JP2005508855A5 - - Google Patents
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- Publication number
- JP2005508855A5 JP2005508855A5 JP2002589487A JP2002589487A JP2005508855A5 JP 2005508855 A5 JP2005508855 A5 JP 2005508855A5 JP 2002589487 A JP2002589487 A JP 2002589487A JP 2002589487 A JP2002589487 A JP 2002589487A JP 2005508855 A5 JP2005508855 A5 JP 2005508855A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- aryl
- substituted
- pyrimidine
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH8732001 | 2001-05-14 | ||
| PCT/EP2002/005241 WO2002092603A1 (en) | 2001-05-14 | 2002-05-13 | Oxazolo-and furopyrimidines and their use in medicaments against tumors |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005508855A JP2005508855A (ja) | 2005-04-07 |
| JP2005508855A5 true JP2005508855A5 (cg-RX-API-DMAC10.html) | 2005-07-28 |
| JP4155827B2 JP4155827B2 (ja) | 2008-09-24 |
Family
ID=4544205
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002589487A Expired - Fee Related JP4155827B2 (ja) | 2001-05-14 | 2002-05-13 | オキサゾロ−およびフロピリミジンならびに腫瘍に対する医薬としてのその使用 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US7294633B2 (cg-RX-API-DMAC10.html) |
| EP (1) | EP1390371B1 (cg-RX-API-DMAC10.html) |
| JP (1) | JP4155827B2 (cg-RX-API-DMAC10.html) |
| CN (1) | CN100378107C (cg-RX-API-DMAC10.html) |
| AT (1) | ATE319718T1 (cg-RX-API-DMAC10.html) |
| BR (1) | BR0209645A (cg-RX-API-DMAC10.html) |
| CA (1) | CA2449188A1 (cg-RX-API-DMAC10.html) |
| DE (1) | DE60209721T2 (cg-RX-API-DMAC10.html) |
| DK (1) | DK1390371T3 (cg-RX-API-DMAC10.html) |
| ES (1) | ES2259707T3 (cg-RX-API-DMAC10.html) |
| PT (1) | PT1390371E (cg-RX-API-DMAC10.html) |
| WO (1) | WO2002092603A1 (cg-RX-API-DMAC10.html) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1689753A4 (en) * | 2003-12-04 | 2010-07-07 | Glaxosmithkline Llc | NEW CHEMICAL COMPOUNDS |
| KR20050091462A (ko) * | 2004-03-12 | 2005-09-15 | 한국과학기술연구원 | 푸로피리미딘 화합물 및 이를 포함하는 ｄｄｒ2 티로신키나아제 활성 저해제 |
| JPWO2005095419A1 (ja) * | 2004-04-01 | 2008-02-21 | 武田薬品工業株式会社 | チアゾロピリミジン誘導体 |
| EP1874769B1 (de) | 2005-04-25 | 2011-09-14 | Merck Patent GmbH | Neuartige aza-heterozyklen als kinase-inhibitoren |
| DE102005061170A1 (de) | 2005-12-21 | 2007-07-05 | Bayer Healthcare Ag | Neue, acyclisch substituierte Furopyrimidin-Derivate und ihre Verwendung |
| DE102005061171A1 (de) | 2005-12-21 | 2007-07-05 | Bayer Healthcare Ag | Neue, cyclisch substituierte Furopyrimidin-Derivate und ihre Verwendung |
| EP3219319A1 (en) * | 2006-06-22 | 2017-09-20 | Nippon Chemiphar Co., Ltd. | Agent for overcoming resistance to anti-cancer agent |
| DE102007019691A1 (de) | 2007-04-26 | 2008-10-30 | Bayer Healthcare Ag | Verwendung von acyclisch substituierten Furopyrimidin-Derivaten zur Behandlung der pulmonalen arteriellen Hypertonie |
| DE102007019690A1 (de) | 2007-04-26 | 2008-10-30 | Bayer Healthcare Ag | Verwendung von cyclisch substituierten Furopyrimidin-Derivaten zur Behandlung der pulmonalen arteriellen Hypertonie |
| DE102007027799A1 (de) | 2007-06-16 | 2008-12-18 | Bayer Healthcare Ag | Substituierte Furopyrimidine und ihre Verwendung |
| DE102007027800A1 (de) | 2007-06-16 | 2008-12-18 | Bayer Healthcare Ag | Substituierte bicyclische Heteroaryl-Verbindungen und ihre Verwendung |
| RU2345996C1 (ru) * | 2007-07-17 | 2009-02-10 | Андрей Александрович Иващенко | Аннелированные азагетероциклические амиды, включающие пиримидиновый фрагмент, способ их получения и применения |
| EP2318415B1 (en) * | 2008-07-15 | 2013-02-20 | Sanofi | Oxazolopyrimidines as edg-1 receptor agonists |
| UY32240A (es) | 2008-11-14 | 2010-06-30 | Boeringer Ingelheim Kg | Nuevas 2,4-diaminopirimidinas, sus sales farmacéuticamente aceptables, composiciones conteniéndolas y aplicaciones. |
| CN101899057A (zh) * | 2010-07-21 | 2010-12-01 | 中国药科大学 | 嘧啶并噁唑衍生物的一种制备方法及其在医学上的用途 |
| US8907093B2 (en) * | 2011-07-07 | 2014-12-09 | Sanofi | Carboxylic acid derivatives having an oxazolo[4,5-c]pyridine ring |
| US8580816B2 (en) * | 2011-07-07 | 2013-11-12 | Sanofi | Carboxylic acid derivatives having an oxazolo[5,4-b]pyridine ring |
| CN103087077B (zh) * | 2011-11-03 | 2016-05-18 | 上海希迈医药科技有限公司 | 噻吩并嘧啶和呋喃并嘧啶类衍生物、其制备方法及其在医药上的应用 |
| CN103360407B (zh) * | 2012-04-10 | 2016-06-22 | 上海希迈医药科技有限公司 | 一种噻吩并嘧啶类衍生物、其制备方法及其在医药上的应用 |
| WO2015162518A1 (en) | 2014-04-25 | 2015-10-29 | Pfizer Inc. | Heteroaromatic compounds and their use as dopamine d1 ligands |
| CN104650111A (zh) * | 2015-01-14 | 2015-05-27 | 中国药科大学 | 芳基脲及芳基酰胺取代的噁唑并嘧啶类化合物及其制备和应用 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5137879A (en) | 1990-03-30 | 1992-08-11 | Dowelanco | Furopyrimidin-4-imine derivatives |
| US5227387A (en) * | 1991-09-03 | 1993-07-13 | Dowelanco | Quinoline nematicidal method |
| ES2109796T3 (es) | 1994-05-03 | 1998-01-16 | Ciba Geigy Ag | Derivados de pirrolopirimidilo con efecto antiproliferante. |
| JPH1184248A (ja) * | 1997-09-12 | 1999-03-26 | Nikon Corp | 反射屈折縮小光学系 |
| KR100600550B1 (ko) * | 2000-10-20 | 2006-07-13 | 에자이 가부시키가이샤 | 질소 함유 방향환 유도체 |
-
2002
- 2002-05-13 CA CA002449188A patent/CA2449188A1/en not_active Abandoned
- 2002-05-13 BR BR0209645-5A patent/BR0209645A/pt not_active IP Right Cessation
- 2002-05-13 AT AT02740590T patent/ATE319718T1/de active
- 2002-05-13 ES ES02740590T patent/ES2259707T3/es not_active Expired - Lifetime
- 2002-05-13 DE DE60209721T patent/DE60209721T2/de not_active Expired - Lifetime
- 2002-05-13 EP EP02740590A patent/EP1390371B1/en not_active Expired - Lifetime
- 2002-05-13 CN CNB028100026A patent/CN100378107C/zh not_active Expired - Fee Related
- 2002-05-13 WO PCT/EP2002/005241 patent/WO2002092603A1/en not_active Ceased
- 2002-05-13 DK DK02740590T patent/DK1390371T3/da active
- 2002-05-13 JP JP2002589487A patent/JP4155827B2/ja not_active Expired - Fee Related
- 2002-05-13 US US10/476,818 patent/US7294633B2/en not_active Expired - Fee Related
- 2002-05-13 PT PT02740590T patent/PT1390371E/pt unknown
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