JP2009298801A5 - - Google Patents
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- Publication number
- JP2009298801A5 JP2009298801A5 JP2009187938A JP2009187938A JP2009298801A5 JP 2009298801 A5 JP2009298801 A5 JP 2009298801A5 JP 2009187938 A JP2009187938 A JP 2009187938A JP 2009187938 A JP2009187938 A JP 2009187938A JP 2009298801 A5 JP2009298801 A5 JP 2009298801A5
- Authority
- JP
- Japan
- Prior art keywords
- pharmaceutical composition
- compound
- acceptable salt
- pharmaceutically acceptable
- agent
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 150000001875 compounds Chemical class 0.000 claims 6
- 239000008194 pharmaceutical composition Substances 0.000 claims 5
- 150000003839 salts Chemical class 0.000 claims 4
- 239000011780 sodium chloride Substances 0.000 claims 4
- 241000124008 Mammalia Species 0.000 claims 2
- 239000003795 chemical substances by application Substances 0.000 claims 2
- 239000000203 mixture Substances 0.000 claims 2
- 241000282472 Canis lupus familiaris Species 0.000 claims 1
- 241000283086 Equidae Species 0.000 claims 1
- 241000282326 Felis catus Species 0.000 claims 1
- 241000283973 Oryctolagus cuniculus Species 0.000 claims 1
- 241000283898 Ovis Species 0.000 claims 1
- 241000283984 Rodentia Species 0.000 claims 1
- 241000555745 Sciuridae Species 0.000 claims 1
- 241000282887 Suidae Species 0.000 claims 1
- 241000282458 Ursus sp. Species 0.000 claims 1
- 230000001154 acute Effects 0.000 claims 1
- 239000004599 antimicrobial Substances 0.000 claims 1
- 239000000969 carrier Substances 0.000 claims 1
- 230000001684 chronic Effects 0.000 claims 1
- 201000009910 diseases by infectious agent Diseases 0.000 claims 1
- HZOVBXHLEVMAML-FIMAOPCTSA-N CCN(CC)Cc(cc1)c(C[C@@H](C[C@@H]([C@H](C(O)=C(C(N)=O)C2=O)N(C)C)[C@@]22O)C(C3=O)=C2O)c3c1O Chemical compound CCN(CC)Cc(cc1)c(C[C@@H](C[C@@H]([C@H](C(O)=C(C(N)=O)C2=O)N(C)C)[C@@]22O)C(C3=O)=C2O)c3c1O HZOVBXHLEVMAML-FIMAOPCTSA-N 0.000 description 1
- 0 CCN(CC)Cc1ccc(*)c(C(C2=C([C@@]([C@@](C3)C(C(O)=C4C(*)=*)N(C)C)(C4=O)O)O)=O)c1C[C@]23[U] Chemical compound CCN(CC)Cc1ccc(*)c(C(C2=C([C@@]([C@@](C3)C(C(O)=C4C(*)=*)N(C)C)(C4=O)O)O)=O)c1C[C@]23[U] 0.000 description 1
Claims (7)
- 下記の化合物、またはその薬学的に許容される塩。
- 該化合物が
である、請求項１記載の化合物、またはその薬学的に許容される塩。 - 請求項１または２に記載の化合物、またはその薬学的に許容される塩を含む、哺乳類における急性または慢性の感染を治療するための薬学的組成物。
- 前記哺乳類が、ネコ、イヌ、ウマ、ブタ、ウシ、ヒツジ、齧歯類、ウサギ、リス、およびクマからなる群から選択される、請求項３記載の薬学的組成物。
- 前記化合物が、第二の薬剤と組み合わせて投与されるように用いられる、請求項３または４記載の薬学的組成物。
- 前記第二の薬剤が、抗感染剤である、請求項５記載の薬学的組成物。
- 担体と組み合わせて、請求項１または２記載の化合物、またはその薬学的に許容される塩の有効な量を含む、薬学的組成物。
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US30554601P | 2001-07-13 | 2001-07-13 | |
| US60/305,546 | 2001-07-13 | ||
| US39574102P | 2002-07-12 | 2002-07-12 | |
| US60/395,741 | 2002-07-12 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003511780A Division JP2004537544A (ja) | 2001-07-13 | 2002-07-15 | 標的治療活性を有するテトラサイクリン化合物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2009298801A JP2009298801A (ja) | 2009-12-24 |
| JP2009298801A5 true JP2009298801A5 (ja) | 2012-06-21 |
| JP5182956B2 JP5182956B2 (ja) | 2013-04-17 |
Family
ID=29553007
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003511780A Pending JP2004537544A (ja) | 2001-07-13 | 2002-07-15 | 標的治療活性を有するテトラサイクリン化合物 |
| JP2009187938A Expired - Fee Related JP5182956B2 (ja) | 2001-07-13 | 2009-08-14 | 標的治療活性を有するテトラサイクリン化合物 |
| JP2010256651A Pending JP2011057693A (ja) | 2001-07-13 | 2010-11-17 | 標的治療活性を有するテトラサイクリン化合物 |
| JP2010256652A Pending JP2011057694A (ja) | 2001-07-13 | 2010-11-17 | 標的治療活性を有するテトラサイクリン化合物 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003511780A Pending JP2004537544A (ja) | 2001-07-13 | 2002-07-15 | 標的治療活性を有するテトラサイクリン化合物 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010256651A Pending JP2011057693A (ja) | 2001-07-13 | 2010-11-17 | 標的治療活性を有するテトラサイクリン化合物 |
| JP2010256652A Pending JP2011057694A (ja) | 2001-07-13 | 2010-11-17 | 標的治療活性を有するテトラサイクリン化合物 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20040063674A1 (ja) |
| EP (11) | EP2332546A1 (ja) |
| JP (4) | JP2004537544A (ja) |
| AU (1) | AU2002318238A1 (ja) |
| WO (1) | WO2003005971A2 (ja) |
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-
2002
- 2002-07-15 EP EP10185605A patent/EP2332546A1/en not_active Withdrawn
- 2002-07-15 AU AU2002318238A patent/AU2002318238A1/en not_active Abandoned
- 2002-07-15 EP EP10185627A patent/EP2327409A1/en not_active Withdrawn
- 2002-07-15 EP EP02748169.6A patent/EP1408987B1/en not_active Expired - Lifetime
- 2002-07-15 WO PCT/US2002/022451 patent/WO2003005971A2/en active Search and Examination
- 2002-07-15 JP JP2003511780A patent/JP2004537544A/ja active Pending
- 2002-07-15 EP EP10185596A patent/EP2301550A1/en not_active Withdrawn
- 2002-07-15 EP EP10185600A patent/EP2301915A1/en not_active Withdrawn
- 2002-07-15 EP EP10185619A patent/EP2329828A1/en not_active Withdrawn
- 2002-07-15 US US10/196,010 patent/US20040063674A1/en not_active Abandoned
- 2002-07-15 EP EP10185614A patent/EP2332547A1/en not_active Withdrawn
- 2002-07-15 EP EP10185677A patent/EP2332550A1/en not_active Withdrawn
- 2002-07-15 EP EP10185610A patent/EP2329826A1/en not_active Withdrawn
- 2002-07-15 EP EP10185623A patent/EP2332548A1/en not_active Withdrawn
- 2002-07-15 EP EP10185666A patent/EP2332549A1/en not_active Withdrawn
-
2009
- 2009-08-14 JP JP2009187938A patent/JP5182956B2/ja not_active Expired - Fee Related
-
2010
- 2010-11-17 JP JP2010256651A patent/JP2011057693A/ja active Pending
- 2010-11-17 JP JP2010256652A patent/JP2011057694A/ja active Pending
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