JP2009507844A - 安定化ｇｌｐ−１類似体 - Google Patents
安定化ｇｌｐ−１類似体 Download PDFInfo
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- JP2009507844A JP2009507844A JP2008530161A JP2008530161A JP2009507844A JP 2009507844 A JP2009507844 A JP 2009507844A JP 2008530161 A JP2008530161 A JP 2008530161A JP 2008530161 A JP2008530161 A JP 2008530161A JP 2009507844 A JP2009507844 A JP 2009507844A
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Cited By (2)
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| JP2016185931A (ja) * | 2015-03-27 | 2016-10-27 | 株式会社東洋新薬 | Ｇｌｐ−１分泌促進剤 |
| JP2022512908A (ja) * | 2018-10-30 | 2022-02-07 | リウ、チアンニン | Ｇｌｐ－１受容体アゴニスト活性を有するｇｌｐ－１ポリペプチドおよびその使用 |
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| CA2525574C (en) * | 2003-05-15 | 2015-06-30 | Trustees Of Tufts College | Stable analogs of peptide and polypeptide therapeutics |
| WO2009149148A2 (en) * | 2008-06-03 | 2009-12-10 | Trustees Of Tufts College | Long-acting glp-1 derivatives, and methods of treating cardiac dysfunction |
| EP2569000B1 (en) | 2010-05-13 | 2017-09-27 | Indiana University Research and Technology Corporation | Glucagon superfamily peptides exhibiting nuclear hormone receptor activity |
| CN103124739B (zh) * | 2010-05-17 | 2015-11-25 | 贝达药业股份有限公司 | 一种新胰高血糖素样肽类似物、组合物及其用途 |
| CA2796894A1 (en) | 2010-06-24 | 2011-12-29 | Indiana University Research And Technology Corporation | Amide based glucagon superfamily peptide prodrugs |
| CN102363633B (zh) * | 2011-11-16 | 2013-11-20 | 天津拓飞生物科技有限公司 | 胰高血糖素样肽-1突变体多肽及其制备方法、药物组合物和其应用 |
| US8859491B2 (en) | 2011-11-17 | 2014-10-14 | Indiana University Research And Technology Corporation | Glucagon superfamily peptides exhibiting glucocorticoid receptor activity |
| EP2630965A1 (en) * | 2012-02-24 | 2013-08-28 | Curatis Pharma GmbH | A polypeptide for the protection from neurodegeneration in patients with amyotrophic lateral sclerosis (ALS) |
| CN105934257B (zh) | 2013-12-06 | 2020-10-09 | 韩捷 | 用于含氮和羟基的药物的生物可逆引入基团 |
| TWI726889B (zh) * | 2015-06-10 | 2021-05-11 | 英商梅迪繆思有限公司 | 蛋白酶抗性之脂化肽 |
| JP7250814B2 (ja) | 2018-04-05 | 2023-04-03 | サン ファーマシューティカル インダストリーズ リミテッド | 新規ｇｌｐ－１類似体 |
Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20030119736A1 (en) * | 2001-04-02 | 2003-06-26 | Hans-Ulrich Demuth | Methods for improving islet signaling in diabetes mellitus and for its prevention |
| WO2004103390A2 (en) * | 2003-05-15 | 2004-12-02 | Trustees Of Tufts College | Stable analogs of peptide and polypeptide therapeutics |
| JP2005501058A (ja) * | 2001-07-31 | 2005-01-13 | ザ ガバメント オブ ザ ユナイテッドステイツ オブ アメリカ アズ リプレゼンテッド バイ ザ セクレタリー デパートメント オブ ヘルス アンド ヒューマン サービシーズ ザ ナショナル インステ | Ｇｌｐ−１、ｅｘｅｎｄｉｎ−４、そのペプチド・アナログ及びその使用 |
| JP2005508895A (ja) * | 2001-08-28 | 2005-04-07 | イーライ・リリー・アンド・カンパニー | Ｇｌｐ−１および基礎インスリンの予備混合物 |
| JP2005514337A (ja) * | 2001-10-18 | 2005-05-19 | ブリストル−マイヤーズ スクイブ カンパニー | ヒトグルカゴン様ペプチド−１模倣体、並びに糖尿病および関連疾患の処置におけるその使用 |
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|---|---|---|---|---|
| US3773919A (en) | 1969-10-23 | 1973-11-20 | Du Pont | Polylactide-drug mixtures |
| IE52535B1 (en) | 1981-02-16 | 1987-12-09 | Ici Plc | Continuous release pharmaceutical compositions |
| US5545618A (en) | 1990-01-24 | 1996-08-13 | Buckley; Douglas I. | GLP-1 analogs useful for diabetes treatment |
| WO1993018797A1 (en) | 1992-03-25 | 1993-09-30 | Mallinckrodt Medical, Inc. | Method of intraoperatively detecting and locating tumoral tissues |
| SG47043A1 (en) | 1993-01-06 | 1998-03-20 | Kinerton Ltd | Ionic molecular conjugates of biodegradeble polyesters and bioactive polypeptides |
| US7238671B2 (en) * | 2001-10-18 | 2007-07-03 | Bristol-Myers Squibb Company | Human glucagon-like-peptide-1 mimics and their use in the treatment of diabetes and related conditions |
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2006
- 2006-09-07 AU AU2006287562A patent/AU2006287562B2/en not_active Ceased
- 2006-09-07 JP JP2008530161A patent/JP2009507844A/ja not_active Ceased
- 2006-09-07 EP EP11194831A patent/EP2497781A1/en not_active Withdrawn
- 2006-09-07 CN CNA2006800331050A patent/CN101262874A/zh active Pending
- 2006-09-07 EP EP06814219A patent/EP1940438A4/en not_active Withdrawn
- 2006-09-07 KR KR1020087008178A patent/KR20080052649A/ko not_active Ceased
- 2006-09-07 WO PCT/US2006/034685 patent/WO2007030519A2/en not_active Ceased
- 2006-09-07 US US12/066,324 patent/US8318668B2/en active Active
- 2006-09-07 BR BRPI0615573-1A patent/BRPI0615573A2/pt not_active Application Discontinuation
- 2006-09-07 CA CA002621699A patent/CA2621699A1/en not_active Abandoned
-
2008
- 2008-03-06 IL IL189996A patent/IL189996A0/en unknown
- 2008-04-03 NO NO20081654A patent/NO20081654L/no not_active Application Discontinuation
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| US20030119736A1 (en) * | 2001-04-02 | 2003-06-26 | Hans-Ulrich Demuth | Methods for improving islet signaling in diabetes mellitus and for its prevention |
| JP2005501058A (ja) * | 2001-07-31 | 2005-01-13 | ザ ガバメント オブ ザ ユナイテッドステイツ オブ アメリカ アズ リプレゼンテッド バイ ザ セクレタリー デパートメント オブ ヘルス アンド ヒューマン サービシーズ ザ ナショナル インステ | Ｇｌｐ−１、ｅｘｅｎｄｉｎ−４、そのペプチド・アナログ及びその使用 |
| JP2005508895A (ja) * | 2001-08-28 | 2005-04-07 | イーライ・リリー・アンド・カンパニー | Ｇｌｐ−１および基礎インスリンの予備混合物 |
| JP2005514337A (ja) * | 2001-10-18 | 2005-05-19 | ブリストル−マイヤーズ スクイブ カンパニー | ヒトグルカゴン様ペプチド−１模倣体、並びに糖尿病および関連疾患の処置におけるその使用 |
| WO2004103390A2 (en) * | 2003-05-15 | 2004-12-02 | Trustees Of Tufts College | Stable analogs of peptide and polypeptide therapeutics |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2016185931A (ja) * | 2015-03-27 | 2016-10-27 | 株式会社東洋新薬 | Ｇｌｐ−１分泌促進剤 |
| JP2022512908A (ja) * | 2018-10-30 | 2022-02-07 | リウ、チアンニン | Ｇｌｐ－１受容体アゴニスト活性を有するｇｌｐ－１ポリペプチドおよびその使用 |
| JP7221385B2 (ja) | 2018-10-30 | 2023-02-13 | リウ、チアンニン | Ｇｌｐ－１受容体アゴニスト活性を有するｇｌｐ－１ポリペプチドおよびその使用 |
Also Published As
| Publication number | Publication date |
|---|---|
| US8318668B2 (en) | 2012-11-27 |
| CA2621699A1 (en) | 2007-03-15 |
| BRPI0615573A2 (pt) | 2011-05-24 |
| EP1940438A2 (en) | 2008-07-09 |
| KR20080052649A (ko) | 2008-06-11 |
| AU2006287562B2 (en) | 2012-05-10 |
| NO20081654L (no) | 2008-04-03 |
| CN101262874A (zh) | 2008-09-10 |
| WO2007030519A3 (en) | 2007-11-29 |
| EP2497781A1 (en) | 2012-09-12 |
| WO2007030519A2 (en) | 2007-03-15 |
| AU2006287562A1 (en) | 2007-03-15 |
| US20090306338A1 (en) | 2009-12-10 |
| EP1940438A4 (en) | 2009-10-21 |
| IL189996A0 (en) | 2008-08-07 |
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