JP2009544756A5 - - Google Patents

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Publication number
JP2009544756A5
JP2009544756A5 JP2009522952A JP2009522952A JP2009544756A5 JP 2009544756 A5 JP2009544756 A5 JP 2009544756A5 JP 2009522952 A JP2009522952 A JP 2009522952A JP 2009522952 A JP2009522952 A JP 2009522952A JP 2009544756 A5 JP2009544756 A5 JP 2009544756A5
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JP
Japan
Prior art keywords
formula
compound
disease
oxo
salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2009522952A
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English (en)
Japanese (ja)
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JP2009544756A (ja
JP5236643B2 (ja
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Publication date
Priority claimed from US11/782,742 external-priority patent/US7629351B2/en
Application filed filed Critical
Publication of JP2009544756A publication Critical patent/JP2009544756A/ja
Publication of JP2009544756A5 publication Critical patent/JP2009544756A5/ja
Application granted granted Critical
Publication of JP5236643B2 publication Critical patent/JP5236643B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009522952A 2006-07-28 2007-07-26 ケモカイン受容体活性のモジュレーター、結晶形および方法 Expired - Fee Related JP5236643B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US83423506P 2006-07-28 2006-07-28
US60/834,235 2006-07-28
US89602607P 2007-03-21 2007-03-21
US60/896,026 2007-03-21
US11/782,742 US7629351B2 (en) 2006-07-28 2007-07-25 N-((1R,2S,5R)-5-(tert-butylamino)-2-((S)-2-oxo-3-(6-(trifluoromethyl)quinazolin-4-ylamino) pyrrolidin-1-yl)cyclohexyl)acetamide and other modulators of chemokine receptor activity, crystalline forms and process
US11/782,742 2007-07-25
PCT/US2007/074377 WO2008014360A2 (en) 2006-07-28 2007-07-26 Modulators of chemokine receptor activity, crystalline forms and process

Publications (3)

Publication Number Publication Date
JP2009544756A JP2009544756A (ja) 2009-12-17
JP2009544756A5 true JP2009544756A5 (enExample) 2010-08-12
JP5236643B2 JP5236643B2 (ja) 2013-07-17

Family

ID=38829183

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009522952A Expired - Fee Related JP5236643B2 (ja) 2006-07-28 2007-07-26 ケモカイン受容体活性のモジュレーター、結晶形および方法

Country Status (26)

Country Link
US (2) US7629351B2 (enExample)
EP (2) EP2046779B1 (enExample)
JP (1) JP5236643B2 (enExample)
KR (1) KR20090033915A (enExample)
CN (1) CN101535301B (enExample)
AR (1) AR062124A1 (enExample)
AT (2) ATE509926T1 (enExample)
AU (1) AU2007279333B2 (enExample)
BR (1) BRPI0715415A2 (enExample)
CA (2) CA2659253A1 (enExample)
CY (1) CY1111744T1 (enExample)
DK (1) DK2046779T3 (enExample)
EA (1) EA016563B1 (enExample)
ES (1) ES2365264T3 (enExample)
HR (1) HRP20110465T1 (enExample)
IL (2) IL196427A (enExample)
MX (1) MX2009000808A (enExample)
NO (1) NO20090190L (enExample)
NZ (1) NZ574425A (enExample)
PE (1) PE20080732A1 (enExample)
PL (1) PL2046779T3 (enExample)
PT (1) PT2046779E (enExample)
SG (1) SG158924A1 (enExample)
SI (1) SI2046779T1 (enExample)
TW (2) TWI421249B (enExample)
WO (1) WO2008014360A2 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7687508B2 (en) * 2006-07-28 2010-03-30 Bristol-Myers Squibb Company Cyclic derivatives as modulators of chemokine receptor activity
US8383812B2 (en) * 2009-10-13 2013-02-26 Bristol-Myers Squibb Company N-((1R,2S,5R)-5-(tert-butylamino)-2-((S)-3-(7-tert-butylpyrazolo[1,5-A][1,3,5]triazin-4-ylamino)-2-oxopyrrolidin-1-yl)cyclohexyl)acetamide, a dual modulator of chemokine receptor activity, crystalline forms and processes
KR20120135716A (ko) * 2011-06-07 2012-12-17 한미사이언스 주식회사 이중대칭 구조의 퀴나졸린 유도체 화합물 및 이의 용도
EP2567959B1 (en) 2011-09-12 2014-04-16 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
US8669281B1 (en) 2013-03-14 2014-03-11 Alkermes Pharma Ireland Limited Prodrugs of fumarates and their use in treating various diseases
MA40320A (fr) * 2014-07-17 2017-05-24 Santen Pharmaceutical Co Ltd Agent prophylactique ou thérapeutique pour des troubles du segment postérieur de l'œil
BR112020000418A2 (pt) * 2017-07-20 2020-07-14 Bristol-Myers Squibb Company processo para a preparação de n-((1r,2s,5r)-5-(terc-butilamino)-2-((s)-3-(7-terc-butilpirazolo[1,5-a][1,3,5]triazin-4-ilamino)-2-oxopirrolidin-1-il) ciclo-hexil)acetamida
CN115677728A (zh) * 2022-11-02 2023-02-03 成都科岭源医药技术有限公司 一种海鞘素类化合物中间体的制备方法

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