JP2005537296A5 - - Google Patents
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- JP2005537296A5 JP2005537296A5 JP2004525996A JP2004525996A JP2005537296A5 JP 2005537296 A5 JP2005537296 A5 JP 2005537296A5 JP 2004525996 A JP2004525996 A JP 2004525996A JP 2004525996 A JP2004525996 A JP 2004525996A JP 2005537296 A5 JP2005537296 A5 JP 2005537296A5
- Authority
- JP
- Japan
- Prior art keywords
- halogen
- sealed container
- alkyl
- alkoxy
- pharmaceutical composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
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- 150000002367 halogens Chemical group 0.000 claims 26
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- 125000000217 alkyl group Chemical group 0.000 claims 18
- 125000003545 alkoxy group Chemical group 0.000 claims 11
- 239000002126 C01EB10 - Adenosine Substances 0.000 claims 10
- 229960005305 adenosine Drugs 0.000 claims 10
- 239000008194 pharmaceutical composition Substances 0.000 claims 10
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- HQKMJHAJHXVSDF-UHFFFAOYSA-L magnesium stearate Chemical compound [Mg+2].CCCCCCCCCCCCCCCCCC([O-])=O.CCCCCCCCCCCCCCCCCC([O-])=O HQKMJHAJHXVSDF-UHFFFAOYSA-L 0.000 claims 2
- HEBKCHPVOIAQTA-UHFFFAOYSA-N meso ribitol Natural products OCC(O)C(O)C(O)CO HEBKCHPVOIAQTA-UHFFFAOYSA-N 0.000 claims 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 2
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- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 2
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- WQZGKKKJIJFFOK-QTVWNMPRSA-N D-mannopyranose Chemical compound OC[C@H]1OC(O)[C@@H](O)[C@@H](O)[C@@H]1O WQZGKKKJIJFFOK-QTVWNMPRSA-N 0.000 claims 1
- 229920002307 Dextran Polymers 0.000 claims 1
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- UNXHWFMMPAWVPI-UHFFFAOYSA-N Erythritol Natural products OCC(O)C(O)CO UNXHWFMMPAWVPI-UHFFFAOYSA-N 0.000 claims 1
- VZCYOOQTPOCHFL-OWOJBTEDSA-N Fumaric acid Chemical compound OC(=O)\C=C\C(O)=O VZCYOOQTPOCHFL-OWOJBTEDSA-N 0.000 claims 1
- 108010010803 Gelatin Proteins 0.000 claims 1
- 239000004471 Glycine Substances 0.000 claims 1
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- 206010061218 Inflammation Diseases 0.000 claims 1
- LKDRXBCSQODPBY-AMVSKUEXSA-N L-(-)-Sorbose Chemical compound OCC1(O)OC[C@H](O)[C@@H](O)[C@@H]1O LKDRXBCSQODPBY-AMVSKUEXSA-N 0.000 claims 1
- QNAYBMKLOCPYGJ-REOHCLBHSA-N L-alanine Chemical compound C[C@H](N)C(O)=O QNAYBMKLOCPYGJ-REOHCLBHSA-N 0.000 claims 1
- ODKSFYDXXFIFQN-BYPYZUCNSA-P L-argininium(2+) Chemical compound NC(=[NH2+])NCCC[C@H]([NH3+])C(O)=O ODKSFYDXXFIFQN-BYPYZUCNSA-P 0.000 claims 1
- HNDVDQJCIGZPNO-YFKPBYRVSA-N L-histidine Chemical compound OC(=O)[C@@H](N)CC1=CN=CN1 HNDVDQJCIGZPNO-YFKPBYRVSA-N 0.000 claims 1
- ROHFNLRQFUQHCH-YFKPBYRVSA-N L-leucine Chemical compound CC(C)C[C@H](N)C(O)=O ROHFNLRQFUQHCH-YFKPBYRVSA-N 0.000 claims 1
- COLNVLDHVKWLRT-QMMMGPOBSA-N L-phenylalanine Chemical compound OC(=O)[C@@H](N)CC1=CC=CC=C1 COLNVLDHVKWLRT-QMMMGPOBSA-N 0.000 claims 1
- QIVBCDIJIAJPQS-VIFPVBQESA-N L-tryptophane Chemical compound C1=CC=C2C(C[C@H](N)C(O)=O)=CNC2=C1 QIVBCDIJIAJPQS-VIFPVBQESA-N 0.000 claims 1
- OUYCCCASQSFEME-QMMMGPOBSA-N L-tyrosine Chemical compound OC(=O)[C@@H](N)CC1=CC=C(O)C=C1 OUYCCCASQSFEME-QMMMGPOBSA-N 0.000 claims 1
- ROHFNLRQFUQHCH-UHFFFAOYSA-N Leucine Natural products CC(C)CC(N)C(O)=O ROHFNLRQFUQHCH-UHFFFAOYSA-N 0.000 claims 1
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- 229910019142 PO4 Inorganic materials 0.000 claims 1
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- MUPFEKGTMRGPLJ-RMMQSMQOSA-N Raffinose Natural products O(C[C@H]1[C@@H](O)[C@H](O)[C@@H](O)[C@@H](O[C@@]2(CO)[C@H](O)[C@@H](O)[C@@H](CO)O2)O1)[C@@H]1[C@H](O)[C@@H](O)[C@@H](O)[C@@H](CO)O1 MUPFEKGTMRGPLJ-RMMQSMQOSA-N 0.000 claims 1
- 206010038687 Respiratory distress Diseases 0.000 claims 1
- 229930006000 Sucrose Natural products 0.000 claims 1
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- HDTRYLNUVZCQOY-LIZSDCNHSA-N alpha,alpha-trehalose Chemical compound O[C@@H]1[C@@H](O)[C@H](O)[C@@H](CO)O[C@@H]1O[C@@H]1[C@H](O)[C@@H](O)[C@H](O)[C@@H](CO)O1 HDTRYLNUVZCQOY-LIZSDCNHSA-N 0.000 claims 1
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US38924202P | 2002-06-17 | 2002-06-17 | |
| US47798703P | 2003-06-11 | 2003-06-11 | |
| PCT/US2003/018944 WO2004012653A2 (en) | 2002-06-17 | 2003-06-17 | Nebulizer formulations of dehydroepiandrosterone and methods of treating asthma or chronic obstructive pulmonary disease using compostions thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005537296A JP2005537296A (ja) | 2005-12-08 |
| JP2005537296A5 true JP2005537296A5 (enExample) | 2006-08-10 |
Family
ID=29740120
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004512683A Pending JP2005530820A (ja) | 2002-06-17 | 2003-06-17 | 二水和デヒドロエピアンドロステロン及びその組成物を用いた喘息又は慢性閉塞性肺疾患の治療方法 |
| JP2004525996A Pending JP2005537296A (ja) | 2002-06-17 | 2003-06-17 | デヒドロエピアンドロステロンの噴霧器製剤及びその組成物を使用することでの喘息又は慢性閉塞性肺疾患を治療するための方法 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004512683A Pending JP2005530820A (ja) | 2002-06-17 | 2003-06-17 | 二水和デヒドロエピアンドロステロン及びその組成物を用いた喘息又は慢性閉塞性肺疾患の治療方法 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20090087389A1 (enExample) |
| EP (2) | EP1513509A4 (enExample) |
| JP (2) | JP2005530820A (enExample) |
| KR (2) | KR20060011784A (enExample) |
| CN (2) | CN1681520A (enExample) |
| AU (2) | AU2003269889B2 (enExample) |
| BR (2) | BR0311883A (enExample) |
| CA (2) | CA2489124A1 (enExample) |
| IL (2) | IL165291A0 (enExample) |
| MX (2) | MXPA04012728A (enExample) |
| WO (2) | WO2003105775A2 (enExample) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2496867A1 (en) * | 2002-08-28 | 2004-03-11 | Hollis-Eden Pharmaceuticals, Inc. | Therapeutic treatment methods |
| EP1638549A4 (en) | 2003-03-10 | 2011-06-15 | Optimer Pharmaceuticals Inc | NEW ANTIBACTERIAL AGENTS |
| US7858607B2 (en) | 2003-03-14 | 2010-12-28 | Mamchur Stephen A | System for use by compounding pharmacists to produce hormone replacement medicine customized for each consumer |
| EP1898894A1 (en) * | 2005-06-17 | 2008-03-19 | Boehringer Ingelheim International GmbH | Mrp iv inhibitors for the treatment of respiratory diseases |
| GB0520794D0 (en) * | 2005-10-12 | 2005-11-23 | Innovata Biomed Ltd | Inhaler |
| BRPI0709872A2 (pt) * | 2006-04-03 | 2011-07-26 | Teva Pharma | micropartÍculas de drogas |
| EP2170270B1 (en) * | 2007-06-05 | 2016-01-13 | Paka Pulmonary Pharmaceuticals, Inc. | Compositions for delivering medicaments into the lungs, uses thereof |
| US9453042B2 (en) | 2007-10-25 | 2016-09-27 | Cempra Pharmaceuticals, Inc. | Process for the preparation of macrolide antibacterial agents |
| HRP20160222T1 (hr) | 2008-10-24 | 2016-04-08 | Cempra Pharmaceuticals, Inc. | Biozaštite uporabom makrolida koji sadrže triazol |
| WO2010068754A2 (en) | 2008-12-10 | 2010-06-17 | Paka Pulmonary Pharmaceuticals, Inc. | Methods and compositions for delivery of medicaments to the lungs |
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2003
- 2003-06-17 IL IL16529103A patent/IL165291A0/xx unknown
- 2003-06-17 JP JP2004512683A patent/JP2005530820A/ja active Pending
- 2003-06-17 CA CA002489124A patent/CA2489124A1/en not_active Abandoned
- 2003-06-17 CN CNA038136813A patent/CN1681520A/zh active Pending
- 2003-06-17 CA CA002491846A patent/CA2491846A1/en not_active Abandoned
- 2003-06-17 BR BR0311883-5A patent/BR0311883A/pt not_active IP Right Cessation
- 2003-06-17 WO PCT/US2003/018945 patent/WO2003105775A2/en not_active Ceased
- 2003-06-17 MX MXPA04012728A patent/MXPA04012728A/es not_active Application Discontinuation
- 2003-06-17 AU AU2003269889A patent/AU2003269889B2/en not_active Ceased
- 2003-06-17 EP EP03766816A patent/EP1513509A4/en not_active Withdrawn
- 2003-06-17 EP EP03751776A patent/EP1553954A4/en not_active Withdrawn
- 2003-06-17 WO PCT/US2003/018944 patent/WO2004012653A2/en not_active Ceased
- 2003-06-17 CN CNB038136910A patent/CN100540007C/zh not_active Expired - Fee Related
- 2003-06-17 IL IL16537803A patent/IL165378A0/xx unknown
- 2003-06-17 MX MXPA04012720A patent/MXPA04012720A/es active IP Right Grant
- 2003-06-17 AU AU2003276836A patent/AU2003276836B2/en not_active Ceased
- 2003-06-17 BR BR0311885-1A patent/BR0311885A/pt not_active IP Right Cessation
- 2003-06-17 KR KR1020047020469A patent/KR20060011784A/ko not_active Abandoned
- 2003-06-17 JP JP2004525996A patent/JP2005537296A/ja active Pending
- 2003-06-17 KR KR1020047020590A patent/KR101005819B1/ko not_active Expired - Fee Related
-
2008
- 2008-09-25 US US12/238,403 patent/US20090087389A1/en not_active Abandoned
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