JP2005514456A5 - - Google Patents

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Publication number
JP2005514456A5
JP2005514456A5 JP2003559979A JP2003559979A JP2005514456A5 JP 2005514456 A5 JP2005514456 A5 JP 2005514456A5 JP 2003559979 A JP2003559979 A JP 2003559979A JP 2003559979 A JP2003559979 A JP 2003559979A JP 2005514456 A5 JP2005514456 A5 JP 2005514456A5
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JP
Japan
Prior art keywords
alkyl
halogen
nhc
alkoxy
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2003559979A
Other languages
English (en)
Japanese (ja)
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JP2005514456A (ja
Filing date
Publication date
Priority claimed from IT2002RM000014A external-priority patent/ITRM20020014A1/it
Application filed filed Critical
Publication of JP2005514456A publication Critical patent/JP2005514456A/ja
Publication of JP2005514456A5 publication Critical patent/JP2005514456A5/ja
Pending legal-status Critical Current

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JP2003559979A 2002-01-15 2003-01-15 PPARα活性化に応答する疾患の治療に有用なα−フェニルチオカルボン酸およびα−フェニルオキシカルボン酸の誘導体 Pending JP2005514456A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT2002RM000014A ITRM20020014A1 (it) 2002-01-15 2002-01-15 Derivati di acidi a-feniltiocarbossilici e a-fenilossicarbossilici utili per il trattamento di patologie che rispondono all'attivazione del
PCT/IT2003/000011 WO2003059875A2 (en) 2002-01-15 2003-01-15 DERIVATIVES OF α-PHENYLTHIOCARBOXYLIC AND α-PHENYLOXY-CARBOXYLIC ACIDS USEFUL FOR THE TREATMENT OF DISEASES RESPONDING TO PPARα ACTIVATION

Publications (2)

Publication Number Publication Date
JP2005514456A JP2005514456A (ja) 2005-05-19
JP2005514456A5 true JP2005514456A5 (https=) 2006-07-13

Family

ID=11455954

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003559979A Pending JP2005514456A (ja) 2002-01-15 2003-01-15 PPARα活性化に応答する疾患の治療に有用なα−フェニルチオカルボン酸およびα−フェニルオキシカルボン酸の誘導体

Country Status (16)

Country Link
US (2) US20050054671A1 (https=)
EP (1) EP1474387B1 (https=)
JP (1) JP2005514456A (https=)
KR (1) KR100975961B1 (https=)
CN (1) CN100522940C (https=)
AR (1) AR038146A1 (https=)
AT (1) ATE489361T1 (https=)
AU (1) AU2003209679B2 (https=)
BR (1) BR0306824A (https=)
CA (1) CA2472223A1 (https=)
DE (1) DE60335083D1 (https=)
IT (1) ITRM20020014A1 (https=)
MX (1) MXPA04006803A (https=)
PL (1) PL372666A1 (https=)
TW (1) TW200305410A (https=)
WO (1) WO2003059875A2 (https=)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003261935A1 (en) * 2002-09-06 2004-03-29 Takeda Pharmaceutical Company Limited Furan or thiophene derivative and medicinal use thereof
ITRM20020629A1 (it) * 2002-12-19 2004-06-20 Sigma Tau Ind Farmaceuti Uso di acidi alfa-feniltiocarbossilici e alfa-fenilossicarbossilici ad attivita' ipoglicemizzante e/o ipolipidemizzante.
WO2005042478A2 (en) 2003-09-19 2005-05-12 Janssen Pharmaceutica, N.V. 4-((phenoxyalkyl)thio)-phenoxyacetic acids and analogs
MXPA06003019A (es) * 2003-10-28 2006-06-23 Reddys Lab Ltd Dr Nuevos compuestos y su uso en medicina: proceso para su preparacion y composiciones farmaceuticas que los contienen.
AU2005272389B2 (en) 2004-08-11 2011-08-04 Kyorin Pharmaceutical Co., Ltd. Novel cyclic aminobenzoic acid derivative
MY147518A (en) * 2004-09-15 2012-12-31 Janssen Pharmaceutica Nv 4-((phenoxyalkyl)thio)-phenoxyacetic acids and analogs
FR2880886B1 (fr) * 2005-01-14 2007-04-06 Merck Sante Soc Par Actions Si Derives de l'acide 6-phenylhex-5-enoique, procedes pour leur preparation, compositions pharmaceutiques les contenant et applications en therapeutique
WO2006082495A1 (en) * 2005-02-02 2006-08-10 Ranbaxy Laboratories Limited Peroxisome proliferator activated receptor modulators
FR2882359A1 (fr) * 2005-02-24 2006-08-25 Negma Lerads Soc Par Actions S Derives activateurs de ppar, procede de preparation et application en therapeutique
JPWO2006101108A1 (ja) * 2005-03-23 2008-09-04 杏林製薬株式会社 新規環状アミノフェニルアルカン酸誘導体
JO3006B1 (ar) 2005-09-14 2016-09-05 Janssen Pharmaceutica Nv املاح ليسين مبتكرة من مشتقات حامض 4-((فينوكسي الكيل)ثيو) فينوكسي الخليك
PE20080188A1 (es) 2006-04-18 2008-03-10 Janssen Pharmaceutica Nv Derivados del acido benzoazepin-oxi-acetico como agonistas de ppar-delta usados para aumentar hdl-c, reducir ldl-c y reducir colesterol
ES2745411T3 (es) * 2006-07-27 2020-03-02 Wang Nai Fang Compuestos y composiciones de arilsulfanilo para administración de agentes activos
JP5305818B2 (ja) * 2008-10-03 2013-10-02 キヤノン株式会社 生体情報取得装置
JP5669889B2 (ja) * 2013-06-27 2015-02-18 キヤノン株式会社 生体情報取得装置
CN106179111B (zh) * 2016-07-16 2018-08-14 江南大学 一种由羧酸盐阴离子表面活性剂和二聚季铵盐形成的粘弹溶液

Family Cites Families (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1121722A (en) * 1966-03-31 1968-07-31 Ici Ltd New carboxylic acid derivatives
US3663540A (en) * 1970-06-19 1972-05-16 R & L Molecular Research Ltd 7 - (p-aminomethylphenylthio)acetamido-3 -(pyridiniummethyl)ceph - 3 - em - 4-carboxylate
US3965093A (en) * 1971-09-24 1976-06-22 E. R. Squibb & Sons, Inc. 6-Arylthio penicillanic acid and derivatives thereof
GB1422679A (en) * 1972-11-16 1976-01-28 Funai Pharmaceutical Ind Ltd Substituted phenoxy-a-methylpropionic acid derivatives and a process for producing the same
FR2285859A1 (fr) * 1974-09-30 1976-04-23 Lafon Labor Phenylsulfinyl-amidines et derives
DE2861187D1 (en) * 1977-07-07 1981-12-24 Ciba Geigy Ag Phenoxy-phenylsulfinyl-and-sulfonylalkanecarboxylic acid derivatives, method for their preparation and their use as herbicides and plant growth regulators.
JPH0311045A (ja) * 1989-06-08 1991-01-18 Hodogaya Chem Co Ltd ベンズアミド誘導体
JPH06234732A (ja) * 1992-09-10 1994-08-23 Banyu Pharmaceut Co Ltd 置換アセトアミド誘導体
FR2700166B1 (fr) * 1993-01-07 1995-02-17 Rhone Poulenc Rorer Sa Dérivés de pyrrolidine, leur préparation et les médicaments les contenant.
JP3583529B2 (ja) * 1995-12-04 2004-11-04 富士写真フイルム株式会社 ハロゲン化銀感光材料
JP2002515865A (ja) * 1996-02-02 2002-05-28 メルク エンド カンパニー インコーポレーテッド 抗糖尿病薬
AU4050797A (en) 1996-08-02 1998-02-25 Ligand Pharmaceuticals Incorporated Prevention or treatment of type 2 diabetes or cardiovascular disease with ppar modulators
US6197791B1 (en) * 1997-02-27 2001-03-06 American Cyanamid Company N-hdroxy-2-(alkyl, aryl, or heteroaryl, sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
US6294573B1 (en) * 1997-08-06 2001-09-25 Abbott Laboratories Reverse hydroxamate inhibitors of matrix metalloproteinases
JP4033630B2 (ja) * 1998-06-22 2008-01-16 バジリア ファルマスーチカ アーゲー プロペニルセファロスポリン誘導体
JP4618845B2 (ja) * 1999-06-09 2011-01-26 杏林製薬株式会社 ヒトペルオキシゾーム増殖薬活性化受容体(PPAR)αアゴニストとしての置換フェニルプロピオン酸誘導体
DE19940415A1 (de) * 1999-08-26 2001-03-08 Friedrich Spener Verzweigtkettige Fettsäuren als fettabbauende Wirkstoffe
US6525093B1 (en) * 1999-11-08 2003-02-25 Calyx Therapeutics Inc. Compounds to treat diabetes and associated conditions
CN1396904A (zh) * 2000-01-28 2003-02-12 诺沃挪第克公司 新颖的化合物、它们的制备和用途
WO2001079150A1 (en) * 2000-04-17 2001-10-25 Novo Nordisk A/S New compounds, their preparation and use
PT1285908E (pt) * 2000-05-29 2008-12-04 Kyorin Seiyaku Kk Derivados do ácido fenilpropiónico substituídos
JP2004509084A (ja) * 2000-08-23 2004-03-25 イーライ・リリー・アンド・カンパニー オキサゾリル−アリールオキシ酢酸誘導体およびそのpparアゴニストとしての使用
GB0111523D0 (en) * 2001-05-11 2001-07-04 Glaxo Group Ltd Chemical compounds

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