DE60208815T2 - Phenyl substituierte 5-gliedrige stickstoff enthaltende heterocyclen zur behandlung von fettleibigkeit - Google Patents

Phenyl substituierte 5-gliedrige stickstoff enthaltende heterocyclen zur behandlung von fettleibigkeit Download PDF

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Publication number
DE60208815T2
DE60208815T2 DE60208815T DE60208815T DE60208815T2 DE 60208815 T2 DE60208815 T2 DE 60208815T2 DE 60208815 T DE60208815 T DE 60208815T DE 60208815 T DE60208815 T DE 60208815T DE 60208815 T2 DE60208815 T2 DE 60208815T2
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alkyl
group
formula
hydrogen
optionally substituted
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DE60208815D1 (de
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D. Philip New Haven COISH
J. Stephen Guilford O'CONNOR
Philip Wallingford WICKENS
Chengzhi Orange ZHANG
Hai-Jun Middletown ZHANG
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Bayer Pharmaceuticals Corp
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    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D231/18—One oxygen or sulfur atom
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    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Organic Chemistry (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
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  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
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  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Emergency Medicine (AREA)
  • Gynecology & Obstetrics (AREA)
  • Anesthesiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Gastroenterology & Hepatology (AREA)
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  • Pregnancy & Childbirth (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
DE60208815T 2001-10-12 2002-10-15 Phenyl substituierte 5-gliedrige stickstoff enthaltende heterocyclen zur behandlung von fettleibigkeit Expired - Fee Related DE60208815T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US32923601P 2001-10-12 2001-10-12
US329236P 2001-10-12
PCT/US2002/032895 WO2003037332A1 (en) 2001-10-12 2002-10-15 Phenyl substituted 5-membered nitrogen containing heterocycles for the treatment of obesity

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Publication Number Publication Date
DE60208815D1 DE60208815D1 (de) 2006-04-06
DE60208815T2 true DE60208815T2 (de) 2006-07-20

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US (1) US20050014805A1 (enExample)
EP (1) EP1435951B1 (enExample)
JP (1) JP2005507932A (enExample)
CA (1) CA2463441A1 (enExample)
DE (1) DE60208815T2 (enExample)
ES (1) ES2256560T3 (enExample)
MX (1) MXPA04002931A (enExample)
WO (1) WO2003037332A1 (enExample)

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