JP2009531441A5 - - Google Patents
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- Publication number
- JP2009531441A5 JP2009531441A5 JP2009502946A JP2009502946A JP2009531441A5 JP 2009531441 A5 JP2009531441 A5 JP 2009531441A5 JP 2009502946 A JP2009502946 A JP 2009502946A JP 2009502946 A JP2009502946 A JP 2009502946A JP 2009531441 A5 JP2009531441 A5 JP 2009531441A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- salt
- composition
- patient
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 CC(C)CN(C[C@]([C@](Cc(cc1)ccc1C#N)NC(*)=O)O)S(c(cc1)ccc1OC)(=O)=O Chemical compound CC(C)CN(C[C@]([C@](Cc(cc1)ccc1C#N)NC(*)=O)O)S(c(cc1)ccc1OC)(=O)=O 0.000 description 3
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US78712606P | 2006-03-29 | 2006-03-29 | |
| US60/787,126 | 2006-03-29 | ||
| PCT/US2007/007564 WO2007126812A2 (en) | 2006-03-29 | 2007-03-29 | Process for preparation of hiv protease inhibitors |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012271186A Division JP2013082717A (ja) | 2006-03-29 | 2012-12-12 | Ｈｉｖプロテアーゼインヒビターの調製方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2009531441A JP2009531441A (ja) | 2009-09-03 |
| JP2009531441A5 true JP2009531441A5 (enExample) | 2010-05-20 |
| JP5430395B2 JP5430395B2 (ja) | 2014-02-26 |
Family
ID=38323963
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009502946A Active JP5430395B2 (ja) | 2006-03-29 | 2007-03-29 | Ｈｉｖプロテアーゼインヒビターの調製方法 |
| JP2012271186A Withdrawn JP2013082717A (ja) | 2006-03-29 | 2012-12-12 | Ｈｉｖプロテアーゼインヒビターの調製方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012271186A Withdrawn JP2013082717A (ja) | 2006-03-29 | 2012-12-12 | Ｈｉｖプロテアーゼインヒビターの調製方法 |
Country Status (24)
| Country | Link |
|---|---|
| US (4) | US20110065631A1 (enExample) |
| EP (2) | EP2570416B1 (enExample) |
| JP (2) | JP5430395B2 (enExample) |
| KR (2) | KR101429300B1 (enExample) |
| CN (2) | CN102516259B (enExample) |
| AP (2) | AP2013006690A0 (enExample) |
| AU (1) | AU2007245194B2 (enExample) |
| BR (1) | BRPI0710199A2 (enExample) |
| CA (1) | CA2647316C (enExample) |
| DK (1) | DK1999133T3 (enExample) |
| EA (2) | EA016140B1 (enExample) |
| ES (2) | ES2572001T3 (enExample) |
| HR (2) | HRP20140626A2 (enExample) |
| IL (2) | IL194122A (enExample) |
| MX (1) | MX2008012398A (enExample) |
| NO (2) | NO342102B1 (enExample) |
| NZ (2) | NZ596074A (enExample) |
| PL (1) | PL1999133T3 (enExample) |
| PT (1) | PT1999133E (enExample) |
| SG (1) | SG170794A1 (enExample) |
| SI (1) | SI1999133T1 (enExample) |
| UA (1) | UA97241C2 (enExample) |
| WO (1) | WO2007126812A2 (enExample) |
| ZA (1) | ZA200808046B (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8921415B2 (en) | 2009-01-29 | 2014-12-30 | Mapi Pharma Ltd. | Polymorphs of darunavir |
| PL2528923T3 (pl) | 2010-01-28 | 2015-01-30 | Mapi Pharma Ltd | Sposób wytwarzania darunawiru i pochodnych darunawiru |
| CN102190638A (zh) * | 2010-03-16 | 2011-09-21 | 中国科学院上海药物研究所 | 联芳基醇二胺类化合物、其药物组合物、制备方法及应用 |
| CN102584748B (zh) * | 2011-01-13 | 2015-02-11 | 浙江九洲药业股份有限公司 | 夫沙那韦中间体的制备方法 |
| EP2702045B1 (en) * | 2011-04-26 | 2017-10-18 | Mylan Laboratories Ltd. | Novel process for the preparation of etravirine |
| ES2661705T3 (es) | 2011-10-07 | 2018-04-03 | Gilead Sciences, Inc. | Métodos para la preparación de análogos de nucleótidos antivirales |
| EP2634180A1 (en) | 2012-03-01 | 2013-09-04 | Lonza Ltd. | Enzymatic process for the preparation of butyrolactones |
| CN103664976B (zh) * | 2013-12-12 | 2015-11-04 | 惠州市莱佛士制药技术有限公司 | 一种顺式六氢呋喃并[2,3-b]呋喃-3-醇的制备方法 |
| ES2802376T3 (es) | 2014-02-12 | 2021-01-19 | Firmenich Incorporated | Procedimiento mejorado para la síntesis de 1-bencil-3-(1-(isoxazol-4-ilmetil)-1h-pirazol-4-il)imidazolidin-2,4-dionas sustituidas |
| WO2016106050A1 (en) | 2014-12-26 | 2016-06-30 | Emory University | N4-hydroxycytidine and derivatives and anti-viral uses related thereto |
| JP6435907B2 (ja) * | 2015-02-16 | 2018-12-12 | 住友化学株式会社 | ヘキサヒドロフロフラノール誘導体の製造方法 |
| CN108610227B (zh) * | 2016-12-10 | 2021-02-09 | 中国科学院大连化学物理研究所 | 一种制备双环芳香化合物的方法 |
| RU2020116571A (ru) | 2017-12-07 | 2021-11-22 | Эмори Юниверсити | N4-гидроксицитидин и производные и связанные с этим противовирусные применения |
| MX2021008751A (es) | 2019-01-25 | 2021-11-12 | Univ Brown | Composiciones y metodos para tratar, prevenir o revertir la inflamacion y los trastornos asociados a la edad. |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1994026749A1 (en) * | 1993-05-14 | 1994-11-24 | Merck & Co., Inc. | Hiv protease inhibitors |
| AU1369001A (en) * | 1995-12-13 | 2001-03-22 | Abbott Laboratories | Retroviral protease inhibiting compounds |
| ATE401298T1 (de) | 1999-12-23 | 2008-08-15 | Ampac Fine Chemicals Llc | Verbessertes verfahren zur herstellung von 2s,3s- n-isobutyl-n-(2-hydroxy-3-amino-4-phenylbutyl)- - nitrobenzenesulfonylamid hydrochlorid und anderen derivaten von 2-hydroxy-1,3-diamin |
| WO2002060905A2 (en) * | 2000-10-24 | 2002-08-08 | Glaxo Group Ltd | Process for preparing intermediates of hiv protease inhibitors |
| EP1436884A2 (en) | 2001-07-20 | 2004-07-14 | Koninklijke Philips Electronics N.V. | Oscillating circuit, converter with such oscillating circuit, and preconditioner with such converter |
| TW200408645A (en) * | 2002-04-26 | 2004-06-01 | Gilead Sciences Inc | Non nucleoside reverse transcriptase inhibitors |
| US20050239054A1 (en) * | 2002-04-26 | 2005-10-27 | Arimilli Murty N | Method and compositions for identifying anti-HIV therapeutic compounds |
| WO2005042773A1 (en) * | 2003-10-24 | 2005-05-12 | Gilead Sciences, Inc. | Methods and compositions for identifying therapeutic compounds |
-
2007
- 2007-03-29 EA EA200802074A patent/EA016140B1/ru not_active IP Right Cessation
- 2007-03-29 NZ NZ596074A patent/NZ596074A/xx not_active IP Right Cessation
- 2007-03-29 HR HRP20140626AA patent/HRP20140626A2/hr not_active Application Discontinuation
- 2007-03-29 EA EA201100994A patent/EA020088B1/ru not_active IP Right Cessation
- 2007-03-29 SG SG201102217-5A patent/SG170794A1/en unknown
- 2007-03-29 PL PL07754134T patent/PL1999133T3/pl unknown
- 2007-03-29 BR BRPI0710199-6A patent/BRPI0710199A2/pt not_active IP Right Cessation
- 2007-03-29 AP AP2013006690A patent/AP2013006690A0/xx unknown
- 2007-03-29 ES ES12192910T patent/ES2572001T3/es active Active
- 2007-03-29 KR KR1020087026569A patent/KR101429300B1/ko active Active
- 2007-03-29 PT PT77541340T patent/PT1999133E/pt unknown
- 2007-03-29 AU AU2007245194A patent/AU2007245194B2/en active Active
- 2007-03-29 CA CA2647316A patent/CA2647316C/en active Active
- 2007-03-29 DK DK07754134.0T patent/DK1999133T3/da active
- 2007-03-29 SI SI200731323T patent/SI1999133T1/sl unknown
- 2007-03-29 US US12/293,450 patent/US20110065631A1/en not_active Abandoned
- 2007-03-29 CN CN201110315578.2A patent/CN102516259B/zh active Active
- 2007-03-29 EP EP12192910.3A patent/EP2570416B1/en active Active
- 2007-03-29 HR HRP20080554AA patent/HRP20080554B1/hr not_active IP Right Cessation
- 2007-03-29 NZ NZ571302A patent/NZ571302A/en not_active IP Right Cessation
- 2007-03-29 MX MX2008012398A patent/MX2008012398A/es active IP Right Grant
- 2007-03-29 KR KR1020137034899A patent/KR101395377B1/ko active Active
- 2007-03-29 JP JP2009502946A patent/JP5430395B2/ja active Active
- 2007-03-29 US US11/729,522 patent/US8173623B2/en active Active
- 2007-03-29 WO PCT/US2007/007564 patent/WO2007126812A2/en not_active Ceased
- 2007-03-29 UA UAA200811574A patent/UA97241C2/uk unknown
- 2007-03-29 ES ES07754134T patent/ES2430557T3/es active Active
- 2007-03-29 CN CN2007800178888A patent/CN101448838B/zh active Active
- 2007-03-29 AP AP2008004641A patent/AP2757A/xx active
- 2007-03-29 EP EP07754134.0A patent/EP1999133B1/en active Active
-
2008
- 2008-09-16 IL IL194122A patent/IL194122A/en not_active IP Right Cessation
- 2008-09-19 ZA ZA200808046A patent/ZA200808046B/xx unknown
- 2008-10-28 NO NO20084547A patent/NO342102B1/no unknown
-
2012
- 2012-02-21 US US13/401,659 patent/US8431745B2/en active Active
- 2012-12-12 JP JP2012271186A patent/JP2013082717A/ja not_active Withdrawn
-
2013
- 2013-02-27 US US13/779,188 patent/US20130172295A1/en not_active Abandoned
- 2013-03-12 IL IL225167A patent/IL225167A/en not_active IP Right Cessation
-
2018
- 2018-01-17 NO NO20180086A patent/NO342965B1/no unknown
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