JP2010509356A5 - - Google Patents

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Publication number
JP2010509356A5
JP2010509356A5 JP2009536454A JP2009536454A JP2010509356A5 JP 2010509356 A5 JP2010509356 A5 JP 2010509356A5 JP 2009536454 A JP2009536454 A JP 2009536454A JP 2009536454 A JP2009536454 A JP 2009536454A JP 2010509356 A5 JP2010509356 A5 JP 2010509356A5
Authority
JP
Japan
Prior art keywords
pyrrolo
pyridin
substituted
phenyl
benzamide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2009536454A
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English (en)
Japanese (ja)
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JP2010509356A (ja
JP5244118B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2007/083850 external-priority patent/WO2008060907A2/en
Publication of JP2010509356A publication Critical patent/JP2010509356A/ja
Publication of JP2010509356A5 publication Critical patent/JP2010509356A5/ja
Application granted granted Critical
Publication of JP5244118B2 publication Critical patent/JP5244118B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009536454A 2006-11-10 2007-11-07 新規キナーゼ阻害剤 Expired - Fee Related JP5244118B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US86518106P 2006-11-10 2006-11-10
US60/865,181 2006-11-10
PCT/US2007/083850 WO2008060907A2 (en) 2006-11-10 2007-11-07 Pyrrolo-pyridine kinase inhibitors

Publications (3)

Publication Number Publication Date
JP2010509356A JP2010509356A (ja) 2010-03-25
JP2010509356A5 true JP2010509356A5 (enExample) 2010-10-21
JP5244118B2 JP5244118B2 (ja) 2013-07-24

Family

ID=39261598

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009536454A Expired - Fee Related JP5244118B2 (ja) 2006-11-10 2007-11-07 新規キナーゼ阻害剤

Country Status (6)

Country Link
US (1) US8148361B2 (enExample)
EP (1) EP2081928B1 (enExample)
JP (1) JP5244118B2 (enExample)
CN (1) CN101600714B (enExample)
NO (1) NO20091708L (enExample)
WO (1) WO2008060907A2 (enExample)

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JP2016512815A (ja) 2013-03-15 2016-05-09 バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ Ａｔｒキナーゼの阻害剤として有用な縮合ピラゾロピリミジン誘導体
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HUE046727T2 (hu) 2013-12-06 2020-03-30 Vertex Pharma Az ATR-kináz inhibitoraként használható vegyület, 2-amino-6-fluoro-N-[5-fluoro-piridin-3-IL]-pirazolo-[1,5-A]-pirimidin-3-karboxamid, ennek elõállítása, különbözõ szilárd formái és ezek radioaktív nyomjelzett származékai
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MA41551A (fr) 2015-02-20 2017-12-26 Incyte Corp Hétérocycles bicycliques utilisés en tant qu'inhibiteurs de fgfr4
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US10478494B2 (en) 2015-04-03 2019-11-19 Astex Therapeutics Ltd FGFR/PD-1 combination therapy for the treatment of cancer
KR102678021B1 (ko) 2015-09-30 2024-06-26 버텍스 파마슈티칼스 인코포레이티드 Dna 손상제와 병용되는, atr 저해제를 포함하는 암 치료용 약제학적 조성물
PL3362449T3 (pl) 2015-10-13 2021-12-13 Institut National De La Santé Et De La Recherche Médicale (Inserm) Pochodne sybiriliny do zastosowania do zapobiegania i/lub leczenia zaburzeń związanych z nekroptozą komórkową
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JP2024522189A (ja) 2021-06-09 2024-06-11 インサイト・コーポレイション Ｆｇｆｒ阻害剤としての三環式ヘテロ環
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