JP2012528858A5 - - Google Patents

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Publication number
JP2012528858A5
JP2012528858A5 JP2012513932A JP2012513932A JP2012528858A5 JP 2012528858 A5 JP2012528858 A5 JP 2012528858A5 JP 2012513932 A JP2012513932 A JP 2012513932A JP 2012513932 A JP2012513932 A JP 2012513932A JP 2012528858 A5 JP2012528858 A5 JP 2012528858A5
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JP
Japan
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JP2012513932A
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English (en)
Japanese (ja)
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JP2012528858A (ja
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Priority claimed from PCT/US2010/001596 external-priority patent/WO2010141074A2/en
Publication of JP2012528858A publication Critical patent/JP2012528858A/ja
Publication of JP2012528858A5 publication Critical patent/JP2012528858A5/ja
Pending legal-status Critical Current

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JP2012513932A 2009-06-01 2010-06-01 O−GlcNAc転移酵素阻害剤およびその使用 Pending JP2012528858A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US21751409P 2009-06-01 2009-06-01
US61/217,514 2009-06-01
PCT/US2010/001596 WO2010141074A2 (en) 2009-06-01 2010-06-01 O-glcnac transferase inhibitors and uses thereof

Publications (2)

Publication Number Publication Date
JP2012528858A JP2012528858A (ja) 2012-11-15
JP2012528858A5 true JP2012528858A5 (enExample) 2014-05-22

Family

ID=43298360

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012513932A Pending JP2012528858A (ja) 2009-06-01 2010-06-01 O−GlcNAc転移酵素阻害剤およびその使用

Country Status (4)

Country Link
US (1) US8957075B2 (enExample)
EP (1) EP2438046A4 (enExample)
JP (1) JP2012528858A (enExample)
WO (1) WO2010141074A2 (enExample)

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WO2010141074A2 (en) 2009-06-01 2010-12-09 President And Fellows Of Harvard College O-glcnac transferase inhibitors and uses thereof
US9573911B2 (en) 2011-07-06 2017-02-21 President And Fellows Of Harvard College Diphosphate mimetics and uses thereof
WO2013027168A1 (en) * 2011-08-22 2013-02-28 Pfizer Inc. Novel heterocyclic compounds as bromodomain inhibitors
CN104470515B (zh) * 2012-05-03 2016-12-07 圣路易斯药学院 用于增加神经营养肽的组合物和方法
US20170166558A1 (en) * 2014-07-01 2017-06-15 President And Fellows Of Harvard College O-glcnac transferase (ogt) inhibitors and uses thereof
CN107903185B (zh) * 2017-11-08 2020-05-26 四川大学 新型eEF2K抑制剂的制备及应用
WO2020047251A1 (en) * 2018-08-29 2020-03-05 President And Fellows Of Harvard College O-glcnac transferase inhibitors and uses thereof
UY38934A (es) * 2019-10-29 2021-05-31 Biogen Ma Inc Inhibidores de o-glucoproteína-2-acetamido-2-deoxi-3-d-glucopiranosidasa espirocíclica
DE102019129527A1 (de) 2019-10-31 2021-05-06 Forschungszentrum Jülich GmbH Inhibitoren für Bromodomänen
KR102571503B1 (ko) * 2020-09-14 2023-08-28 부산대학교 산학협력단 암질환 예방 또는 치료용 조성물

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