JP2009502804A - ４−［６−メトキシ−７−（３−ピペリジン−１−イル−プロポキシ）キナゾリン−４−イル］ピペラジン−１−カルボン酸（４−イソプロポキシフェニル）−アミドの新規な結晶形 - Google Patents
４−［６−メトキシ−７−（３−ピペリジン−１−イル−プロポキシ）キナゾリン−４−イル］ピペラジン−１−カルボン酸（４−イソプロポキシフェニル）−アミドの新規な結晶形 Download PDFInfo
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- JP2009502804A JP2009502804A JP2008522965A JP2008522965A JP2009502804A JP 2009502804 A JP2009502804 A JP 2009502804A JP 2008522965 A JP2008522965 A JP 2008522965A JP 2008522965 A JP2008522965 A JP 2008522965A JP 2009502804 A JP2009502804 A JP 2009502804A
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- isopropoxyphenyl
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/94—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
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- Pharmacology & Pharmacy (AREA)
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- Veterinary Medicine (AREA)
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- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| US70092605P | 2005-07-20 | 2005-07-20 | |
| PCT/US2006/028231 WO2007012042A1 (en) | 2005-07-20 | 2006-07-20 | New crystal forms of 4-[6-methoxy-7-(3-piperidin-1-yl-propoxy)quinazolin-4-yl]piperazine-1-carboxylic acid(4-isopropoxyphenyl)-amide |
Publications (2)
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| JP2009502804A true JP2009502804A (ja) | 2009-01-29 |
| JP2009502804A5 JP2009502804A5 (enExample) | 2009-08-27 |
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| US (1) | US20100179162A1 (enExample) |
| EP (1) | EP1904459A1 (enExample) |
| JP (1) | JP2009502804A (enExample) |
| CN (1) | CN101208310A (enExample) |
| AU (1) | AU2006269917A1 (enExample) |
| CA (1) | CA2612459A1 (enExample) |
| WO (1) | WO2007012042A1 (enExample) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012509321A (ja) * | 2008-11-21 | 2012-04-19 | ミレニアム ファーマシューティカルズ， インコーポレイテッド | 癌および他の疾患または障害の処置のための、４−［６−メトキシ−７−（３−ピペリジン−１−イル−プロポキシ）キナゾリン−４−イル］ピペラジン−１−カルボン酸（４−イソプロポキシフェニル）−アミドの乳酸塩およびその薬学的組成物 |
| JP2014513044A (ja) * | 2011-02-10 | 2014-05-29 | マイラン ラボラトリーズ リミテッド | ホスアンプレナビルカルシウム結晶およびその調製方法 |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2015009889A1 (en) | 2013-07-18 | 2015-01-22 | Concert Pharmaceuticals, Inc. | Deuterated intedanib derivatives and their use for the treatment of proliferative disorders |
| CN109549941A (zh) * | 2017-09-26 | 2019-04-02 | 广西梧州制药（集团）股份有限公司 | 一种吡唑并嘧啶衍生物在制备治疗疾病药物方面的用途 |
Citations (1)
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| JP2004513126A (ja) * | 2000-11-01 | 2004-04-30 | ミレニアム・ファーマシューティカルズ・インコーポレイテッド | 窒素性複素環式化合物、ならびに窒素性複素環式化合物およびその中間体を作製するための方法 |
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| US642376A (en) * | 1898-10-24 | 1900-01-30 | John W Skilton | Car-axle box. |
| WO1998014431A1 (en) * | 1996-10-01 | 1998-04-09 | Kyowa Hakko Kogyo Co., Ltd. | Nitrogenous heterocyclic compounds |
| JP3011904B2 (ja) * | 1997-06-10 | 2000-02-21 | 明久 井上 | 金属ガラスの製造方法および装置 |
| EP1309568B1 (en) * | 2000-08-18 | 2011-02-16 | Millennium Pharmaceuticals, Inc. | [(quinazolin-4-yl)piperazin-4-yl]thiocarboxamide compounds as inhibitors of the phosphorylation of a PDGF receptor |
| MXPA03001359A (es) * | 2000-08-18 | 2004-12-13 | Millennium Pharm Inc | Derivados de quinazolina como inhibidores de cinasa. |
| WO2002016362A2 (en) * | 2000-08-18 | 2002-02-28 | Cor Therapeutics, Inc. | Nitrogenous heterocyclic compounds |
| US20040259881A1 (en) * | 2001-02-02 | 2004-12-23 | Anjali Pandey | Nitrogenous heterocyclic compounds |
| AU2002254152A1 (en) * | 2001-03-08 | 2002-09-24 | Millennium Pharmaceuticals | (homo) piperazine substituted quinolines for inhibiting the phosphorylation of kinases |
| US7456189B2 (en) * | 2003-09-30 | 2008-11-25 | Boehringer Ingelheim International Gmbh | Bicyclic heterocycles, medicaments containing these compounds, their use and processes for their preparation |
-
2006
- 2006-07-20 WO PCT/US2006/028231 patent/WO2007012042A1/en not_active Ceased
- 2006-07-20 EP EP06788010A patent/EP1904459A1/en not_active Withdrawn
- 2006-07-20 CA CA002612459A patent/CA2612459A1/en not_active Abandoned
- 2006-07-20 AU AU2006269917A patent/AU2006269917A1/en not_active Abandoned
- 2006-07-20 US US11/988,956 patent/US20100179162A1/en not_active Abandoned
- 2006-07-20 JP JP2008522965A patent/JP2009502804A/ja active Pending
- 2006-07-20 CN CNA2006800232271A patent/CN101208310A/zh active Pending
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2004513126A (ja) * | 2000-11-01 | 2004-04-30 | ミレニアム・ファーマシューティカルズ・インコーポレイテッド | 窒素性複素環式化合物、ならびに窒素性複素環式化合物およびその中間体を作製するための方法 |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012509321A (ja) * | 2008-11-21 | 2012-04-19 | ミレニアム ファーマシューティカルズ， インコーポレイテッド | 癌および他の疾患または障害の処置のための、４−［６−メトキシ−７−（３−ピペリジン−１−イル−プロポキシ）キナゾリン−４−イル］ピペラジン−１−カルボン酸（４−イソプロポキシフェニル）−アミドの乳酸塩およびその薬学的組成物 |
| JP2014513044A (ja) * | 2011-02-10 | 2014-05-29 | マイラン ラボラトリーズ リミテッド | ホスアンプレナビルカルシウム結晶およびその調製方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| CA2612459A1 (en) | 2007-01-25 |
| CN101208310A (zh) | 2008-06-25 |
| AU2006269917A1 (en) | 2007-01-25 |
| EP1904459A1 (en) | 2008-04-02 |
| US20100179162A1 (en) | 2010-07-15 |
| WO2007012042A1 (en) | 2007-01-25 |
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