|
FR2713225B1
(fr)
|
1993-12-02 |
1996-03-01 |
Sanofi Sa |
N-pipéridino-3-pyrazolecarboxamide substitué.
|
|
FR2692575B1
(fr)
|
1992-06-23 |
1995-06-30 |
Sanofi Elf |
Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
|
|
US6100042A
(en)
|
1993-03-31 |
2000-08-08 |
Cadus Pharmaceutical Corporation |
Yeast cells engineered to produce pheromone system protein surrogates, and uses therefor
|
|
GB9719496D0
(en)
|
1997-09-13 |
1997-11-19 |
Glaxo Group Ltd |
G protien chimeras
|
|
WO2000012704A2
(en)
|
1998-09-01 |
2000-03-09 |
Basf Aktiengesellschaft |
Enhanced functional expression of g protein-coupled receptors
|
|
US6221660B1
(en)
|
1999-02-22 |
2001-04-24 |
Synaptic Pharmaceutical Corporation |
DNA encoding SNORF25 receptor
|
|
US20040229911A1
(en)
*
|
2000-05-17 |
2004-11-18 |
Pfizer Inc |
New pharmaceutical combinations for NOS inhibitors
|
|
FR2829028B1
(fr)
|
2001-08-29 |
2004-12-17 |
Aventis Pharma Sa |
Association d'un antagoniste du recepteur cb1 et d'un produit qui active la neurotransmission dopaminergique dans le cerveau, les compositions pharmaceutiques les contenant et leur utilisation pour le traitement de la maladie de
|
|
FR2829027A1
(fr)
|
2001-08-29 |
2003-03-07 |
Aventis Pharma Sa |
Association avec un antagoniste du recepteur cb1, les compositions pharmaceutiques les contenant et leur utilisation pour le traitement de la maladie de parkinson
|
|
EP1421077A4
(en)
|
2001-08-31 |
2004-11-17 |
Univ Connecticut |
NEW PYRAZOLANALOGS ON CANNABINOID RECEPTORS
|
|
TWI231757B
(en)
|
2001-09-21 |
2005-05-01 |
Solvay Pharm Bv |
1H-Imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1-antagonistic activity
|
|
ES2272809T3
(es)
|
2001-09-21 |
2007-05-01 |
Solvay Pharm Bv |
Nuevos derivados de 4,5-dihidro-1h-pirazol con actividad antagonista de cb1.
|
|
AU2002333853B2
(en)
|
2001-09-21 |
2006-07-13 |
Solvay Pharmaceuticals B.V. |
4,5-dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activity
|
|
FR2831883B1
(fr)
|
2001-11-08 |
2004-07-23 |
Sanofi Synthelabo |
Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant
|
|
SE0104330D0
(sv)
|
2001-12-19 |
2001-12-19 |
Astrazeneca Ab |
Therapeutic agents
|
|
SE0104332D0
(sv)
|
2001-12-19 |
2001-12-19 |
Astrazeneca Ab |
Therapeutic agents
|
|
FR2833842B1
(fr)
|
2001-12-21 |
2004-02-13 |
Aventis Pharma Sa |
Compositions pharmaceutiques a base de derives d'azetidine
|
|
AU2003209388A1
(en)
|
2002-01-29 |
2003-09-02 |
Merck And Co., Inc. |
Substituted imidazoles as cannabinoid receptor modulators
|
|
WO2003075660A1
(en)
|
2002-03-06 |
2003-09-18 |
Merck & Co., Inc. |
Method of treatment or prevention of obesity
|
|
WO2003077847A2
(en)
|
2002-03-12 |
2003-09-25 |
Merck & Co., Inc. |
Substituted amides
|
|
TW200800167A
(en)
*
|
2002-03-15 |
2008-01-01 |
Novartis Ag |
Organic compounds
|
|
AR038966A1
(es)
|
2002-03-18 |
2005-02-02 |
Solvay Pharm Bv |
Derivados de tiazol que tienen actividad antagonista, agonista o agonista parcial de cb1
|
|
EP1490043A4
(en)
|
2002-03-26 |
2007-05-30 |
Merck & Co Inc |
SPIROCYCLIC AMIDS AS CANNABINOID RECEPTOR MODULATORS
|
|
ES2192494B1
(es)
|
2002-03-27 |
2005-02-16 |
Consejo Superior De Investigaciones Cientificas |
Derivados de 1,2,4-triazol con propiedades cannabinoides.
|
|
WO2003082191A2
(en)
|
2002-03-28 |
2003-10-09 |
Merck & Co., Inc. |
Substituted 2,3-diphenyl pyridines
|
|
JP2005527586A
(ja)
|
2002-04-05 |
2005-09-15 |
メルク エンド カムパニー インコーポレーテッド |
置換アリールアミド
|
|
FR2838438A1
(fr)
|
2002-04-11 |
2003-10-17 |
Sanofi Synthelabo |
Derives de diphenylpyridine,leur preparation, les compositions pharmaceutiques en contenant
|
|
FR2838439B1
(fr)
|
2002-04-11 |
2005-05-20 |
Sanofi Synthelabo |
Derives de terphenyle, leur preparation, les compositions pharmaceutqiues en contenant
|
|
US7667053B2
(en)
|
2002-04-12 |
2010-02-23 |
Merck & Co., Inc. |
Bicyclic amides
|
|
US6825209B2
(en)
|
2002-04-15 |
2004-11-30 |
Research Triangle Institute |
Compounds having unique CB1 receptor binding selectivity and methods for their production and use
|
|
CA2493313C
(en)
|
2002-07-29 |
2010-03-09 |
F. Hoffmann-La Roche Ag |
Novel benzodioxoles
|
|
WO2004012671A2
(en)
|
2002-08-02 |
2004-02-12 |
Merck & Co., Inc. |
Substituted furo [2,3-b] pyridine derivatives
|
|
US20050101542A1
(en)
|
2002-08-20 |
2005-05-12 |
Regents Of The University Of California |
Combination therapy for controlling appetites
|
|
HRP20050053A2
(en)
|
2002-09-19 |
2005-04-30 |
Solvay Pharmaceuticals B.V. |
1 h-1,2,4-triazole-3-carboxamide derivatives as cannabinoid-cb1 receptor ligands
|
|
US7405221B2
(en)
|
2002-09-27 |
2008-07-29 |
Merck & Co., Inc. |
Substituted pyrimidines
|
|
EP1556373A1
(en)
|
2002-10-18 |
2005-07-27 |
Pfizer Products Inc. |
Cannabinoid receptor ligands and uses thereof
|
|
US7129239B2
(en)
|
2002-10-28 |
2006-10-31 |
Pfizer Inc. |
Purine compounds and uses thereof
|
|
US7247628B2
(en)
|
2002-12-12 |
2007-07-24 |
Pfizer, Inc. |
Cannabinoid receptor ligands and uses thereof
|
|
AU2003300967B2
(en)
|
2002-12-19 |
2009-05-28 |
Merck Sharp & Dohme Corp. |
Substituted amides
|
|
GB0230087D0
(en)
|
2002-12-24 |
2003-01-29 |
Astrazeneca Ab |
Therapeutic agents
|
|
CN100360527C
(zh)
|
2003-01-02 |
2008-01-09 |
霍夫曼-拉罗奇有限公司 |
Cb1受体反激动剂
|
|
TW200413328A
(en)
|
2003-01-02 |
2004-08-01 |
Hoffmann La Roche |
Novel CB 1 receptor inverse agonists
|
|
US7329658B2
(en)
|
2003-02-06 |
2008-02-12 |
Pfizer Inc |
Cannabinoid receptor ligands and uses thereof
|
|
JP2006517550A
(ja)
|
2003-02-13 |
2006-07-27 |
サノフィ−アベンティス・ドイチュラント・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング |
置換ヘキサヒドロピラジノ[1,2−a]ピリミジン−4,7−ジオン誘導体、その製造方法および医薬としてのその使用
|
|
RS20050572A
(sr)
|
2003-02-13 |
2007-09-21 |
Sanofi-Aventis Deutschland Gmbh., |
AZOTOM SUPSTITUISANI HEKSAHIDRO- PIRAZINO(1,2-A)PIRIMIDIN -4,7-DION DERIVATI, POSTUPAK ZA NjIHOVU PROIZVODNjU I NjIHOVA PRIMENA KAO LEKA
|
|
EP1606019A1
(en)
|
2003-03-07 |
2005-12-21 |
The University Court of The University of Aberdeen |
Cannabinoid receptor inverse agonists and neutral antagonists as therapeutic agents for the treatment of bone disorders
|
|
US7232823B2
(en)
|
2003-06-09 |
2007-06-19 |
Pfizer, Inc. |
Cannabinoid receptor ligands and uses thereof
|
|
EP1711491A1
(en)
|
2003-12-24 |
2006-10-18 |
Prosidion Limited |
Heterocyclic derivatives as gpcr receptor agonists
|
|
BRPI0516407A
(pt)
|
2004-12-24 |
2008-09-02 |
Prosidion Ltd |
agonistas de receptor acoplado à proteìna g (gpr116) e uso destes para o tratamento de obesidade e diabetes
|
|
WO2006067532A1
(en)
|
2004-12-24 |
2006-06-29 |
Prosidion Ltd |
G-protein coupled receptor agonists
|
|
GB0428514D0
(en)
|
2004-12-31 |
2005-02-09 |
Prosidion Ltd |
Compounds
|
|
CA2613236A1
(en)
|
2005-06-30 |
2007-01-11 |
Prosidion Limited |
G-protein coupled receptor agonists
|
|
MX2007016508A
(es)
|
2005-06-30 |
2008-03-04 |
Prosidion Ltd |
Agonistas del receptor acoplado a la proteina g.
|
|
WO2007003961A2
(en)
|
2005-06-30 |
2007-01-11 |
Prosidion Limited |
Gpcr agonists
|
|
EP1907383A1
(en)
|
2005-06-30 |
2008-04-09 |
Prosidion Limited |
Gpcr agonists
|
|
WO2007116229A1
(en)
|
2006-04-06 |
2007-10-18 |
Prosidion Limited |
Heterocyclic gpcr agonists
|
|
GB0607196D0
(en)
*
|
2006-04-11 |
2006-05-17 |
Prosidion Ltd |
G-protein coupled receptor agonists
|