JP2008525502A5 - - Google Patents

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Publication number
JP2008525502A5
JP2008525502A5 JP2007548611A JP2007548611A JP2008525502A5 JP 2008525502 A5 JP2008525502 A5 JP 2008525502A5 JP 2007548611 A JP2007548611 A JP 2007548611A JP 2007548611 A JP2007548611 A JP 2007548611A JP 2008525502 A5 JP2008525502 A5 JP 2008525502A5
Authority
JP
Japan
Prior art keywords
phenyl
pyrazol
urea
dichlorophenyl
oxoethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
JP2007548611A
Other languages
English (en)
Japanese (ja)
Other versions
JP2008525502A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2005/047597 external-priority patent/WO2006081034A2/en
Publication of JP2008525502A publication Critical patent/JP2008525502A/ja
Publication of JP2008525502A5 publication Critical patent/JP2008525502A5/ja
Abandoned legal-status Critical Current

Links

JP2007548611A 2004-12-23 2005-12-23 抗炎症薬 Abandoned JP2008525502A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US63898704P 2004-12-23 2004-12-23
PCT/US2005/047597 WO2006081034A2 (en) 2004-12-23 2005-12-23 Anti-inflammatory medicaments

Publications (2)

Publication Number Publication Date
JP2008525502A JP2008525502A (ja) 2008-07-17
JP2008525502A5 true JP2008525502A5 (enExample) 2009-01-29

Family

ID=36740941

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007548611A Abandoned JP2008525502A (ja) 2004-12-23 2005-12-23 抗炎症薬

Country Status (6)

Country Link
US (1) US20090312349A1 (enExample)
EP (1) EP1836173A4 (enExample)
JP (1) JP2008525502A (enExample)
AU (1) AU2005325676A1 (enExample)
CA (1) CA2592116A1 (enExample)
WO (1) WO2006081034A2 (enExample)

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US7678792B2 (en) 2006-10-20 2010-03-16 Irm Llc Compositions and methods for modulating c-kit and PDGFR receptors
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US9790178B2 (en) 2012-11-13 2017-10-17 Array Biopharma Inc. Pyrrolidinyl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
WO2014078328A1 (en) 2012-11-13 2014-05-22 Array Biopharma Inc. N-bicyclic aryl,n'-pyrazolyl urea, thiourea, guanidine and cyanoguanidine compounds as trka kinase inhibitors
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US9822118B2 (en) 2012-11-13 2017-11-21 Array Biopharma Inc. Bicyclic heteroaryl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
EP2920166B1 (en) 2012-11-13 2016-11-02 Array Biopharma, Inc. Bicyclic urea, thiourea, guanidine and cyanoguanidine compounds useful for the treatment of pain
US9981959B2 (en) 2012-11-13 2018-05-29 Array Biopharma Inc. Thiazolyl and oxazolyl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
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LT3154959T (lt) 2014-05-15 2019-09-25 Array Biopharma, Inc. 1-((3s,4r)-4-(3-fluorfenil)-1-(2-metoksietil)pirolidin-3-il)-3-(4-metil-3-(2-metilpirimidin-5-il)-1-fenil-1h-pirazol-5-il)karbamidas kaip trka kinazės inhibitorius
GB201721185D0 (en) 2017-12-18 2018-01-31 Nodthera Ltd Sulphonyl urea derivatives
EA202091763A1 (ru) 2018-01-31 2020-12-14 ДЕСИФЕРА ФАРМАСЬЮТИКАЛЗ, ЭлЭлСи Комбинированная терапия для лечения мастоцитоза
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WO2019241311A1 (en) * 2018-06-11 2019-12-19 Northeastern University Selective ligands for modulation of girk channels
CN109134451A (zh) * 2018-09-10 2019-01-04 遵义医学院 1,3-二取代脲类与硫脲类衍生物及其应用
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CN109456280B (zh) * 2018-12-24 2020-11-10 锦州医科大学 含有脲结构的4-苯基噻唑-2-胺类衍生物及其制备方法与应用
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WO2021013712A1 (en) 2019-07-19 2021-01-28 Anagenesis Biotechnologies S.A.S. Polyaromatic urea derivatives and their use in the treatment of muscle diseases
JP7818502B2 (ja) 2019-08-12 2026-02-20 デシフェラ・ファーマシューティカルズ,エルエルシー 胃腸間質腫瘍を治療するためのリプレチニブ
WO2021030405A1 (en) 2019-08-12 2021-02-18 Deciphera Pharmaceuticals, Llc Ripretinib for treating gastrointestinal stromal tumors
TWI837402B (zh) * 2019-12-20 2024-04-01 大陸商深圳艾欣達偉醫藥科技有限公司 含氟化合物、含氟化合物之製備方法及其抗癌醫藥用途
SI4084778T1 (sl) 2019-12-30 2024-01-31 Deciphera Pharmaceuticals, Llc Formulacije inhibitorja amorfne kinaze in načini njihove uporabe
AU2020417282B2 (en) 2019-12-30 2023-08-31 Deciphera Pharmaceuticals, Llc Compositions of 1-(4-bromo-5-(1-ethyl-7-(methylamino)-2-oxo-1,2-dihydro-1,6-naphthyridin-3-yl)-2-fluorophenyl)-3-phenylurea
EP4029501A1 (en) 2021-01-19 2022-07-20 Anagenesis Biotechnologies Combination of polyaromatic urea derivatives and glucocorticoid or hdac inhibitor for the treatment of diseases or conditions associated with muscle cells and/or satellite cells
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US7202257B2 (en) * 2003-12-24 2007-04-10 Deciphera Pharmaceuticals, Llc Anti-inflammatory medicaments
US20070191336A1 (en) * 2003-12-24 2007-08-16 Flynn Daniel L Anti-inflammatory medicaments

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