JP2007518809A5 - - Google Patents

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Publication number
JP2007518809A5
JP2007518809A5 JP2006551237A JP2006551237A JP2007518809A5 JP 2007518809 A5 JP2007518809 A5 JP 2007518809A5 JP 2006551237 A JP2006551237 A JP 2006551237A JP 2006551237 A JP2006551237 A JP 2006551237A JP 2007518809 A5 JP2007518809 A5 JP 2007518809A5
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JP
Japan
Prior art keywords
alkyl
substituted
tert
pyridin
butylphenoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2006551237A
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English (en)
Japanese (ja)
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JP2007518809A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2005/001705 external-priority patent/WO2005070920A1/en
Publication of JP2007518809A publication Critical patent/JP2007518809A/ja
Publication of JP2007518809A5 publication Critical patent/JP2007518809A5/ja
Ceased legal-status Critical Current

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JP2006551237A 2004-01-21 2005-01-20 Ｐ２ｙ１レセプター阻害剤としてのアミノベンズアゾール化合物 Ceased JP2007518809A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US53786904P 2004-01-21 2004-01-21
US63816704P 2004-12-22 2004-12-22
PCT/US2005/001705 WO2005070920A1 (en) 2004-01-21 2005-01-20 Amino-benzazoles as p2y1 receptor inhibitors

Publications (2)

Publication Number Publication Date
JP2007518809A JP2007518809A (ja) 2007-07-12
JP2007518809A5 true JP2007518809A5 (https=) 2008-01-31

Family

ID=34811340

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006551237A Ceased JP2007518809A (ja) 2004-01-21 2005-01-20 Ｐ２ｙ１レセプター阻害剤としてのアミノベンズアゾール化合物

Country Status (8)

Country Link
US (2) US7470712B2 (https=)
EP (1) EP1706398B1 (https=)
JP (1) JP2007518809A (https=)
AR (1) AR047449A1 (https=)
NO (1) NO20063191L (https=)
PE (1) PE20050767A1 (https=)
TW (1) TW200530217A (https=)
WO (1) WO2005070920A1 (https=)

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TW200726764A (en) 2005-06-27 2007-07-16 Bristol Myers Squibb Co N-linked heterocyclic antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
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TWI396689B (zh) 2008-11-14 2013-05-21 Amgen Inc 作為磷酸二酯酶１０抑制劑之吡衍生物
TW201030001A (en) 2008-11-14 2010-08-16 Amgen Inc Pyridine and pyrimidine derivatives as phosphodiesterase 10 inhibitors
WO2010135014A1 (en) * 2009-02-27 2010-11-25 Vertex Pharmaceuticals Incorporated Tri-cyclic pyrazolopyridine kinase inhibitors
UY32470A (es) * 2009-03-05 2010-10-29 Boehringer Ingelheim Int Derivados de 2-{2-cloro-5-[(sustituido) metil]fenilamino} -1-metil]fenilamino}-1-metilbencimidazol-5-carboxamidas-n-(sustituidas) y sus sales fisiológicamente aceptables, composiciones conteniéndolos y aplicaciones
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US8586604B2 (en) 2010-08-20 2013-11-19 Boehringer Ingelheim International Gmbh Inhibitors of the microsomal prostaglandin E2 synthase-1
US8759537B2 (en) 2010-08-20 2014-06-24 Boehringer Ingelheim International Gmbh 3H-imidazo [4, 5-C] pyridine-6-carboxamides as anti-inflammatory agents
US9102602B2 (en) * 2010-11-29 2015-08-11 Nissan Chemical Industries, Ltd. Method for producing isothiocyanate compound
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UY33779A (es) 2010-12-10 2012-07-31 Boehringer Ingelheim Int ?2-(fenilamino)-1H-bencimidazol-5-carboxamidas novedosas?
FR2974576B1 (fr) * 2011-04-29 2013-07-19 Sanofi Aventis Derives de n-[(1h-pyrazol-1-yl)aryl]-1h-indole ou 1h- indazole-3-carboxamide, leur preparation et leurs applications en therapeutique
AR086744A1 (es) * 2011-06-28 2014-01-22 Nippon Soda Co Compuesto heterociclico conteniendo nitrogeno y fungicida para el uso en agricultura y jardineria
AU2012322095B2 (en) 2011-10-14 2017-06-29 Ambit Biosciences Corporation Heterocyclic compounds and use thereof as modulators of type III receptor tyrosine kinases
EP2725025A1 (fr) * 2012-10-26 2014-04-30 Sanofi Dérives de 1H-indole-3-carboxamide et leurs utilisation comme antagonistes du P2Y12
KR102494596B1 (ko) * 2014-07-31 2023-01-31 재단법인 한국파스퇴르연구소 2-아미노-벤즈이미다졸 유도체 및 5-리폭시게나아제 및/또는 프로스타글란딘 e 합성효소 억제제로서의 이들의 용도
WO2018211442A1 (en) 2017-05-18 2018-11-22 Pi Industries Ltd. Formimidamidine compounds useful against phytopathogenic microorganisms
CN107903274A (zh) * 2017-12-28 2018-04-13 窦玉玲 一种胺类化合物及其在抗肿瘤药物中的应用
CN113967257B (zh) * 2020-07-24 2025-07-01 上海交通大学医学院附属瑞金医院 一种c-Src SH3 RT-loop作为靶点用于抗血栓
WO2024151919A1 (en) * 2023-01-13 2024-07-18 Ifm Due, Inc. Compounds and compositions for treating conditions associated with sting activity
KR102840252B1 (ko) * 2023-04-27 2025-07-30 한국화학연구원 시아노벤즈이미다졸 유도체, 약제학적으로 허용가능한 염, 이의 제조방법 및 이를 유효성분으로 함유하는 약제학적 조성물
CN117143040B (zh) * 2023-08-02 2025-06-10 苏州大学 一种环丁烯二酮基苯并恶唑衍生物及其制备方法和应用

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AU2005245389A1 (en) 2004-05-12 2005-12-01 Bristol-Myers Squibb Company Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
WO2006078621A2 (en) 2005-01-19 2006-07-27 Bristol-Myers Squibb Company 2-phenoxy-n- (1, 3 , 4-thiadizol-2-yl) pyridin-3-amine derivatives and related compounds as p2y1 receptor inhibitors for the treatment of thromboembolic disorders
WO2007002634A1 (en) 2005-06-27 2007-01-04 Bristol-Myers Squibb Company Carbocycle and heterocycle antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
ATE502924T1 (de) 2005-06-27 2011-04-15 Bristol Myers Squibb Co Lineare harnstoffmimetika-antagonisten des p2y1- rezeptors zur behandlung von thromboseleiden

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