JP2005507932A - 肥満の処置のためのフェニル置換5−員窒素含有複素環 - Google Patents

肥満の処置のためのフェニル置換5−員窒素含有複素環 Download PDF

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JP2005507932A
JP2005507932A JP2003539676A JP2003539676A JP2005507932A JP 2005507932 A JP2005507932 A JP 2005507932A JP 2003539676 A JP2003539676 A JP 2003539676A JP 2003539676 A JP2003539676 A JP 2003539676A JP 2005507932 A JP2005507932 A JP 2005507932A
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コイシユ,フイリツプ・デイ・ジー
オコナー,ステイーブン・ジエイ
ウイケンス,フイリツプ
ツアング,チエンツイー
ツアング,ハイ−ジユン
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バイエル・フアーマシユーチカルズ・コーポレーシヨン
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JP2003539676A 2001-10-12 2002-10-15 肥満の処置のためのフェニル置換5−員窒素含有複素環 Withdrawn JP2005507932A (ja)

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US32923601P 2001-10-12 2001-10-12
PCT/US2002/032895 WO2003037332A1 (en) 2001-10-12 2002-10-15 Phenyl substituted 5-membered nitrogen containing heterocycles for the treatment of obesity

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JP2005507932A true JP2005507932A (ja) 2005-03-24
JP2005507932A5 JP2005507932A5 (enExample) 2006-01-05

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US (1) US20050014805A1 (enExample)
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CA (1) CA2463441A1 (enExample)
DE (1) DE60208815T2 (enExample)
ES (1) ES2256560T3 (enExample)
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Cited By (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007052843A1 (ja) * 2005-11-04 2007-05-10 Takeda Pharmaceutical Company Limited 複素環アミド化合物およびその用途
JP2016512209A (ja) * 2013-03-13 2016-04-25 エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト ベンゾオキサゼピン化合物の作製方法
JP2018500286A (ja) * 2014-10-30 2018-01-11 ヤンセン ファーマシューティカ エヌ.ベー. RORγtのモジュレーターとしてのアミド置換チアゾール
JP2019506415A (ja) * 2016-02-11 2019-03-07 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 有害生物防除剤としての置換2−(ヘタ)アリール−イミダゾリル−カルボキサミド類
US10975037B2 (en) 2018-06-18 2021-04-13 Janssen Pharmaceutica Nv Phenyl substituted pyrazoles as modulators of RORγt
US10975068B2 (en) 2016-04-27 2021-04-13 Janssen Pharmaceutica Nv 6-aminopyridin-3-yl thiazoles as modulators of RORγT
US10975057B2 (en) 2018-06-18 2021-04-13 Janssen Pharmaceutica Nv 6-aminopyridin-3-yl pyrazoles as modulators of RORgT
US11034658B2 (en) 2018-06-18 2021-06-15 Janssen Pharmaceutica Nv Pyridinyl pyrazoles as modulators of RORγT
US11345666B2 (en) 2018-06-18 2022-05-31 Janssen Pharmaceutica Nv Phenyl and pyridinyl substituted imidazoles as modulators of RORγT

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AU2002319627A1 (en) 2001-07-20 2003-03-03 Merck And Co., Inc. Substituted imidazoles as cannabinoid receptor modulators
NZ534757A (en) 2002-03-12 2006-07-28 Merck & Co Inc Substituted amides
AU2003299791A1 (en) * 2002-12-20 2004-07-22 Bayer Pharmaceuticals Corporation Substituted 3,5-dihydro-4h-imidazol-4-ones for the treatment of obesity
US7772188B2 (en) 2003-01-28 2010-08-10 Ironwood Pharmaceuticals, Inc. Methods and compositions for the treatment of gastrointestinal disorders
AU2004210711B2 (en) * 2003-02-12 2010-07-08 Transtech Pharma, Inc. Substituted azole derivatives as therapeutic agents
WO2004099157A1 (en) * 2003-05-07 2004-11-18 Pfizer Products Inc. Cannabinoid receptor ligands and uses thereof
NZ619746A (en) 2003-08-06 2014-05-30 Senomyx Inc Novel flavors, flavor modifiers, tastants, taste enhancers, umami or sweet tastants, and/or enhancers and use thereof
JP4436369B2 (ja) 2004-01-28 2010-03-24 エフ.ホフマン−ラ ロシュ アーゲー スピロ−ベンゾジオキソール類およびそれらのcb1アンタゴニストとしての使用
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