JP2006522790A - エレトリプタンと重炭酸ナトリウムを含む医薬組み合わせ物 - Google Patents
エレトリプタンと重炭酸ナトリウムを含む医薬組み合わせ物 Download PDFInfo
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- JP2006522790A JP2006522790A JP2006506461A JP2006506461A JP2006522790A JP 2006522790 A JP2006522790 A JP 2006522790A JP 2006506461 A JP2006506461 A JP 2006506461A JP 2006506461 A JP2006506461 A JP 2006506461A JP 2006522790 A JP2006522790 A JP 2006522790A
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- Prior art keywords
- eletriptan
- sodium bicarbonate
- migraine
- pharmaceutically acceptable
- treatment
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/405—Indole-alkanecarboxylic acids; Derivatives thereof, e.g. tryptophan, indomethacin
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- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Inorganic Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0308469A GB0308469D0 (en) | 2003-04-11 | 2003-04-11 | Pharmaceutical combination |
| GB0312479A GB0312479D0 (en) | 2003-05-30 | 2003-05-30 | Pharmaceutical combination |
| PCT/IB2004/001115 WO2004089365A1 (en) | 2003-04-11 | 2004-03-31 | Pharmaceutical combination comprising eletriptan and sodium bicarbonate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JP2006522790A true JP2006522790A (ja) | 2006-10-05 |
Family
ID=33161221
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006506461A Pending JP2006522790A (ja) | 2003-04-11 | 2004-03-31 | エレトリプタンと重炭酸ナトリウムを含む医薬組み合わせ物 |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP1615635A1 (pt) |
| JP (1) | JP2006522790A (pt) |
| AR (1) | AR044009A1 (pt) |
| BR (1) | BRPI0409127A (pt) |
| CA (1) | CA2521902A1 (pt) |
| MX (1) | MXPA05010070A (pt) |
| NL (1) | NL1025908C2 (pt) |
| PA (1) | PA8599901A1 (pt) |
| PE (1) | PE20050086A1 (pt) |
| TW (1) | TW200423929A (pt) |
| UY (1) | UY28260A1 (pt) |
| WO (1) | WO2004089365A1 (pt) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2017137306A (ja) * | 2016-02-02 | 2017-08-10 | 第一三共ヘルスケア株式会社 | トリプタンとアスコルビン酸を含有する医薬組成物 |
| JP2021529759A (ja) * | 2018-07-03 | 2021-11-04 | アクスサム セラピューティクス インコーポレイテッド | メロキシカムを含有する医薬組成物 |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009142771A2 (en) * | 2008-05-22 | 2009-11-26 | Plus Chemicals, S.A. | Salts of (r)-5-(2-phenylsulphonylethenyl)-3-(n- methylpyrrolidin-2-ylmethyl)-1h-indole, 5-bromo-3-[(r)-1- methyl-pyrrolidin-2- ylmethyl]-1h-indole and of eletriptan |
| IT1393700B1 (it) | 2009-04-22 | 2012-05-08 | F S I Fabbrica Italiana Sint | Sintesi di 3-{[(2r)-1-metilpirrolidin-2-il]metil}-5-[2-(fenilsulfonil)etil]-1h-indolo |
Citations (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6341420A (ja) * | 1986-08-01 | 1988-02-22 | ザンボン グループ エス ピー エー | 鎮痛作用を有する医薬組成物 |
| JPH06321777A (ja) * | 1993-03-26 | 1994-11-22 | Zambon Group Spa | 鎮痛作用を有する薬剤組成物 |
| JP2000344667A (ja) * | 1999-05-14 | 2000-12-12 | Pfizer Prod Inc | 片頭痛処置のための併用療法 |
| JP2001513801A (ja) * | 1997-03-05 | 2001-09-04 | スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー | パラセタモールを含む嚥下錠剤 |
| WO2002009675A1 (en) * | 2000-08-02 | 2002-02-07 | Pfizer Limited | Particulate composition of eletriptan showing a sigmoidal pattern of controlled release |
| JP2004529893A (ja) * | 2001-03-01 | 2004-09-30 | ファイザー・インク | 改善されたバイオアベイラビリティーを有する組成物 |
| JP2005515991A (ja) * | 2001-12-05 | 2005-06-02 | グラクソ グループ リミテッド | ５ｈｔ１レセプターアゴニストを含む医薬組成物 |
| JP2006523620A (ja) * | 2003-02-19 | 2006-10-19 | バイオヴェイル ラボラトリーズ インコーポレイテッド | 急速吸収選択的５−ｈｔ作用剤製剤 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5607951A (en) | 1990-10-15 | 1997-03-04 | Pfizer Inc | Indole derivatives |
| GB9417310D0 (en) | 1994-08-27 | 1994-10-19 | Pfizer Ltd | Therapeutic agents |
| US6488961B1 (en) | 1996-09-20 | 2002-12-03 | Ethypharm, Inc. | Effervescent granules and methods for their preparation |
| GB9816556D0 (en) | 1998-07-30 | 1998-09-30 | Pfizer Ltd | Therapy |
| GB9825988D0 (en) | 1998-11-27 | 1999-01-20 | Pfizer Ltd | Indole derivatives |
-
2004
- 2004-03-31 MX MXPA05010070A patent/MXPA05010070A/es active IP Right Grant
- 2004-03-31 WO PCT/IB2004/001115 patent/WO2004089365A1/en active Application Filing
- 2004-03-31 JP JP2006506461A patent/JP2006522790A/ja active Pending
- 2004-03-31 BR BRPI0409127-2A patent/BRPI0409127A/pt not_active IP Right Cessation
- 2004-03-31 EP EP04724671A patent/EP1615635A1/en not_active Withdrawn
- 2004-03-31 CA CA002521902A patent/CA2521902A1/en not_active Abandoned
- 2004-04-06 UY UY28260A patent/UY28260A1/es not_active Application Discontinuation
- 2004-04-07 PE PE2004000356A patent/PE20050086A1/es not_active Application Discontinuation
- 2004-04-07 AR ARP040101192A patent/AR044009A1/es unknown
- 2004-04-07 PA PA20048599901A patent/PA8599901A1/es unknown
- 2004-04-08 NL NL1025908A patent/NL1025908C2/nl not_active IP Right Cessation
- 2004-04-09 TW TW093109936A patent/TW200423929A/zh unknown
Patent Citations (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6341420A (ja) * | 1986-08-01 | 1988-02-22 | ザンボン グループ エス ピー エー | 鎮痛作用を有する医薬組成物 |
| JPH06321777A (ja) * | 1993-03-26 | 1994-11-22 | Zambon Group Spa | 鎮痛作用を有する薬剤組成物 |
| JP2001513801A (ja) * | 1997-03-05 | 2001-09-04 | スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー | パラセタモールを含む嚥下錠剤 |
| JP2000344667A (ja) * | 1999-05-14 | 2000-12-12 | Pfizer Prod Inc | 片頭痛処置のための併用療法 |
| WO2002009675A1 (en) * | 2000-08-02 | 2002-02-07 | Pfizer Limited | Particulate composition of eletriptan showing a sigmoidal pattern of controlled release |
| JP2004529893A (ja) * | 2001-03-01 | 2004-09-30 | ファイザー・インク | 改善されたバイオアベイラビリティーを有する組成物 |
| JP2005515991A (ja) * | 2001-12-05 | 2005-06-02 | グラクソ グループ リミテッド | ５ｈｔ１レセプターアゴニストを含む医薬組成物 |
| JP2006523620A (ja) * | 2003-02-19 | 2006-10-19 | バイオヴェイル ラボラトリーズ インコーポレイテッド | 急速吸収選択的５−ｈｔ作用剤製剤 |
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2017137306A (ja) * | 2016-02-02 | 2017-08-10 | 第一三共ヘルスケア株式会社 | トリプタンとアスコルビン酸を含有する医薬組成物 |
| JP2021529759A (ja) * | 2018-07-03 | 2021-11-04 | アクスサム セラピューティクス インコーポレイテッド | メロキシカムを含有する医薬組成物 |
| JP7237375B2 (ja) | 2018-07-03 | 2023-03-13 | アクスサム セラピューティクス インコーポレイテッド | メロキシカムを含有する医薬組成物 |
| JP7485807B2 (ja) | 2018-07-03 | 2024-05-16 | アクスサム セラピューティクス インコーポレイテッド | メロキシカムを含有する医薬組成物 |
Also Published As
| Publication number | Publication date |
|---|---|
| BRPI0409127A (pt) | 2006-03-28 |
| TW200423929A (en) | 2004-11-16 |
| CA2521902A1 (en) | 2004-10-21 |
| EP1615635A1 (en) | 2006-01-18 |
| UY28260A1 (es) | 2004-11-30 |
| NL1025908C2 (nl) | 2005-11-22 |
| MXPA05010070A (es) | 2005-11-23 |
| NL1025908A1 (nl) | 2004-10-13 |
| WO2004089365A1 (en) | 2004-10-21 |
| PA8599901A1 (es) | 2005-02-04 |
| PE20050086A1 (es) | 2005-03-01 |
| AR044009A1 (es) | 2005-08-24 |
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