PL206962B1 - Związek heterocykliczny o budowie skondensowanej - Google Patents
Związek heterocykliczny o budowie skondensowanejInfo
- Publication number
- PL206962B1 PL206962B1 PL371191A PL37119102A PL206962B1 PL 206962 B1 PL206962 B1 PL 206962B1 PL 371191 A PL371191 A PL 371191A PL 37119102 A PL37119102 A PL 37119102A PL 206962 B1 PL206962 B1 PL 206962B1
- Authority
- PL
- Poland
- Prior art keywords
- formula
- isoindol
- compound
- phenyl
- compounds
- Prior art date
Links
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
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| US20040077605A1 (en) * | 2001-06-20 | 2004-04-22 | Salvati Mark E. | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
| US7001911B2 (en) * | 2000-06-28 | 2006-02-21 | Bristol-Myers Squibb Company | Fused cyclic modulators of nuclear hormone receptor function |
| EP1854798A3 (en) * | 2000-09-19 | 2007-11-28 | Bristol-Myers Squibb Company | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
| US20040087548A1 (en) | 2001-02-27 | 2004-05-06 | Salvati Mark E. | Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
| DE60228330D1 (de) * | 2001-12-19 | 2008-09-25 | Bristol Myers Squibb Co | Kondensierte heterocyclische verbindungen und deren analoga; modulatoren der funktion von nukleären hormonrezeptoren |
| FR2860793A1 (fr) * | 2003-10-14 | 2005-04-15 | Entomed | Composes derives de norcantharidine, leurs procedes de preparation, les compositions les contenant et leurs utilisations |
| CN1918151A (zh) * | 2003-12-19 | 2007-02-21 | 伊莱利利公司 | 三环甾类激素核受体调节剂 |
| EP1750862B1 (en) | 2004-06-04 | 2011-01-05 | Teva Pharmaceutical Industries Ltd. | Pharmaceutical composition containing irbesartan |
| WO2005123043A2 (en) * | 2004-06-10 | 2005-12-29 | Duramed Pharmaceuticals, Inc. | Formulations of sumatriptan for absorption across biological membranes, and methods of making and using the same |
| SE0500055D0 (sv) * | 2005-01-10 | 2005-01-10 | Astrazeneca Ab | Therapeutic agents 3 |
| US7776859B2 (en) * | 2005-10-14 | 2010-08-17 | Bristol-Myers Squibb Company | Hexahydroimidazopyrazin-3-one compounds useful as modulators of androgen receptor function |
| AR056893A1 (es) * | 2005-12-28 | 2007-10-31 | Takeda Pharmaceutical | Compuestos heterociclicos fusionados y no fusionados, antagonistas de receptores mineralocorticoides |
| US7468439B2 (en) * | 2006-09-06 | 2008-12-23 | Bristol-Myers Squibb Company | Alkylene bridged sultam compounds useful as modulators of nuclear hormone receptor function |
| WO2008064136A2 (en) * | 2006-11-17 | 2008-05-29 | Acadia Pharmaceuticals Inc. | Compounds with activity at retinoic acid receptors |
| EP2170899A1 (en) | 2007-06-27 | 2010-04-07 | Bristol-Myers Squibb Company | Fused heterocyclic compounds useful as modulators of nuclear hormone receptor function |
| WO2009059077A1 (en) * | 2007-11-01 | 2009-05-07 | Bristol-Myers Squibb Company | Fused heterocyclic compounds useful as modulators of nuclear hormone receptor function |
| EP2782584B1 (en) | 2011-11-23 | 2021-06-09 | TherapeuticsMD, Inc. | Natural combination hormone replacement formulations and therapies |
| US9301920B2 (en) | 2012-06-18 | 2016-04-05 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
| US20130338122A1 (en) | 2012-06-18 | 2013-12-19 | Therapeuticsmd, Inc. | Transdermal hormone replacement therapies |
| US20150196640A1 (en) | 2012-06-18 | 2015-07-16 | Therapeuticsmd, Inc. | Progesterone formulations having a desirable pk profile |
| US10806697B2 (en) | 2012-12-21 | 2020-10-20 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
| US10806740B2 (en) | 2012-06-18 | 2020-10-20 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
| US9180091B2 (en) | 2012-12-21 | 2015-11-10 | Therapeuticsmd, Inc. | Soluble estradiol capsule for vaginal insertion |
| US10568891B2 (en) | 2012-12-21 | 2020-02-25 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
| US11266661B2 (en) | 2012-12-21 | 2022-03-08 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
| US10471072B2 (en) | 2012-12-21 | 2019-11-12 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
| US11246875B2 (en) | 2012-12-21 | 2022-02-15 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
| US10537581B2 (en) | 2012-12-21 | 2020-01-21 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
| AU2015264003A1 (en) | 2014-05-22 | 2016-11-17 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
| US10328087B2 (en) | 2015-07-23 | 2019-06-25 | Therapeuticsmd, Inc. | Formulations for solubilizing hormones |
| WO2017173071A1 (en) | 2016-04-01 | 2017-10-05 | Therapeuticsmd, Inc. | Steroid hormone pharmaceutical composition |
| US10286077B2 (en) | 2016-04-01 | 2019-05-14 | Therapeuticsmd, Inc. | Steroid hormone compositions in medium chain oils |
| US11633405B2 (en) | 2020-02-07 | 2023-04-25 | Therapeuticsmd, Inc. | Steroid hormone pharmaceutical formulations |
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| GB1039020A (en) | 1964-09-21 | 1966-08-17 | Biorex Laboratories Ltd | Process for the preparation of 5-nitrofurfuraldehyde diacetate |
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| JPS4916937B1 (enExample) | 1970-01-21 | 1974-04-25 | ||
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| JPS5188631U (enExample) | 1975-01-10 | 1976-07-15 | ||
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| JPS5386035U (enExample) | 1976-12-16 | 1978-07-15 | ||
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-
2002
- 2002-12-18 DE DE60228330T patent/DE60228330D1/de not_active Expired - Lifetime
- 2002-12-18 AU AU2002364082A patent/AU2002364082A1/en not_active Abandoned
- 2002-12-18 AT AT02798550T patent/ATE404544T1/de not_active IP Right Cessation
- 2002-12-18 US US10/322,276 patent/US7087636B2/en not_active Expired - Lifetime
- 2002-12-18 EP EP02798550A patent/EP1467979B1/en not_active Expired - Lifetime
- 2002-12-18 JP JP2003554118A patent/JP4434740B2/ja not_active Expired - Fee Related
- 2002-12-18 ES ES02798550T patent/ES2310622T3/es not_active Expired - Lifetime
- 2002-12-18 WO PCT/US2002/040737 patent/WO2003053358A2/en not_active Ceased
- 2002-12-18 HU HU0500096A patent/HUP0500096A3/hu unknown
- 2002-12-18 PL PL371191A patent/PL206962B1/pl not_active IP Right Cessation
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2005
- 2005-04-21 US US11/111,606 patent/US7291637B2/en not_active Expired - Lifetime
- 2005-09-21 US US11/231,447 patent/US7342034B2/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| EP1467979A4 (en) | 2006-03-15 |
| DE60228330D1 (de) | 2008-09-25 |
| US7087636B2 (en) | 2006-08-08 |
| PL371191A1 (en) | 2005-06-13 |
| WO2003053358A3 (en) | 2003-10-02 |
| US7342034B2 (en) | 2008-03-11 |
| US20030181728A1 (en) | 2003-09-25 |
| EP1467979A2 (en) | 2004-10-20 |
| AU2002364082A8 (en) | 2003-07-09 |
| US20050187273A1 (en) | 2005-08-25 |
| US7291637B2 (en) | 2007-11-06 |
| ES2310622T3 (es) | 2009-01-16 |
| AU2002364082A1 (en) | 2003-07-09 |
| US20060020002A1 (en) | 2006-01-26 |
| EP1467979B1 (en) | 2008-08-13 |
| JP2005518382A (ja) | 2005-06-23 |
| HUP0500096A3 (en) | 2012-08-28 |
| ATE404544T1 (de) | 2008-08-15 |
| WO2003053358A2 (en) | 2003-07-03 |
| JP4434740B2 (ja) | 2010-03-17 |
| HUP0500096A2 (hu) | 2005-05-30 |
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