PL2702045T3 - Nowy sposób sporządzania Etrawiryny - Google Patents

Nowy sposób sporządzania Etrawiryny

Info

Publication number
PL2702045T3
PL2702045T3 PL12731178T PL12731178T PL2702045T3 PL 2702045 T3 PL2702045 T3 PL 2702045T3 PL 12731178 T PL12731178 T PL 12731178T PL 12731178 T PL12731178 T PL 12731178T PL 2702045 T3 PL2702045 T3 PL 2702045T3
Authority
PL
Poland
Prior art keywords
etravirine
preparation
novel process
novel
Prior art date
Application number
PL12731178T
Other languages
English (en)
Inventor
Vinayak Gore
Choudhari BHARATI
Mahesh Hublikar
Prakash Bansode
Sandip SINORE
Original Assignee
Mylan Laboratories Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mylan Laboratories Ltd. filed Critical Mylan Laboratories Ltd.
Publication of PL2702045T3 publication Critical patent/PL2702045T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PL12731178T 2011-04-26 2012-04-25 Nowy sposób sporządzania Etrawiryny PL2702045T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN1441CH2011 2011-04-26
EP12731178.5A EP2702045B1 (en) 2011-04-26 2012-04-25 Novel process for the preparation of etravirine
PCT/IN2012/000303 WO2012147104A1 (en) 2011-04-26 2012-04-25 Novel process for the preparation of etravirine

Publications (1)

Publication Number Publication Date
PL2702045T3 true PL2702045T3 (pl) 2018-04-30

Family

ID=46420480

Family Applications (1)

Application Number Title Priority Date Filing Date
PL12731178T PL2702045T3 (pl) 2011-04-26 2012-04-25 Nowy sposób sporządzania Etrawiryny

Country Status (6)

Country Link
US (1) US8653266B2 (pl)
EP (1) EP2702045B1 (pl)
ES (1) ES2655525T3 (pl)
PL (1) PL2702045T3 (pl)
PT (1) PT2702045T (pl)
WO (1) WO2012147104A1 (pl)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20130123498A1 (en) * 2011-10-19 2013-05-16 Maja Sepelj MAJER Process for the preparation of etravirine and intermediates in the synthesis thereof
CN105085410B (zh) * 2015-08-21 2017-10-10 武汉工程大学 一种二芳基嘧啶类hiv‑1抑制剂及其制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU762523C (en) 1998-11-10 2004-02-12 Janssen Pharmaceutica N.V. HIV replication inhibiting pyrimidines
NZ571302A (en) * 2006-03-29 2011-11-25 Gilead Sciences Inc Process for preparation of HIV protease inhibitors via bisfuran intermediates
AP2858A (en) 2009-06-22 2014-02-28 Emcure Pharmaceuticals Ltd Process for synthesis of a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor
US8153790B2 (en) * 2009-07-27 2012-04-10 Krizmanic Irena Process for the preparation and purification of etravirine and intermediates thereof

Also Published As

Publication number Publication date
ES2655525T3 (es) 2018-02-20
US8653266B2 (en) 2014-02-18
WO2012147104A1 (en) 2012-11-01
US20130116433A1 (en) 2013-05-09
EP2702045A1 (en) 2014-03-05
PT2702045T (pt) 2018-01-11
EP2702045B1 (en) 2017-10-18

Similar Documents

Publication Publication Date Title
IL246265B (en) A method for the production of intermediates for the preparation of 5-fluoro-h1-pyrazolopyridines and such compounds
ZA201103820B (en) Process for the preparation of tenofovir
ZA201305972B (en) Method for the preparation of biphephos
PT2734536T (pt) Processo para a preparação de estetrol
PL2668163T3 (pl) Sposób wytwarzania 6-podstawionych 4-amino-3-chloro-5-fluoro-pikolinianów
ZA201404440B (en) Process for the preparation of travoprost
GB201004876D0 (en) Process for the preparation of vitamin K2
SG11201400939YA (en) Process for the preparation of methoxymelonal
ZA201302020B (en) Process for preparation of rilpivirine intermediate
PL399418A1 (pl) Sposób wytwarzania 4-metoksydihydrochalkonu
PL399419A1 (pl) Sposób wytwarzania 4-metoksydihydrochalkonu
IL236450A (en) Process for making 5-fluoro-h1-pyrazoles
EP2596007A4 (en) PROCESS FOR THE PREPARATION OF 17-DEOXY-CORTICOSTEROIDS
ZA201405824B (en) Process for the preparation of substituted phenylpropanones
ZA201300546B (en) Process for the preparation of 3-haloalkylpyrazoles
GB201119690D0 (en) Process for the preparation of compounds
PT2702045T (pt) Método inovador para a preparação de etravirina
PT2390246T (pt) Processo para a preparação de aminaftona
PL393916A1 (pl) Sposób wytwarzania związków karbapenamowych
PL2598504T3 (pl) Sposób otrzymywania dimiracetamu
PL394378A1 (pl) Sposób otrzymywania E-2-amino-4-nitrostilbenów
PL394420A1 (pl) Sposób wytwarzania dilauroilofluoresceiny
HUP1200675A2 (en) Process for the preparation of pyrimidinyl-piperazines
IL224304A (en) A process for making dichlorobulben
PL2782924T3 (pl) Proces otrzymywania drospirenonu