JP2007524707A5 - - Google Patents

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Publication number
JP2007524707A5
JP2007524707A5 JP2007500262A JP2007500262A JP2007524707A5 JP 2007524707 A5 JP2007524707 A5 JP 2007524707A5 JP 2007500262 A JP2007500262 A JP 2007500262A JP 2007500262 A JP2007500262 A JP 2007500262A JP 2007524707 A5 JP2007524707 A5 JP 2007524707A5
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JP
Japan
Prior art keywords
group
alkyl
formula
cycloalkyl
hydrogen atom
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2007500262A
Other languages
English (en)
Japanese (ja)
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JP4812745B2 (ja
JP2007524707A (ja
Filing date
Publication date
Priority claimed from FR0401950A external-priority patent/FR2866884B1/fr
Application filed filed Critical
Publication of JP2007524707A publication Critical patent/JP2007524707A/ja
Publication of JP2007524707A5 publication Critical patent/JP2007524707A5/ja
Application granted granted Critical
Publication of JP4812745B2 publication Critical patent/JP4812745B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2007500262A 2004-02-26 2005-02-25 アリール及びヘテロアリールピペリジンカルボン酸誘導体、その製造並びにfaah酵素阻害剤としてのその使用 Expired - Fee Related JP4812745B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR0401950 2004-02-26
FR0401950A FR2866884B1 (fr) 2004-02-26 2004-02-26 Derives d'aryl-et d'heteroaryl-piperidinecarboxylates, leur preparation et leur application en therapeutique
PCT/FR2005/000453 WO2005090347A1 (fr) 2004-02-26 2005-02-25 Derives d’aryl- et d’heteroaryl-piperidinecarboxylates, leur preparation et leur application comme inhibiteurs de l'enzyme faah

Publications (3)

Publication Number Publication Date
JP2007524707A JP2007524707A (ja) 2007-08-30
JP2007524707A5 true JP2007524707A5 (US07794700-20100914-C00152.png) 2008-04-03
JP4812745B2 JP4812745B2 (ja) 2011-11-09

Family

ID=34834067

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007500262A Expired - Fee Related JP4812745B2 (ja) 2004-02-26 2005-02-25 アリール及びヘテロアリールピペリジンカルボン酸誘導体、その製造並びにfaah酵素阻害剤としてのその使用

Country Status (27)

Country Link
US (1) US20070021405A1 (US07794700-20100914-C00152.png)
EP (1) EP1720872B1 (US07794700-20100914-C00152.png)
JP (1) JP4812745B2 (US07794700-20100914-C00152.png)
KR (1) KR20060134080A (US07794700-20100914-C00152.png)
CN (1) CN100549012C (US07794700-20100914-C00152.png)
AR (1) AR047817A1 (US07794700-20100914-C00152.png)
AT (1) ATE506361T1 (US07794700-20100914-C00152.png)
AU (1) AU2005223424B2 (US07794700-20100914-C00152.png)
BR (1) BRPI0508103A (US07794700-20100914-C00152.png)
CA (1) CA2554610A1 (US07794700-20100914-C00152.png)
CY (1) CY1111706T1 (US07794700-20100914-C00152.png)
DE (1) DE602005027546D1 (US07794700-20100914-C00152.png)
DK (1) DK1720872T3 (US07794700-20100914-C00152.png)
ES (1) ES2365896T3 (US07794700-20100914-C00152.png)
FR (1) FR2866884B1 (US07794700-20100914-C00152.png)
HK (1) HK1104287A1 (US07794700-20100914-C00152.png)
IL (1) IL177326A (US07794700-20100914-C00152.png)
MA (1) MA28365A1 (US07794700-20100914-C00152.png)
NO (1) NO20064326L (US07794700-20100914-C00152.png)
NZ (1) NZ550006A (US07794700-20100914-C00152.png)
PL (1) PL1720872T3 (US07794700-20100914-C00152.png)
PT (1) PT1720872E (US07794700-20100914-C00152.png)
RU (1) RU2376305C2 (US07794700-20100914-C00152.png)
SI (1) SI1720872T1 (US07794700-20100914-C00152.png)
TW (1) TWI353834B (US07794700-20100914-C00152.png)
WO (1) WO2005090347A1 (US07794700-20100914-C00152.png)
ZA (1) ZA200606725B (US07794700-20100914-C00152.png)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2866888B1 (fr) * 2004-02-26 2006-05-05 Sanofi Synthelabo Derives de alkylpiperazine- et alkylhomopiperazine- carboxylates, leur preparation et leur application en therapeutique
US7269708B2 (en) * 2004-04-20 2007-09-11 Rambus Inc. Memory controller for non-homogenous memory system
TW200633990A (en) 2004-11-18 2006-10-01 Takeda Pharmaceuticals Co Amide compound
KR101063663B1 (ko) 2005-02-17 2011-09-07 아스텔라스세이야쿠 가부시키가이샤 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르유도체
US7918848B2 (en) 2005-03-25 2011-04-05 Maquet Cardiovascular, Llc Tissue welding and cutting apparatus and method
US8197472B2 (en) 2005-03-25 2012-06-12 Maquet Cardiovascular, Llc Tissue welding and cutting apparatus and method
WO2007005510A1 (en) 2005-06-30 2007-01-11 Janssen Pharmaceutica N.V. N-heteroarylpiperazinyl ureas as modulators of fatty acid amide hydrolase
CA2665804A1 (en) * 2006-08-23 2008-02-28 Astellas Pharma Inc. Urea compound or salt thereof
JP4388997B2 (ja) 2006-09-05 2009-12-24 協和発酵キリン株式会社 イミダゾール誘導体
EP2178858B1 (en) * 2007-08-02 2011-12-28 Recordati Ireland Limited Novel heterocyclic compounds as mglu5 antagonists
KR101536021B1 (ko) 2007-10-16 2015-07-10 다이이찌 산쿄 가부시키가이샤 피리미딜 인돌린 화합물
EA017842B1 (ru) * 2008-03-04 2013-03-29 Вернэлис (Р&Д) Лтд. Производные азетидина и их применение
TW200948805A (en) * 2008-03-07 2009-12-01 Sigma Tau Ind Farmaceuti Enol carbamate derivatives as modulators of fatty acid amide hydrolase
EP3175806B1 (en) 2008-05-27 2018-10-17 Maquet Cardiovascular LLC Surgical instrument
US9968396B2 (en) 2008-05-27 2018-05-15 Maquet Cardiovascular Llc Surgical instrument and method
US9402680B2 (en) 2008-05-27 2016-08-02 Maquet Cardiovasular, Llc Surgical instrument and method
TWI434842B (zh) * 2008-07-14 2014-04-21 Astellas Pharma Inc Azole compounds
FR2945531A1 (fr) * 2009-05-12 2010-11-19 Sanofi Aventis Derives de 7-aza-spiro°3,5!nonane-7-carboxylates, leur preparation et leur application en therapeutique
FR2945533B1 (fr) * 2009-05-12 2011-05-27 Sanofi Aventis Derives de cyclopenta°c!pyrrolyl-alkylcarbamates d'heterocycles a 5 chainons, leur preparation et leur application en therapeutique
TW201044234A (en) * 2009-06-08 2010-12-16 Chunghwa Picture Tubes Ltd Method of scanning touch panel
US9955858B2 (en) 2009-08-21 2018-05-01 Maquet Cardiovascular Llc Surgical instrument and method for use
CA2787476C (en) * 2010-01-20 2017-07-11 Sanofi Alkyl-heterocycle carbamate derivatives, their preparation and their therapeutic application
FR2955580A1 (fr) * 2010-01-28 2011-07-29 Sanofi Aventis Derives de carbamate d'alkyl-heterocycles, leur preparation et leur application en therapeutique
FR2955325B1 (fr) * 2010-01-20 2012-01-20 Sanofi Aventis Derives de carbamates d'alkyl-heterocycles, leur preparation et leur application en therapeutique
TW201206440A (en) * 2010-04-28 2012-02-16 Astellas Pharma Inc Prophylactic or therapeutic agent for diseases associated with pains in urinary organs
JP2013147430A (ja) * 2010-04-28 2013-08-01 Astellas Pharma Inc 夜間頻尿の予防又は治療剤
DE102012018115A1 (de) 2012-09-13 2014-03-13 Matthias Lehr Aryl-N-(arylalkyl)carbamate als Hemmstoffe der Fatty Acid Amide Hydrolase
WO2014054635A1 (ja) * 2012-10-02 2014-04-10 大日本住友製薬株式会社 イミダゾール誘導体
DE102013016573A1 (de) 2013-10-04 2015-04-09 Matthias Lehr 1-Tetrazolylpropan-2-one als Inhibitoren von cytosolischer Phospholipase A2 und Fatty Acid Amide Hydrolase, insbesondere geeignet zur topischen Anwendung

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE319445T1 (de) * 1997-11-24 2006-03-15 Scripps Research Inst HEMMER DER ßGAP JUNCTION COMMUNICATIONß
CA2445294A1 (en) * 2001-04-27 2002-11-07 Bristol-Myers Squibb Company Bisarylimidazolyl fatty acid amide hydrolase inhibitors
US6982263B2 (en) * 2001-06-08 2006-01-03 Boehringer Ingelheim Pharmaceuticals, Inc. Nitriles useful as reversible inhibitors of cysteine proteases
FR2843964B1 (fr) * 2002-08-29 2004-10-01 Sanofi Synthelabo Derives de dioxane-2-alkylcarbamates, leur preparation et leur application en therapeutique
FR2850377B1 (fr) * 2003-01-23 2009-02-20 Sanofi Synthelabo Derives d'arylalkylcarbamates, leur preparation et leur application en therapeutique
FR2854633B1 (fr) * 2003-05-07 2005-06-24 Sanofi Synthelabo Derives de piperidinyl-et piperazinyl-alkylcarbamates, leur preparation et leur application en therapeutique
FR2865205B1 (fr) * 2004-01-16 2006-02-24 Sanofi Synthelabo Derives de type aryloxyalkylcarbamates, leur preparation et leur application en therapeutique
FR2866888B1 (fr) * 2004-02-26 2006-05-05 Sanofi Synthelabo Derives de alkylpiperazine- et alkylhomopiperazine- carboxylates, leur preparation et leur application en therapeutique
FR2866886B1 (fr) * 2004-02-26 2007-08-31 Sanofi Synthelabo Derives d'aryl-et d'heteroaryl-akylcarbamates, leur preparation et leur application en therapeutique
FR2866885B1 (fr) * 2004-02-26 2007-08-31 Sanofi Synthelabo Derives de piperidinylalkylcarbamates, leur prepation et leur application en therapeutique

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