JP2006504761A - Ｍｃｈ拮抗活性を有する新規アミド化合物及びこれらの化合物を含む薬物 - Google Patents

Ｍｃｈ拮抗活性を有する新規アミド化合物及びこれらの化合物を含む薬物 Download PDF

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JP2006504761A
JP2006504761A JP2004547576A JP2004547576A JP2006504761A JP 2006504761 A JP2006504761 A JP 2006504761A JP 2004547576 A JP2004547576 A JP 2004547576A JP 2004547576 A JP2004547576 A JP 2004547576A JP 2006504761 A JP2006504761 A JP 2006504761A
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chloro
phenyl
group
phenoxy
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JP2006504761A5 (enExample
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ディルク シュテンカンプ
シュテファン ゲオルグ ミューラー
ゲラルト ユールゲン ロート
フィリップ ルシュテンベルガー
クラウス ルドルフ
リンツ トルシュテン レーマン
キルシュテン アールント
ラルフ エル ハー ロッツ
マルティン レンター
ハイケ アンドレア ヴィーラント
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ベーリンガー インゲルハイム ファルマ ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディトゲゼルシャフト
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Publication of JP2006504761A publication Critical patent/JP2006504761A/ja
Publication of JP2006504761A5 publication Critical patent/JP2006504761A5/ja
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    • C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/088—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
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US11261186B2 (en) 2014-12-24 2022-03-01 Lg Chem. Ltd. Biaryl derivative as GPR120 agonist
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JP2016124812A (ja) * 2014-12-26 2016-07-11 株式会社ヤクルト本社 Ｚｎｆ１４３阻害活性を有する化合物およびその利用
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