JP2005518382A5 - - Google Patents

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JP2005518382A5
JP2005518382A5 JP2003554118A JP2003554118A JP2005518382A5 JP 2005518382 A5 JP2005518382 A5 JP 2005518382A5 JP 2003554118 A JP2003554118 A JP 2003554118A JP 2003554118 A JP2003554118 A JP 2003554118A JP 2005518382 A5 JP2005518382 A5 JP 2005518382A5
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Japan
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substituted
alkyl
aryl
heterocycle
cycloalkenyl
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JP2003554118A
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Japanese (ja)
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JP2005518382A (ja
JP4434740B2 (ja
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Priority claimed from PCT/US2002/040737 external-priority patent/WO2003053358A2/en
Publication of JP2005518382A publication Critical patent/JP2005518382A/ja
Publication of JP2005518382A5 publication Critical patent/JP2005518382A5/ja
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Publication of JP4434740B2 publication Critical patent/JP4434740B2/ja
Anticipated expiration legal-status Critical
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JP2003554118A 2001-12-19 2002-12-18 核ホルモン受容体機能の調節剤である、縮合ヘテロ環化合物およびその類似体 Expired - Fee Related JP4434740B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US34196201P 2001-12-19 2001-12-19
PCT/US2002/040737 WO2003053358A2 (en) 2001-12-19 2002-12-18 Fused heterocyclic compounds and analogs thereof: modulators of nuclear hormone receptor function

Publications (3)

Publication Number Publication Date
JP2005518382A JP2005518382A (ja) 2005-06-23
JP2005518382A5 true JP2005518382A5 (enExample) 2006-02-02
JP4434740B2 JP4434740B2 (ja) 2010-03-17

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JP2003554118A Expired - Fee Related JP4434740B2 (ja) 2001-12-19 2002-12-18 核ホルモン受容体機能の調節剤である、縮合ヘテロ環化合物およびその類似体

Country Status (10)

Country Link
US (3) US7087636B2 (enExample)
EP (1) EP1467979B1 (enExample)
JP (1) JP4434740B2 (enExample)
AT (1) ATE404544T1 (enExample)
AU (1) AU2002364082A1 (enExample)
DE (1) DE60228330D1 (enExample)
ES (1) ES2310622T3 (enExample)
HU (1) HUP0500096A3 (enExample)
PL (1) PL206962B1 (enExample)
WO (1) WO2003053358A2 (enExample)

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US9180091B2 (en) 2012-12-21 2015-11-10 Therapeuticsmd, Inc. Soluble estradiol capsule for vaginal insertion
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US11266661B2 (en) 2012-12-21 2022-03-08 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10471072B2 (en) 2012-12-21 2019-11-12 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US11246875B2 (en) 2012-12-21 2022-02-15 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10537581B2 (en) 2012-12-21 2020-01-21 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
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US10328087B2 (en) 2015-07-23 2019-06-25 Therapeuticsmd, Inc. Formulations for solubilizing hormones
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