JP2010523556A5 - - Google Patents

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Publication number
JP2010523556A5
JP2010523556A5 JP2010502052A JP2010502052A JP2010523556A5 JP 2010523556 A5 JP2010523556 A5 JP 2010523556A5 JP 2010502052 A JP2010502052 A JP 2010502052A JP 2010502052 A JP2010502052 A JP 2010502052A JP 2010523556 A5 JP2010523556 A5 JP 2010523556A5
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JP
Japan
Prior art keywords
pyrido
indole
tetrahydro
methyl
pyridin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2010502052A
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English (en)
Japanese (ja)
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JP2010523556A (ja
JP5580731B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/RU2008/000196 external-priority patent/WO2008123796A2/ru
Publication of JP2010523556A publication Critical patent/JP2010523556A/ja
Publication of JP2010523556A5 publication Critical patent/JP2010523556A5/ja
Application granted granted Critical
Publication of JP5580731B2 publication Critical patent/JP5580731B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2010502052A 2007-04-05 2008-04-01 置換された２，３，４，５−テトラヒドロ−１ｈ−ピリド［４，３−ｂ］インドール、その製造のための方法及び使用 Expired - Fee Related JP5580731B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
RU2007112666A RU2334747C3 (ru) 2007-04-05 ЗАМЕЩЕННЫЕ 2,3,4,5-ТЕТРАГИДРО-1Н-ПИРИДО[4,3-b]ИНДОЛЫ, СПОСОБ ИХ ПОЛУЧЕНИЯ И ПРИМЕНЕНИЯ
RU2007112666 2007-05-04
PCT/RU2008/000196 WO2008123796A2 (ru) 2007-04-05 2008-04-01 Замещенные 2,3,4,5-tetpaгидpo-1h-пиpидo[4,3-b]иhдoлы, способ их получения и применения

Publications (3)

Publication Number Publication Date
JP2010523556A JP2010523556A (ja) 2010-07-15
JP2010523556A5 true JP2010523556A5 (enExample) 2011-05-19
JP5580731B2 JP5580731B2 (ja) 2014-08-27

Family

ID=39831503

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010502052A Expired - Fee Related JP5580731B2 (ja) 2007-04-05 2008-04-01 置換された２，３，４，５−テトラヒドロ−１ｈ−ピリド［４，３−ｂ］インドール、その製造のための方法及び使用

Country Status (9)

Country Link
US (3) US8541437B2 (enExample)
EP (1) EP2145887B1 (enExample)
JP (1) JP5580731B2 (enExample)
KR (1) KR20090130105A (enExample)
AU (1) AU2008236872B2 (enExample)
CA (1) CA2683453C (enExample)
EA (1) EA016234B1 (enExample)
UA (1) UA98324C2 (enExample)
WO (1) WO2008123796A2 (enExample)

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RU2544856C2 (ru) 2008-01-25 2015-03-20 Сергей Олегович Бачурин НОВЫЕ ПРОИЗВОДНЫЕ 2,3,4,5-ТЕТРАГИДРО-1-ПИРИДО[4,3-b]ИНДОЛА И СПОСОБЫ ИХ ПРИМЕНЕНИЯ
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JP2013504580A (ja) * 2009-09-11 2013-02-07 スノヴィオン ファーマシューティカルズ インコーポレイテッド ヒスタミンｈ３インバースアゴニストおよびアンタゴニストとその使用方法
CN102711466A (zh) 2009-09-23 2012-10-03 梅迪维新技术公司 桥连杂环化合物及其使用方法
WO2011038161A1 (en) 2009-09-23 2011-03-31 Medivation Technologies, Inc. Pyrido[4,3-b]indoles and methods of use
AU2010298168B2 (en) 2009-09-23 2015-11-19 Medivation Technologies, Inc. Pyrido(3,4-b)indoles and methods of use
EP2480079A4 (en) * 2009-09-23 2015-04-08 Medivation Technologies Inc PYRIDO- (3,4-B-) INDOLE AND USE METHOD THEREFOR
US9193728B2 (en) 2010-02-18 2015-11-24 Medivation Technologies, Inc. Fused tetracyclic pyrido [4,3-B] indole and pyrido [3,4-B] indole derivatives and methods of use
US9040519B2 (en) 2010-02-18 2015-05-26 Medivation Technologies, Inc. Fused tetracyclic pyrido [4,3-B] indole and pyrido [3,4-B] indole derivatives and methods of use
US9034865B2 (en) 2010-02-18 2015-05-19 Medivation Technologies, Inc. Pyrido [4,3-B] indole and pyrido [3,4-B] indole derivatives and methods of use
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WO2011103448A1 (en) * 2010-02-19 2011-08-25 Medivation Technologies, Inc. Methods and compositions for treating psychotic disorders using antipsychotic combination therapy
WO2012112965A1 (en) 2011-02-18 2012-08-23 Medivation Technologies, Inc. Compounds and methods of treating diabetes
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UA118010C2 (uk) 2011-08-01 2018-11-12 Вертекс Фармасьютікалз Інкорпорейтед Інгібітори реплікації вірусів грипу
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WO2015070237A1 (en) 2013-11-11 2015-05-14 Board Of Regents Of The University Of Texas System Neuroprotective chemicals and methods for identifying and using same
EP3068388A4 (en) 2013-11-11 2017-04-12 Board of Regents of the University of Texas System Neuroprotective compounds and use thereof
HUE038820T2 (hu) 2013-11-13 2018-11-28 Vertex Pharma Eljárás influenzavírusok replikációjának inhibitorai elõállítására
PT3068776T (pt) 2013-11-13 2019-08-26 Vertex Pharma Inibidores da replicação de vírus da gripe
EP3294717B1 (en) 2015-05-13 2020-07-29 Vertex Pharmaceuticals Inc. Methods of preparing inhibitors of influenza viruses replication
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