JP2009536161A - 医薬化合物 - Google Patents

医薬化合物 Download PDF

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Publication number
JP2009536161A
JP2009536161A JP2009507153A JP2009507153A JP2009536161A JP 2009536161 A JP2009536161 A JP 2009536161A JP 2009507153 A JP2009507153 A JP 2009507153A JP 2009507153 A JP2009507153 A JP 2009507153A JP 2009536161 A JP2009536161 A JP 2009536161A
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Prior art keywords
group
compound
use according
disease
groups
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JP2009507153A
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English (en)
Japanese (ja)
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JP2009536161A5 (https=
Inventor
トーマス、グランモア、デービス
ミシェル、ドーン、ガレット
ロバート、ジョージ、ボイル
イアン、コリンズ
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Cancer Research Technology Ltd
Astex Therapeutics Ltd
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Cancer Research Technology Ltd
Astex Therapeutics Ltd
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Priority claimed from GB0608185A external-priority patent/GB0608185D0/en
Priority claimed from GB0608175A external-priority patent/GB0608175D0/en
Application filed by Cancer Research Technology Ltd, Astex Therapeutics Ltd filed Critical Cancer Research Technology Ltd
Publication of JP2009536161A publication Critical patent/JP2009536161A/ja
Publication of JP2009536161A5 publication Critical patent/JP2009536161A5/ja
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    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Cardiology (AREA)
  • Communicable Diseases (AREA)
  • Immunology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Psychiatry (AREA)
  • Urology & Nephrology (AREA)
  • Molecular Biology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Psychology (AREA)
  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
JP2009507153A 2006-04-25 2007-04-25 医薬化合物 Withdrawn JP2009536161A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0608185A GB0608185D0 (en) 2006-04-25 2006-04-25 Pharmaceutical Compounds
GB0608175A GB0608175D0 (en) 2006-04-25 2006-04-25 Pharmaceutical Compounds
PCT/GB2007/001510 WO2007125315A2 (en) 2006-04-25 2007-04-25 Pharmaceutical compounds

Publications (2)

Publication Number Publication Date
JP2009536161A true JP2009536161A (ja) 2009-10-08
JP2009536161A5 JP2009536161A5 (https=) 2010-06-17

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ID=38543971

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JP2009507153A Withdrawn JP2009536161A (ja) 2006-04-25 2007-04-25 医薬化合物

Country Status (4)

Country Link
US (1) US20090253718A1 (https=)
EP (1) EP2016077A2 (https=)
JP (1) JP2009536161A (https=)
WO (1) WO2007125315A2 (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2015535226A (ja) * 2012-10-26 2015-12-10 エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ ブルートンチロシンキナーゼの阻害剤

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EP1831225A2 (en) 2004-11-19 2007-09-12 The Regents of the University of California Anti-inflammatory pyrazolopyrimidines
WO2007114926A2 (en) 2006-04-04 2007-10-11 The Regents Of The University Of California Kinase antagonists
DK3421471T3 (da) 2006-04-25 2021-06-14 Astex Therapeutics Ltd Purin- og deazapurinderivater som farmaceutiske forbindelser
GB2467670B (en) 2007-10-04 2012-08-01 Intellikine Inc Chemical entities and therapeutic uses thereof
PL2201012T3 (pl) 2007-10-11 2014-11-28 Astrazeneca Ab Pochodne pirolo[2,3-d]pirymidyny jako inhibitory kinazy białkowej b
US8193182B2 (en) 2008-01-04 2012-06-05 Intellikine, Inc. Substituted isoquinolin-1(2H)-ones, and methods of use thereof
MX2010007419A (es) 2008-01-04 2010-11-12 Intellikine Inc Ciertas entidades quimicas, composiciones y metodos.
US8993580B2 (en) 2008-03-14 2015-03-31 Intellikine Llc Benzothiazole kinase inhibitors and methods of use
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