MX2009000808A - Moduladores de la actividad del receptor de quimiocina, formas cristalinas y procesos. - Google Patents
Moduladores de la actividad del receptor de quimiocina, formas cristalinas y procesos.Info
- Publication number
- MX2009000808A MX2009000808A MX2009000808A MX2009000808A MX2009000808A MX 2009000808 A MX2009000808 A MX 2009000808A MX 2009000808 A MX2009000808 A MX 2009000808A MX 2009000808 A MX2009000808 A MX 2009000808A MX 2009000808 A MX2009000808 A MX 2009000808A
- Authority
- MX
- Mexico
- Prior art keywords
- compound
- formula
- oxo
- mcp
- tert
- Prior art date
Links
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Classifications
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- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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Landscapes
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Applications Claiming Priority (4)
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| US83423506P | 2006-07-28 | 2006-07-28 | |
| US89602607P | 2007-03-21 | 2007-03-21 | |
| US11/782,742 US7629351B2 (en) | 2006-07-28 | 2007-07-25 | N-((1R,2S,5R)-5-(tert-butylamino)-2-((S)-2-oxo-3-(6-(trifluoromethyl)quinazolin-4-ylamino) pyrrolidin-1-yl)cyclohexyl)acetamide and other modulators of chemokine receptor activity, crystalline forms and process |
| PCT/US2007/074377 WO2008014360A2 (en) | 2006-07-28 | 2007-07-26 | Modulators of chemokine receptor activity, crystalline forms and process |
Publications (1)
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| MX2009000808A true MX2009000808A (es) | 2009-01-29 |
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| MX2009000808A MX2009000808A (es) | 2006-07-28 | 2007-07-26 | Moduladores de la actividad del receptor de quimiocina, formas cristalinas y procesos. |
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| US7687508B2 (en) * | 2006-07-28 | 2010-03-30 | Bristol-Myers Squibb Company | Cyclic derivatives as modulators of chemokine receptor activity |
| US8383812B2 (en) | 2009-10-13 | 2013-02-26 | Bristol-Myers Squibb Company | N-((1R,2S,5R)-5-(tert-butylamino)-2-((S)-3-(7-tert-butylpyrazolo[1,5-A][1,3,5]triazin-4-ylamino)-2-oxopyrrolidin-1-yl)cyclohexyl)acetamide, a dual modulator of chemokine receptor activity, crystalline forms and processes |
| KR20120135716A (ko) * | 2011-06-07 | 2012-12-17 | 한미사이언스 주식회사 | 이중대칭 구조의 퀴나졸린 유도체 화합물 및 이의 용도 |
| EP2567959B1 (en) | 2011-09-12 | 2014-04-16 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
| US8669281B1 (en) | 2013-03-14 | 2014-03-11 | Alkermes Pharma Ireland Limited | Prodrugs of fumarates and their use in treating various diseases |
| MA40320A (fr) * | 2014-07-17 | 2017-05-24 | Santen Pharmaceutical Co Ltd | Agent prophylactique ou thérapeutique pour des troubles du segment postérieur de l'œil |
| HUE058049T2 (hu) | 2017-07-20 | 2022-06-28 | Bristol Myers Squibb Co | Eljárás N-((1R,2S,SR)-5-(terc-butilamino)-2-((S)-3-(7-terc-butilpirazolo[1,5-A][1,3,5] triazin-4-ilamino)-2-oxopirrolidin-1-il)ciklohexil)acetamid elõállítására |
| CN115677728A (zh) * | 2022-11-02 | 2023-02-03 | 成都科岭源医药技术有限公司 | 一种海鞘素类化合物中间体的制备方法 |
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