (enExample)
TW (1) TW201105666A (enExample)
UY (1) UY32747A (enExample)
WO (1) WO2011000905A1 (enExample)

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CN104350144B (zh) 2012-05-23 2017-08-04 弗·哈夫曼-拉罗切有限公司 获得和使用内胚层和肝细胞的组合物和方法
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US9156831B2 (en) 2013-01-23 2015-10-13 Astrazeneca Ab Chemical compounds
TWI736135B (zh) 2013-03-01 2021-08-11 美商英塞特控股公司 吡唑并嘧啶衍生物治療PI3Kδ相關病症之用途
TW201726140A (zh) 2015-09-17 2017-08-01 瑞典商阿斯特捷利康公司 治療癌症之新型生物標記及方法
AU2019355574A1 (en) 2018-10-05 2021-05-06 Sloan-Kettering Institute For Cancer Research PI3K inhibitors and uses thereof
WO2024089272A1 (en) * 2022-10-28 2024-05-02 Institut National De La Sante Et De La Recherche Medicale New inhibitors of phosphatidylinositol 3-kinase
CN116239591B (zh) * 2023-02-14 2025-09-23 嘉兴大学 一种(4r)-磺酰氨基-l-脯氨酰胺类化合物、制备方法、应用及其药物组合
CN116987072A (zh) * 2023-07-27 2023-11-03 武汉呈瑞生物医药科技有限公司 化合物及其应用
EP4643858A1 (en) * 2024-04-29 2025-11-05 Institut National de la Santé et de la Recherche Médicale Methods and pharmaceutical composition for the treatment of uterine disease

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