JP2011500819A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2011500819A5 JP2011500819A5 JP2010531141A JP2010531141A JP2011500819A5 JP 2011500819 A5 JP2011500819 A5 JP 2011500819A5 JP 2010531141 A JP2010531141 A JP 2010531141A JP 2010531141 A JP2010531141 A JP 2010531141A JP 2011500819 A5 JP2011500819 A5 JP 2011500819A5
- Authority
- JP
- Japan
- Prior art keywords
- formulation
- disease
- diseases
- compound
- subject
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 238000009472 formulation Methods 0.000 claims 12
- 239000000203 mixture Substances 0.000 claims 12
- 201000010099 disease Diseases 0.000 claims 11
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 claims 11
- 150000001875 compounds Chemical class 0.000 claims 7
- 208000024827 Alzheimer disease Diseases 0.000 claims 4
- 208000018737 Parkinson disease Diseases 0.000 claims 3
- 102000007471 Adenosine A2A receptor Human genes 0.000 claims 2
- 108010085277 Adenosine A2A receptor Proteins 0.000 claims 2
- 208000011990 Corticobasal Degeneration Diseases 0.000 claims 2
- 208000023105 Huntington disease Diseases 0.000 claims 2
- 208000016285 Movement disease Diseases 0.000 claims 2
- 208000001089 Multiple system atrophy Diseases 0.000 claims 2
- 208000012902 Nervous system disease Diseases 0.000 claims 2
- 208000025966 Neurological disease Diseases 0.000 claims 2
- 206010039966 Senile dementia Diseases 0.000 claims 2
- 239000004480 active ingredient Substances 0.000 claims 2
- 230000003042 antagnostic effect Effects 0.000 claims 2
- 208000019901 Anxiety disease Diseases 0.000 claims 1
- 208000006096 Attention Deficit Disorder with Hyperactivity Diseases 0.000 claims 1
- 208000036864 Attention deficit/hyperactivity disease Diseases 0.000 claims 1
- 206010012335 Dependence Diseases 0.000 claims 1
- 230000001668 ameliorated effect Effects 0.000 claims 1
- 230000036506 anxiety Effects 0.000 claims 1
- 239000003937 drug carrier Substances 0.000 claims 1
- 239000008194 pharmaceutical composition Substances 0.000 claims 1
- 239000000825 pharmaceutical preparation Substances 0.000 claims 1
- 230000003449 preventive effect Effects 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
- 239000012453 solvate Substances 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US98224707P | 2007-10-24 | 2007-10-24 | |
| PCT/US2008/080256 WO2009055308A1 (en) | 2007-10-24 | 2008-10-17 | Arylindenopyrimidines and their use as adenosine a2a receptor antagonists |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2011500819A JP2011500819A (ja) | 2011-01-06 |
| JP2011500819A5 true JP2011500819A5 (enExample) | 2012-12-20 |
Family
ID=40091927
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010531141A Withdrawn JP2011500819A (ja) | 2007-10-24 | 2008-10-17 | アリルインデノピリミジン及びアデノシンＡ２ａ受容体拮抗物質としてのそれらの使用 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US8017614B2 (enExample) |
| EP (1) | EP2217575A1 (enExample) |
| JP (1) | JP2011500819A (enExample) |
| CN (1) | CN101835759A (enExample) |
| AR (1) | AR069009A1 (enExample) |
| AU (1) | AU2008317034A1 (enExample) |
| CL (1) | CL2008003131A1 (enExample) |
| PA (1) | PA8801501A1 (enExample) |
| PE (1) | PE20091344A1 (enExample) |
| TW (1) | TW200934493A (enExample) |
| UY (1) | UY31420A1 (enExample) |
| WO (1) | WO2009055308A1 (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20110105540A1 (en) * | 2009-10-29 | 2011-05-05 | Jackson Paul F | 2-AMINO-9-[4-(4-METHOXY-PHENOXY)-PIPERIDIN-1-YL]-4-PHENYL-INDENO[1,2-D]PYRIMIDIN-5-ONE AND ITS USE AS A HIGHLY SELECTIVE ADENOSINE A2a RECEPTOR ANTAGONIST |
| US9238643B2 (en) | 2010-09-06 | 2016-01-19 | Guangzhou Institutes Of Biomedicine And Health, Chinese Academy Of Sciences | Amide compounds |
| AU2013251079B2 (en) | 2012-04-20 | 2017-03-23 | Ucb Pharma S.A. | Methods for treating Parkinson's disease |
| JOP20210164A1 (ar) | 2019-01-11 | 2023-01-30 | Omeros Corp | طرق وتركيبات علاج السرطان |
| AU2023252914A1 (en) | 2022-04-13 | 2024-10-17 | Arcus Biosciences, Inc. | Combination therapy for treating trop-2 expressing cancers |
| WO2025137640A1 (en) | 2023-12-22 | 2025-06-26 | Gilead Sciences, Inc. | Azaspiro wrn inhibitors |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20040127510A1 (en) | 2002-04-16 | 2004-07-01 | Heintzelman Geoffrey R. | Arylindenopyridines and arylindenopyrimidines and related therapeutic and prophylactic methods |
| AU2003275430A1 (en) | 2003-10-03 | 2005-05-19 | Ortho-Mcneil Pharmaceutical, Inc. | Arylindenopyridines and arylindenopyridines and their use as adenosine a2a receptor antagonist |
-
2008
- 2008-10-17 US US12/253,358 patent/US8017614B2/en not_active Expired - Fee Related
- 2008-10-17 AU AU2008317034A patent/AU2008317034A1/en not_active Abandoned
- 2008-10-17 WO PCT/US2008/080256 patent/WO2009055308A1/en not_active Ceased
- 2008-10-17 JP JP2010531141A patent/JP2011500819A/ja not_active Withdrawn
- 2008-10-17 CN CN200880112882A patent/CN101835759A/zh active Pending
- 2008-10-17 EP EP08841238A patent/EP2217575A1/en not_active Withdrawn
- 2008-10-23 PA PA20088801501A patent/PA8801501A1/es unknown
- 2008-10-23 AR ARP080104625A patent/AR069009A1/es not_active Application Discontinuation
- 2008-10-23 CL CL2008003131A patent/CL2008003131A1/es unknown
- 2008-10-23 TW TW097140560A patent/TW200934493A/zh unknown
- 2008-10-23 PE PE2008001819A patent/PE20091344A1/es not_active Application Discontinuation
- 2008-10-24 UY UY31420A patent/UY31420A1/es unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CA3094580C (en) | Oral formulations of cytidine analogs and methods of use thereof | |
| MX354423B (es) | Formulaciones de rasagilina de liberación prolongada y usos de las mismas. | |
| TW200829244A (en) | Therapeutic combinations 482 | |
| JP2011500819A5 (enExample) | ||
| JP2019503365A5 (enExample) | ||
| US20230250076A1 (en) | Processes and intermediate for the large-scale preparation of 2,4,6-trifluoro-n-[6-(1-methyl-piperidine-4-carbonyl)-pyridin-2-yl]-benzamide hemisuccinate, and preparation of 2,4,6-trifluoro-n-[6-(1-methyl-piperidine-4-carbonyl)-pyridin-2-yl]-benzamide acetate | |
| JP2015514135A5 (enExample) | ||
| JP2019510039A5 (enExample) | ||
| JP2014517050A5 (enExample) | ||
| US20190117658A1 (en) | Novel compositions and methods | |
| JP2005537268A5 (enExample) | ||
| JP2015509972A5 (enExample) | ||
| JP2012508734A5 (enExample) | ||
| JP2016534063A5 (enExample) | ||
| JP2007533687A (ja) | 月経前の及び他の女性の性的障害の治療におけるフリバンセリンの使用 | |
| MX2011010732A (es) | Pirimidinas sustituidas por imidazol utiles en el tratamiento de trastornos relacionados con glucogeno sintasa cinasa 3 como la enfermedad de alzheimer. | |
| TWI804687B (zh) | 慢性咳嗽治療用醫藥 | |
| TWI377204B (en) | Arylvinylazacycloalkane compounds and methods of preparation and use thereof | |
| MX2009010165A (es) | Nuevas imidazo[4,5-b]piridina-7-carboxamidas 704. | |
| SI3029039T1 (en) | Pharmaceutical formulations containing crystalline forms of (R) -7-chloro-N- (quinuclidin-3-yl) benzo (b) thiophene-2-carboxamide hydrochloride monohydrate | |
| US20250236589A1 (en) | Therapeutic phenethylamine compositions and methods of use | |
| JP2011516588A5 (enExample) | ||
| CA3102762A1 (en) | Eaat2 activators and methods of using thereof | |
| CN116940362A (zh) | 在慢性ssri方案后使用苯二氮䓬增加对裸盖菇素的敏感性 | |
| JP2010500284A5 (enExample) |