JP2007507514A5 - - Google Patents

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Publication number
JP2007507514A5
JP2007507514A5 JP2006534060A JP2006534060A JP2007507514A5 JP 2007507514 A5 JP2007507514 A5 JP 2007507514A5 JP 2006534060 A JP2006534060 A JP 2006534060A JP 2006534060 A JP2006534060 A JP 2006534060A JP 2007507514 A5 JP2007507514 A5 JP 2007507514A5
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JP
Japan
Prior art keywords
alkyl
independently
members
substituent assignments
independent
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2006534060A
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English (en)
Japanese (ja)
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JP2007507514A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2004/032003 external-priority patent/WO2005033088A1/en
Publication of JP2007507514A publication Critical patent/JP2007507514A/ja
Publication of JP2007507514A5 publication Critical patent/JP2007507514A5/ja
Pending legal-status Critical Current

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JP2006534060A 2003-09-30 2004-09-29 キノキサリン化合物 Pending JP2007507514A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US50717603P 2003-09-30 2003-09-30
PCT/US2004/032003 WO2005033088A1 (en) 2003-09-30 2004-09-29 Quinoxaline compounds

Publications (2)

Publication Number Publication Date
JP2007507514A JP2007507514A (ja) 2007-03-29
JP2007507514A5 true JP2007507514A5 (enExample) 2007-11-22

Family

ID=34421591

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006534060A Pending JP2007507514A (ja) 2003-09-30 2004-09-29 キノキサリン化合物

Country Status (11)

Country Link
US (1) US20050070527A1 (enExample)
EP (1) EP1670774A1 (enExample)
JP (1) JP2007507514A (enExample)
KR (1) KR20060111466A (enExample)
CN (1) CN1886389B (enExample)
AU (2) AU2004278372B2 (enExample)
CA (1) CA2540638A1 (enExample)
IL (1) IL174629A0 (enExample)
MX (1) MXPA06003578A (enExample)
WO (1) WO2005033088A1 (enExample)
ZA (1) ZA200603410B (enExample)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0525068D0 (en) 2005-12-08 2006-01-18 Novartis Ag Organic compounds
WO2007117399A2 (en) 2006-03-31 2007-10-18 Janssen Pharmaceutica N.V. Benzoimidazol-2-yl pyrimidines and pyrazines as modulators of the histamine h4 receptor
WO2007120690A2 (en) * 2006-04-10 2007-10-25 Janssen Pharmaceutica N.V. Combination histamine h1r and h4r antagonist therapy for treating pruritus
US20100016293A1 (en) * 2006-07-03 2010-01-21 Rogier Adriaan Smits Quinazolines and Related Heterocyclic Compounds, and Their Therapeutic Use
GB0614471D0 (en) 2006-07-20 2006-08-30 Syngenta Ltd Herbicidal Compounds
US7985745B2 (en) 2006-10-02 2011-07-26 Abbott Laboratories Method for pain treatment
EP2077263A1 (en) * 2008-01-02 2009-07-08 Vereniging voor christelijk hoger onderwijs, wetenschappelijk onderzoek en patiëntenzorg Quinazolines and related heterocyclic compounds and their therapeutic use
EA019143B1 (ru) * 2008-06-12 2014-01-30 Янссен Фармацевтика Нв Использование антагонистов н4-гистаминовых рецепторов для лечения послеоперационных спаек
US9371311B2 (en) 2008-06-30 2016-06-21 Janssen Pharmaceutica Nv Benzoimidazol-2-yl pyrimidine derivatives
EP2201982A1 (en) 2008-12-24 2010-06-30 INSERM (Institut National de la Santé et de la Recherche Médicale) Histamine H4 receptor antagonists for the treatment of vestibular disorders
US8349852B2 (en) 2009-01-13 2013-01-08 Novartis Ag Quinazolinone derivatives useful as vanilloid antagonists
AR080055A1 (es) 2010-02-01 2012-03-07 Novartis Ag Derivados de pirazolo-[5,1-b]-oxazol como antagonistas de los receptores de crf -1
WO2011092293A2 (en) 2010-02-01 2011-08-04 Novartis Ag Cyclohexyl amide derivatives as crf receptor antagonists
ES2527849T3 (es) 2010-02-02 2015-01-30 Novartis Ag Derivados de ciclohexilamida como antagonistas del receptor de CRF
AR086554A1 (es) 2011-05-27 2014-01-08 Novartis Ag Derivados de la piperidina 3-espirociclica como agonistas de receptores de la ghrelina
JP2015525202A (ja) 2012-05-03 2015-09-03 ノバルティス アーゲー グレリン受容体アゴニストとしての2,7−ジアザ−スピロ[4,5]デカ−7−イル誘導体のl−リンゴ酸塩およびその結晶形態
PL2858647T3 (pl) 2012-06-08 2018-10-31 Sensorion Inhibitory receptora h4 do leczenia szumów usznych
RS59909B1 (sr) 2013-03-06 2020-03-31 Janssen Pharmaceutica Nv Benzoimidazol-2-il pirimidinski modulatori histaminskog h4 receptora
CN105001169B (zh) * 2015-07-09 2017-07-21 华侨大学 一种3‑氨基喹喔啉‑2(1h)‑酮类化合物的合成方法
CN110092760B (zh) * 2019-06-04 2020-11-13 杭州师范大学 一种3-氟代烷氧基-2(1h)-喹喔啉酮及其合成方法
CN118076585A (zh) * 2021-07-23 2024-05-24 国家医疗保健研究所 革兰氏阴性菌外排泵抑制剂

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3493572A (en) * 1968-07-05 1970-02-03 Pfizer & Co C Process for producing quinoxaline-di-n-oxides
FI193974A7 (enExample) * 1973-07-13 1975-01-14 Merck & Co Inc
EP0008864A1 (en) * 1978-08-15 1980-03-19 FISONS plc Pyridopyrazine and quinoxaline derivatives, processes for their preparation, and pharmaceutical compositions containing them
DK716188D0 (da) * 1988-12-22 1988-12-22 Ferrosan As Quinoxalinforbindelser, deres fremstilling og anvendelse
DE4342024A1 (de) * 1993-12-09 1995-06-14 Hoechst Ag Kombinationspräparate, enthaltend ein Chinoxalin und ein Nukleosid
MY132385A (en) * 1995-08-31 2007-10-31 Novartis Ag 2,3-dioxo-1,2,3,4-tetrahydro-quinoxalinyl derivatives
MXPA05000784A (es) * 2002-07-19 2005-06-17 Biovitrum Ab Derivados de piperazinil-pirazinona novedosos para el tratamiento de los trastornos relacionados con el receptor 5-ht2a.

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