JP2012514009A5 - - Google Patents

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JP2012514009A5
JP2012514009A5 JP2011543730A JP2011543730A JP2012514009A5 JP 2012514009 A5 JP2012514009 A5 JP 2012514009A5 JP 2011543730 A JP2011543730 A JP 2011543730A JP 2011543730 A JP2011543730 A JP 2011543730A JP 2012514009 A5 JP2012514009 A5 JP 2012514009A5
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pharmaceutically acceptable
acceptable salt
pharmaceutical composition
compound according
treating
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JP2011543730A
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JP2012514009A (ja
JP5502106B2 (ja
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Priority claimed from PCT/US2009/069852 external-priority patent/WO2010078449A2/en
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JP2011543730A 2008-12-31 2009-12-30 体液貯留または塩分過負荷と関連する障害および消化管障害の治療におけるnhe媒介性アンチポートを阻害するための組成物および方法 Active JP5502106B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US14185308P 2008-12-31 2008-12-31
US61/141,853 2008-12-31
US16950909P 2009-04-15 2009-04-15
US61/169,509 2009-04-15
US23784209P 2009-08-28 2009-08-28
US61/237,842 2009-08-28
PCT/US2009/069852 WO2010078449A2 (en) 2008-12-31 2009-12-30 Compounds and methods for inhibiting nhe-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders

Related Child Applications (1)

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JP2014010049A Division JP5805802B2 (ja) 2008-12-31 2014-01-23 体液貯留または塩分過負荷と関連する障害および消化管障害の治療におけるnhe媒介性アンチポートを阻害するための組成物および方法

Publications (3)

Publication Number Publication Date
JP2012514009A JP2012514009A (ja) 2012-06-21
JP2012514009A5 true JP2012514009A5 (enExample) 2014-03-13
JP5502106B2 JP5502106B2 (ja) 2014-05-28

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Family Applications (2)

Application Number Title Priority Date Filing Date
JP2011543730A Active JP5502106B2 (ja) 2008-12-31 2009-12-30 体液貯留または塩分過負荷と関連する障害および消化管障害の治療におけるnhe媒介性アンチポートを阻害するための組成物および方法
JP2014010049A Active JP5805802B2 (ja) 2008-12-31 2014-01-23 体液貯留または塩分過負荷と関連する障害および消化管障害の治療におけるnhe媒介性アンチポートを阻害するための組成物および方法

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JP2014010049A Active JP5805802B2 (ja) 2008-12-31 2014-01-23 体液貯留または塩分過負荷と関連する障害および消化管障害の治療におけるnhe媒介性アンチポートを阻害するための組成物および方法

Country Status (22)

Country Link
US (4) US8541448B2 (enExample)
EP (3) EP2384318B1 (enExample)
JP (2) JP5502106B2 (enExample)
KR (5) KR20220042487A (enExample)
CN (2) CN103819403B (enExample)
AU (1) AU2009334511C1 (enExample)
BR (1) BRPI0923861B8 (enExample)
CA (1) CA2748607A1 (enExample)
CY (1) CY1120451T1 (enExample)
DK (1) DK2384318T3 (enExample)
ES (1) ES2657938T3 (enExample)
HR (1) HRP20180289T1 (enExample)
HU (1) HUE036405T2 (enExample)
IL (3) IL213852A (enExample)
LT (1) LT2384318T (enExample)
MX (3) MX2011007024A (enExample)
NO (1) NO2384318T3 (enExample)
PL (1) PL2384318T3 (enExample)
PT (1) PT2384318T (enExample)
SI (1) SI2384318T1 (enExample)
SM (1) SMT201800071T1 (enExample)
WO (1) WO2010078449A2 (enExample)

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CN109897044A (zh) * 2017-12-07 2019-06-18 北京大学 抗神经病理性疼痛化合物及其制备方法
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WO2020181555A1 (zh) 2019-03-14 2020-09-17 深圳仁泰医药科技有限公司 Nhe3抑制剂的晶型a及其制备方法和应用
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CN111217490B (zh) * 2019-12-30 2024-09-06 北京航天环境工程有限公司 一种轻型填料的双层生物滤池系统和应用
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CN112047881B (zh) * 2020-10-10 2023-04-11 山东汇海医药化工有限公司 一种坦帕诺的制备方法
TWI805137B (zh) * 2020-12-18 2023-06-11 大陸商上海濟煜醫藥科技有限公司 苯并雜環取代四氫異喹啉類化合物
CN114805202A (zh) * 2021-01-28 2022-07-29 江西济民可信集团有限公司 苯磺酰胺类化合物及其制备方法和应用
KR20250047720A (ko) * 2022-06-20 2025-04-04 상하이 제유 파마슈티칼 컴퍼니 리미티드 벤조헤테로고리 치환 테트라히드로이소퀴놀린 화합물 염 형태 및 이의 제조 방법
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