DE60208815T2 - Phenyl substituierte 5-gliedrige stickstoff enthaltende heterocyclen zur behandlung von fettleibigkeit - Google Patents

Phenyl substituierte 5-gliedrige stickstoff enthaltende heterocyclen zur behandlung von fettleibigkeit Download PDF

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DE60208815T2
DE60208815T2 DE60208815T DE60208815T DE60208815T2 DE 60208815 T2 DE60208815 T2 DE 60208815T2 DE 60208815 T DE60208815 T DE 60208815T DE 60208815 T DE60208815 T DE 60208815T DE 60208815 T2 DE60208815 T2 DE 60208815T2
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alkyl
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formula
hydrogen
optionally substituted
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DE60208815D1 (de
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D. Philip New Haven COISH
J. Stephen Guilford O'CONNOR
Philip Wallingford WICKENS
Chengzhi Orange ZHANG
Hai-Jun Middletown ZHANG
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Bayer Pharmaceuticals Corp
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    • C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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DE60208815T 2001-10-12 2002-10-15 Phenyl substituierte 5-gliedrige stickstoff enthaltende heterocyclen zur behandlung von fettleibigkeit Expired - Fee Related DE60208815T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US32923601P 2001-10-12 2001-10-12
US329236P 2001-10-12
PCT/US2002/032895 WO2003037332A1 (en) 2001-10-12 2002-10-15 Phenyl substituted 5-membered nitrogen containing heterocycles for the treatment of obesity

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Publication Number Publication Date
DE60208815D1 DE60208815D1 (de) 2006-04-06
DE60208815T2 true DE60208815T2 (de) 2006-07-20

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US (1) US20050014805A1 (enExample)
EP (1) EP1435951B1 (enExample)
JP (1) JP2005507932A (enExample)
CA (1) CA2463441A1 (enExample)
DE (1) DE60208815T2 (enExample)
ES (1) ES2256560T3 (enExample)
MX (1) MXPA04002931A (enExample)
WO (1) WO2003037332A1 (enExample)

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WO2004058727A1 (en) * 2002-12-20 2004-07-15 Bayer Pharmaceuticals Corporation Substituted 3,5-dihydro-4h-imidazol-4-ones for the treatment of obesity
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JP2006518738A (ja) * 2003-02-12 2006-08-17 トランス　テック　ファーマ，インコーポレイテッド 治療薬としての置換アゾール誘導体
EP1622876A1 (en) * 2003-05-07 2006-02-08 Pfizer Products Inc. Cannabinoid receptor ligands and uses thereof
JP2007512227A (ja) 2003-08-06 2007-05-17 セノミックス、インコーポレイテッド Ｔ１ｒヘテロオリゴマー味覚受容体、この受容体を発現する細胞株、および味覚化合物
CN100572375C (zh) 2004-01-28 2009-12-23 霍夫曼-拉罗奇有限公司 螺－苯并间二氧杂环戊烯及其作为cb1拮抗剂的应用
US20050187277A1 (en) * 2004-02-12 2005-08-25 Mjalli Adnan M. Substituted azole derivatives, compositions, and methods of use
WO2005090340A1 (ja) * 2004-03-22 2005-09-29 Banyu Pharmaceutical Co., Ltd. ピペリジン－１－カルボキサミド誘導体
US20080125403A1 (en) 2004-04-02 2008-05-29 Merck & Co., Inc. Method of Treating Men with Metabolic and Anthropometric Disorders
MXPA06012130A (es) * 2004-04-20 2007-01-31 Transtech Pharma Inc Derivados de tiazol y pirimidina substituidos como moduladores del receptor de melanocortina.
BRPI0517653A (pt) 2004-11-09 2008-10-14 Hoffmann La Roche compostos, processo para a sua manufatura, composições farmacêuticas que compreendem os mesmos, método para o tratamento e/ou profilaxia de enfermidades e utilização dos compostos
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