PT2702045T - Método inovador para a preparação de etravirina - Google Patents
Método inovador para a preparação de etravirinaInfo
- Publication number
- PT2702045T PT2702045T PT127311785T PT12731178T PT2702045T PT 2702045 T PT2702045 T PT 2702045T PT 127311785 T PT127311785 T PT 127311785T PT 12731178 T PT12731178 T PT 12731178T PT 2702045 T PT2702045 T PT 2702045T
- Authority
- PT
- Portugal
- Prior art keywords
- etravirine
- preparation
- novel process
- novel
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN1441CH2011 | 2011-04-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
PT2702045T true PT2702045T (pt) | 2018-01-11 |
Family
ID=46420480
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT127311785T PT2702045T (pt) | 2011-04-26 | 2012-04-25 | Método inovador para a preparação de etravirina |
Country Status (6)
Country | Link |
---|---|
US (1) | US8653266B2 (pt) |
EP (1) | EP2702045B1 (pt) |
ES (1) | ES2655525T3 (pt) |
PL (1) | PL2702045T3 (pt) |
PT (1) | PT2702045T (pt) |
WO (1) | WO2012147104A1 (pt) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2013059572A1 (en) * | 2011-10-19 | 2013-04-25 | Assia Chemical Industries Ltd. | Process for the preparation of etravirine and intermediates in the synthesis thereof |
CN105085410B (zh) * | 2015-08-21 | 2017-10-10 | 武汉工程大学 | 一种二芳基嘧啶类hiv‑1抑制剂及其制备方法 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ511116A (en) | 1998-11-10 | 2003-08-29 | Janssen Pharmaceutica Nv | HIV replication inhibiting pyrimidines |
US7935711B2 (en) * | 2005-02-18 | 2011-05-03 | Tibotec Pharmaceuticals Ltd. | HIV inhibiting 2-(4-cyanophenylamino) pyrimidine oxide derivatives |
KR101395377B1 (ko) * | 2006-03-29 | 2014-05-14 | 길리애드 사이언시즈, 인코포레이티드 | Hiv 단백질 분해 효소 억제제 및 그를 포함하는 약학 조성물 |
UA106972C2 (uk) | 2009-06-22 | 2014-11-10 | Емк'Юр Фармас'Ютікалз Лімітед | Спосіб синтезу діарилпіримідинового ненуклеозидного інгібітора зворотної транскриптази |
US8153790B2 (en) * | 2009-07-27 | 2012-04-10 | Krizmanic Irena | Process for the preparation and purification of etravirine and intermediates thereof |
-
2012
- 2012-04-25 PT PT127311785T patent/PT2702045T/pt unknown
- 2012-04-25 PL PL12731178T patent/PL2702045T3/pl unknown
- 2012-04-25 EP EP12731178.5A patent/EP2702045B1/en not_active Not-in-force
- 2012-04-25 WO PCT/IN2012/000303 patent/WO2012147104A1/en active Application Filing
- 2012-04-25 ES ES12731178.5T patent/ES2655525T3/es active Active
- 2012-04-26 US US13/456,319 patent/US8653266B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
ES2655525T3 (es) | 2018-02-20 |
EP2702045A1 (en) | 2014-03-05 |
US20130116433A1 (en) | 2013-05-09 |
WO2012147104A1 (en) | 2012-11-01 |
US8653266B2 (en) | 2014-02-18 |
EP2702045B1 (en) | 2017-10-18 |
PL2702045T3 (pl) | 2018-04-30 |
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