JP2007536252A5 - - Google Patents
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- Publication number
- JP2007536252A5 JP2007536252A5 JP2007511571A JP2007511571A JP2007536252A5 JP 2007536252 A5 JP2007536252 A5 JP 2007536252A5 JP 2007511571 A JP2007511571 A JP 2007511571A JP 2007511571 A JP2007511571 A JP 2007511571A JP 2007536252 A5 JP2007536252 A5 JP 2007536252A5
- Authority
- JP
- Japan
- Prior art keywords
- carbonyl
- cyclopropyl
- spiro
- pyrrolidin
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 *C(*)(*)C(N1CC(*)(*)CC1)=O Chemical compound *C(*)(*)C(N1CC(*)(*)CC1)=O 0.000 description 2
Applications Claiming Priority (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US56927304P | 2004-05-07 | 2004-05-07 | |
| US60/569,273 | 2004-05-07 | ||
| US60205104P | 2004-08-17 | 2004-08-17 | |
| US60/602,051 | 2004-08-17 | ||
| US60279104P | 2004-08-19 | 2004-08-19 | |
| US60/602,791 | 2004-08-19 | ||
| US63880304P | 2004-12-22 | 2004-12-22 | |
| US60/638,803 | 2004-12-22 | ||
| PCT/US2005/015559 WO2005110992A1 (en) | 2004-05-07 | 2005-05-04 | Amido compounds and their use as pharmaceuticals |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013044576A Division JP2013151519A (ja) | 2004-05-07 | 2013-03-06 | アミド化合物およびその医薬としての使用 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2007536252A JP2007536252A (ja) | 2007-12-13 |
| JP2007536252A5 true JP2007536252A5 (enExample) | 2008-06-26 |
| JP5265913B2 JP5265913B2 (ja) | 2013-08-14 |
Family
ID=35394113
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007511571A Expired - Lifetime JP5265913B2 (ja) | 2004-05-07 | 2005-05-04 | アミド化合物およびその医薬としての使用 |
| JP2013044576A Pending JP2013151519A (ja) | 2004-05-07 | 2013-03-06 | アミド化合物およびその医薬としての使用 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013044576A Pending JP2013151519A (ja) | 2004-05-07 | 2013-03-06 | アミド化合物およびその医薬としての使用 |
Country Status (29)
| Country | Link |
|---|---|
| US (7) | US7304081B2 (enExample) |
| EP (2) | EP1756063B1 (enExample) |
| JP (2) | JP5265913B2 (enExample) |
| KR (1) | KR101252227B1 (enExample) |
| AU (1) | AU2005243222C1 (enExample) |
| BR (1) | BRPI0510736B1 (enExample) |
| CA (1) | CA2565238C (enExample) |
| CR (1) | CR8702A (enExample) |
| CY (1) | CY1116779T1 (enExample) |
| DK (1) | DK1756063T3 (enExample) |
| EA (1) | EA025359B1 (enExample) |
| EC (1) | ECSP066978A (enExample) |
| ES (1) | ES2550006T3 (enExample) |
| GE (1) | GEP201706611B (enExample) |
| HK (1) | HK1218545A1 (enExample) |
| HR (1) | HRP20151064T1 (enExample) |
| HU (1) | HUE025521T2 (enExample) |
| IL (1) | IL179042A (enExample) |
| ME (1) | ME02231B (enExample) |
| MX (1) | MX340538B (enExample) |
| NO (1) | NO340031B1 (enExample) |
| NZ (1) | NZ550775A (enExample) |
| PL (1) | PL1756063T3 (enExample) |
| PT (1) | PT1756063E (enExample) |
| RS (1) | RS54236B1 (enExample) |
| SG (1) | SG151329A1 (enExample) |
| SI (1) | SI1756063T1 (enExample) |
| TW (1) | TWI350168B (enExample) |
| WO (1) | WO2005110992A1 (enExample) |
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| CA2584502A1 (en) * | 2004-06-24 | 2006-01-05 | Incyte Corporation | 2-methylpropanamides and their use as pharmaceuticals |
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| US20060009491A1 (en) * | 2004-06-24 | 2006-01-12 | Incyte Corporation | Amido compounds and their use as pharmaceuticals |
| JP2008504278A (ja) * | 2004-06-24 | 2008-02-14 | インサイト・コーポレイション | アミド化合物およびその医薬としての使用 |
| CA2570637A1 (en) | 2004-06-24 | 2006-02-02 | Wenqing Yao | N-substituted piperidines and their use as pharmaceuticals |
| EP1758882A4 (en) * | 2004-06-24 | 2008-01-23 | Incyte Corp | AMID COMPOUNDS AND THEIR USE AS MEDICAMENTS |
| KR20130047765A (ko) | 2004-07-29 | 2013-05-08 | 아더시스 인코포레이티드 | 세로토닌 수용체 조절제로서의 트리사이클릭 인데노-피롤 유도체 |
| CN101080226A (zh) * | 2004-08-10 | 2007-11-28 | 因塞特公司 | 酰氨基化合物及它们作为药物的用途 |
| AU2005304560C1 (en) * | 2004-11-10 | 2013-05-09 | Incyte Holdings Corporation | Lactam compounds and their use as pharmaceuticals |
| US8110581B2 (en) | 2004-11-10 | 2012-02-07 | Incyte Corporation | Lactam compounds and their use as pharmaceuticals |
| BRPI0518281A2 (pt) * | 2004-11-18 | 2008-11-18 | Incyte Corp | inibidores de 11-beta hidroxilesteràide desidrogenase do tipo i e mÉtodos uso dos mesmos |
| SG176463A1 (en) | 2005-02-22 | 2011-12-29 | Univ Michigan | Small molecule inhibitors of mdm2 and uses thereof |
| WO2006105127A2 (en) | 2005-03-31 | 2006-10-05 | Takeda San Diego, Inc. | Hydroxysteroid dehydrogenase inhibitors |
| MY145694A (en) | 2005-04-11 | 2012-03-30 | Xenon Pharmaceuticals Inc | Spiroheterocyclic compounds and their uses as therapeutic agents |
| AR056968A1 (es) | 2005-04-11 | 2007-11-07 | Xenon Pharmaceuticals Inc | Compuestos espiro-oxindol y composiciones farmacéuticas |
| DE102005044813A1 (de) | 2005-05-19 | 2007-10-04 | Grünenthal GmbH | Substituierte Spiro-Verbindungen und deren Verwendung zur Herstellung von Arzneimitteln |
| AU2006257670A1 (en) * | 2005-06-14 | 2006-12-21 | Merck Frosst Canada Ltd | Reversible inhibitors of monoamine oxidase A and B |
| WO2007038138A2 (en) * | 2005-09-21 | 2007-04-05 | Incyte Corporation | Amido compounds and their use as pharmaceuticals |
| US8293900B2 (en) | 2005-09-29 | 2012-10-23 | Merck Sharp & Dohme Corp | Acylated spiropiperidine derivatives as melanocortin-4 receptor modulators |
| TW200804382A (en) | 2005-12-05 | 2008-01-16 | Incyte Corp | Lactam compounds and methods of using the same |
| US7998959B2 (en) * | 2006-01-12 | 2011-08-16 | Incyte Corporation | Modulators of 11-β hydroxyl steroid dehydrogenase type 1, pharmaceutical compositions thereof, and methods of using the same |
| KR101081293B1 (ko) | 2006-01-18 | 2011-11-08 | 에프. 호프만-라 로슈 아게 | 11 베타-에이치에스디1 억제제로서 티아졸 |
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| US8598164B2 (en) | 2010-05-06 | 2013-12-03 | Vertex Pharmaceuticals Incorporated | Heterocyclic chromene-spirocyclic piperidine amides as modulators of ion channels |
| DK2620428T3 (da) * | 2010-09-24 | 2019-07-01 | Wave Life Sciences Ltd | Asymmetrisk hjælpegruppe |
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2007
- 2007-04-06 US US11/784,450 patent/US20070179142A1/en not_active Abandoned
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2008
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2010
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