JP2012505836A5 - - Google Patents
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- Publication number
- JP2012505836A5 JP2012505836A5 JP2011531305A JP2011531305A JP2012505836A5 JP 2012505836 A5 JP2012505836 A5 JP 2012505836A5 JP 2011531305 A JP2011531305 A JP 2011531305A JP 2011531305 A JP2011531305 A JP 2011531305A JP 2012505836 A5 JP2012505836 A5 JP 2012505836A5
- Authority
- JP
- Japan
- Prior art keywords
- amino
- benzofuran
- oxadiazol
- diol
- propane
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AU2008905369 | 2008-10-17 | ||
| AU2008905369A AU2008905369A0 (en) | 2008-10-17 | S1P Receptors Modulators and Their use Thereof | |
| AU2009903644 | 2009-08-05 | ||
| AU2009903644A AU2009903644A0 (en) | 2009-08-05 | S1P Receptors Modulators and their use Thereof | |
| PCT/AU2009/001371 WO2010043000A1 (en) | 2008-10-17 | 2009-10-19 | S1p receptors modulators and their use thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014192502A Division JP5963823B2 (ja) | 2008-10-17 | 2014-09-22 | S1p受容体モジュレーターおよびそれらの使用 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2012505836A JP2012505836A (ja) | 2012-03-08 |
| JP2012505836A5 true JP2012505836A5 (en:Method) | 2013-02-07 |
Family
ID=42106136
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011531305A Pending JP2012505836A (ja) | 2008-10-17 | 2009-10-19 | S1p受容体モジュレーターおよびそれらの使用 |
| JP2014192502A Active JP5963823B2 (ja) | 2008-10-17 | 2014-09-22 | S1p受容体モジュレーターおよびそれらの使用 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014192502A Active JP5963823B2 (ja) | 2008-10-17 | 2014-09-22 | S1p受容体モジュレーターおよびそれらの使用 |
Country Status (9)
| Country | Link |
|---|---|
| US (3) | US8592399B2 (en:Method) |
| EP (1) | EP2344484B1 (en:Method) |
| JP (2) | JP2012505836A (en:Method) |
| CN (1) | CN102186845B (en:Method) |
| AU (1) | AU2009304598B2 (en:Method) |
| CA (1) | CA2740484C (en:Method) |
| ES (1) | ES2590904T3 (en:Method) |
| NZ (1) | NZ592748A (en:Method) |
| WO (1) | WO2010043000A1 (en:Method) |
Families Citing this family (39)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2010043000A1 (en) | 2008-10-17 | 2010-04-22 | Akaal Pharma Pty Ltd | S1p receptors modulators and their use thereof |
| AU2009304596A1 (en) | 2008-10-17 | 2010-04-22 | Akaal Pharma Pty Ltd | S1P receptors modulators |
| AU2010213794A1 (en) * | 2009-02-10 | 2011-09-01 | Abbott Laboratories | Agonists and antagonists of the S1P5 receptor, and methods of uses thereof |
| EA023283B1 (ru) * | 2010-11-30 | 2016-05-31 | Адэссо Эдванст Материалс Уси Ко., Лтд. | Новые вещества для повторно перерабатываемых эпоксидных смол |
| AU2012242807A1 (en) | 2011-04-14 | 2013-11-07 | Allergan, Inc. | Phenyl bicyclic methyl azetidine derivatives as sphingosine-1 phosphate receptors modulators |
| CN102993027B (zh) * | 2011-09-08 | 2014-08-13 | 中化蓝天集团有限公司 | 4-氟-n-异丙基苯胺的定向单烷基化制备方法 |
| US8895753B2 (en) | 2011-12-23 | 2014-11-25 | Meiji Seika Pharma Co., Ltd. | S1P receptor modulating agent |
| JP6030752B2 (ja) | 2012-05-09 | 2016-11-24 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | オキセタン−3−イルメタンアミンの製造方法 |
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| US8859598B2 (en) * | 2012-10-04 | 2014-10-14 | Allergan, Inc. | 1, 2, 4-oxadiazoles azetidine derivatives as sphingosine-1 phosphate receptors modulators |
| WO2014063199A1 (en) * | 2012-10-26 | 2014-05-01 | Akaal Pharma Pty Ltd | Organic compounds |
| CN108047219A (zh) | 2012-11-07 | 2018-05-18 | 内尔维阿诺医学科学有限公司 | 取代的嘧啶基和吡啶基吡咯并吡啶酮类、其制备方法及其作为激酶抑制剂的用途 |
| US8735433B1 (en) * | 2012-11-14 | 2014-05-27 | Allergan, Inc. | Aryl oxadiazole derivatives as sphingosine 1-phosphate (S1P) receptor modulators |
| CN103304503B (zh) * | 2013-06-02 | 2015-03-04 | 张远强 | 抗糖尿病化合物、其制备方法和用途 |
| CN103304499B (zh) * | 2013-06-02 | 2015-03-04 | 张远强 | 抗糖尿病化合物、其制备方法和用途 |
| US20150051186A1 (en) * | 2013-08-15 | 2015-02-19 | Allergan, Inc. | Aryl azetidine derivatives as sphingosine-1 phosphate receptors modulators |
| US9718771B2 (en) | 2014-02-28 | 2017-08-01 | Kissei Pharmaceutical Co., Ltd. | Aniline derivative, pharmaceutical composition containing same, and use thereof |
| KR20170124602A (ko) | 2015-03-13 | 2017-11-10 | 포르마 세라퓨틱스 인크. | Hdac8 억제제로서의 알파-신나미드 화합물 및 조성물 |
| US20180228778A1 (en) * | 2015-08-11 | 2018-08-16 | Akaal Pharma Pty Ltd | Compositions comprising s1p receptor modulators |
| CN108884049A (zh) | 2016-02-09 | 2018-11-23 | 法玛克亚公司 | 喹啉酮赖氨酰氧化酶样2抑制剂及其用途 |
| WO2018118791A2 (en) | 2016-12-20 | 2018-06-28 | Oligomerix, Inc. | Novel quinazolinones that inhibit the formation of tau oligomers and their method of use |
| US11306075B2 (en) | 2016-12-20 | 2022-04-19 | Oligomerix, Inc. | Benzofuran, benzothiophene, and indole analogs that inhibit the formation of tau oligomers and their method of use |
| IL271149B2 (en) | 2017-06-14 | 2024-05-01 | Trevena Inc | Compounds for modulating s1p1 activity and methods of using the same |
| KR102017324B1 (ko) * | 2018-04-30 | 2019-09-02 | 경북대학교 산학협력단 | 신규한 asm 활성 직접 억제 화합물 2-아미노-2-(1,2,3-트리아졸-4-일)프로판-1,3-디올 유도체 및 이의 용도 |
| WO2020077014A1 (en) | 2018-10-09 | 2020-04-16 | Duke University | Compositions and methods for adjuvant cancer therapeutics |
| CN111630029B (zh) * | 2018-12-06 | 2021-04-30 | 上海济煜医药科技有限公司 | 作为免疫调节剂的化合物及其制备方法和应用 |
| CN109824685B (zh) * | 2019-04-03 | 2021-03-23 | 辽宁中医药大学 | 马齿苋中化合物oleracone G及其提取分离方法与应用 |
| JP2022547079A (ja) * | 2019-09-05 | 2022-11-10 | トレベナ・インコーポレイテッド | てんかんを治療する方法を使用しててんかんを治療する方法 |
| US11884655B2 (en) | 2019-11-19 | 2024-01-30 | Trevena, Inc. | Compounds and methods of preparing compounds S1P1 modulators |
| JP2023515612A (ja) * | 2020-02-28 | 2023-04-13 | アカール・ファーマ・プロプライエタリー・リミテッド | S1p受容体調節物質 |
| US12036286B2 (en) | 2021-03-18 | 2024-07-16 | Seagen Inc. | Selective drug release from internalized conjugates of biologically active compounds |
| TW202430031A (zh) | 2022-09-30 | 2024-08-01 | 瑞士商先正達農作物保護股份公司 | 殺微生物之吡唑衍生物 |
| TW202430514A (zh) | 2022-09-30 | 2024-08-01 | 瑞士商先正達農作物保護股份公司 | 殺微生物之吡唑衍生物 |
| EP4626882A1 (en) | 2022-11-30 | 2025-10-08 | Syngenta Crop Protection AG | Microbiocidal tetrahydroisoquinoline derivatives |
| WO2025114167A1 (en) | 2023-11-28 | 2025-06-05 | Syngenta Crop Protection Ag | Microbiocidal pyrazole derivatives |
| WO2025191053A1 (en) | 2024-03-14 | 2025-09-18 | Syngenta Crop Protection Ag | Microbiocidal pyrazole derivatives |
| WO2025210096A1 (en) | 2024-04-03 | 2025-10-09 | Syngenta Crop Protection Ag | Fungicidal compositions |
| WO2025210095A1 (en) | 2024-04-03 | 2025-10-09 | Syngenta Crop Protection Ag | Microbiocidal tetrahydroisoquinoline compounds |
| CN118878551A (zh) * | 2024-07-08 | 2024-11-01 | 安徽大学 | 一种4-溴噻吩并[2,3-c]吡啶-2-羧酸乙酯的制备方法 |
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| US6221865B1 (en) | 1995-11-06 | 2001-04-24 | University Of Pittsburgh | Inhibitors of protein isoprenyl transferases |
| FR2741876B1 (fr) | 1995-12-01 | 1998-01-09 | Cird Galderma | Composes biaromatiques portant un groupement adamantyl en para, compositions pharmaceutiques et cosmetiques les contenant et utilisations |
| JPH10158192A (ja) * | 1996-10-03 | 1998-06-16 | Eisai Co Ltd | 移植片対宿主疾患(gvhd)の治療および臓器移植時の移植片拒絶反応抑制のための医薬組成物 |
| US6228868B1 (en) | 1998-07-27 | 2001-05-08 | Abbott Laboratories | Oxazoline antiproliferative agents |
| KR20010081117A (ko) | 1998-12-18 | 2001-08-27 | 추후기재 | 신규한 바이사이클릭 화합물 |
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| US20040106794A1 (en) * | 2001-04-16 | 2004-06-03 | Schering Corporation | 3,4-Di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands |
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| ES2754221T3 (es) | 2003-08-29 | 2020-04-16 | Ono Pharmaceutical Co | Compuesto capaz de unirse al receptor de S1P y uso farmacéutico del mismo |
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| AU2009304596A1 (en) | 2008-10-17 | 2010-04-22 | Akaal Pharma Pty Ltd | S1P receptors modulators |
| WO2010043000A1 (en) | 2008-10-17 | 2010-04-22 | Akaal Pharma Pty Ltd | S1p receptors modulators and their use thereof |
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| WO2014063199A1 (en) * | 2012-10-26 | 2014-05-01 | Akaal Pharma Pty Ltd | Organic compounds |
-
2009
- 2009-10-19 WO PCT/AU2009/001371 patent/WO2010043000A1/en not_active Ceased
- 2009-10-19 EP EP09820119.7A patent/EP2344484B1/en active Active
- 2009-10-19 CA CA2740484A patent/CA2740484C/en active Active
- 2009-10-19 CN CN200980141188.9A patent/CN102186845B/zh active Active
- 2009-10-19 JP JP2011531305A patent/JP2012505836A/ja active Pending
- 2009-10-19 ES ES09820119.7T patent/ES2590904T3/es active Active
- 2009-10-19 NZ NZ592748A patent/NZ592748A/xx unknown
- 2009-10-19 US US13/124,549 patent/US8592399B2/en active Active
- 2009-10-19 AU AU2009304598A patent/AU2009304598B2/en active Active
-
2013
- 2013-10-29 US US14/066,276 patent/US9193716B2/en active Active
-
2014
- 2014-09-22 JP JP2014192502A patent/JP5963823B2/ja active Active
-
2015
- 2015-10-22 US US14/920,780 patent/US9707205B2/en active Active
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