JP2005507873A5 - - Google Patents
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- Publication number
- JP2005507873A5 JP2005507873A5 JP2003521208A JP2003521208A JP2005507873A5 JP 2005507873 A5 JP2005507873 A5 JP 2005507873A5 JP 2003521208 A JP2003521208 A JP 2003521208A JP 2003521208 A JP2003521208 A JP 2003521208A JP 2005507873 A5 JP2005507873 A5 JP 2005507873A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- compound
- formula
- haloalkyl
- independently
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 claims description 40
- 229910052739 hydrogen Inorganic materials 0.000 claims description 21
- 238000000034 method Methods 0.000 claims description 21
- 229910052794 bromium Inorganic materials 0.000 claims description 16
- 229910052801 chlorine Inorganic materials 0.000 claims description 16
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 15
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 10
- 229910052736 halogen Inorganic materials 0.000 claims description 10
- 150000002367 halogens Chemical class 0.000 claims description 10
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 claims description 6
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims description 5
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims description 5
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 5
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 5
- 125000006656 (C2-C4) alkenyl group Chemical group 0.000 claims description 5
- 125000006650 (C2-C4) alkynyl group Chemical group 0.000 claims description 5
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims description 5
- -1 C 1 -C 4 alkylthio Chemical group 0.000 claims description 5
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 5
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims description 5
- 125000000217 alkyl group Chemical group 0.000 claims description 5
- 125000006310 cycloalkyl amino group Chemical group 0.000 claims description 5
- 125000004663 dialkyl amino group Chemical group 0.000 claims description 5
- 125000004473 dialkylaminocarbonyl group Chemical group 0.000 claims description 5
- 238000004519 manufacturing process Methods 0.000 claims description 4
- 150000004703 alkoxides Chemical class 0.000 claims description 3
- 230000002152 alkylating effect Effects 0.000 claims description 3
- 239000003795 chemical substances by application Substances 0.000 claims description 3
- 239000002253 acid Substances 0.000 claims description 2
- 230000015572 biosynthetic process Effects 0.000 description 1
- 229910052731 fluorine Inorganic materials 0.000 description 1
- 229910052740 iodine Inorganic materials 0.000 description 1
- 125000001453 quaternary ammonium group Chemical group 0.000 description 1
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US31191901P | 2001-08-13 | 2001-08-13 | |
| US34189401P | 2001-12-19 | 2001-12-19 | |
| US36965902P | 2002-04-02 | 2002-04-02 | |
| PCT/US2002/025612 WO2003016282A2 (en) | 2001-08-13 | 2002-08-13 | Substituted 1h-dihydropyrazoles, their preparation and use |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005507873A JP2005507873A (ja) | 2005-03-24 |
| JP2005507873A5 true JP2005507873A5 (https=) | 2006-01-05 |
| JP4448327B2 JP4448327B2 (ja) | 2010-04-07 |
Family
ID=27405543
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003521208A Expired - Fee Related JP4448327B2 (ja) | 2001-08-13 | 2002-08-13 | 新規置換１ｈ−ジヒドロピラゾール、それらの製造および使用 |
Country Status (8)
| Country | Link |
|---|---|
| US (3) | US7038057B2 (https=) |
| EP (1) | EP1417200B1 (https=) |
| JP (1) | JP4448327B2 (https=) |
| AT (1) | ATE469892T1 (https=) |
| AU (1) | AU2002319814A1 (https=) |
| CA (1) | CA2454298A1 (https=) |
| DE (1) | DE60236600D1 (https=) |
| WO (1) | WO2003016282A2 (https=) |
Families Citing this family (67)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7038057B2 (en) * | 2001-08-13 | 2006-05-02 | E.I. Du Pont De Nemours And Company | Substituted 1H-dihydropyrazoles, their preparation and use |
| AR036872A1 (es) | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| TWI356822B (en) * | 2001-08-13 | 2012-01-21 | Du Pont | Novel substituted dihydro 3-halo-1h-pyrazole-5-car |
| TWI312274B (en) * | 2001-08-13 | 2009-07-21 | Du Pont | Method for controlling particular insect pests by applying anthranilamide compounds |
| AU2002331706B2 (en) * | 2001-08-15 | 2009-01-22 | E.I. Du Pont De Nemours And Company | Ortho-substituted aryl amides for controlling invertebrate pests |
| BR0212183B1 (pt) * | 2001-08-16 | 2014-10-21 | Du Pont | composto de antranilamida substituída, seus n-óxidos e sais, método para o controle de uma praga invertebrada e composição para o controle de uma praga invertebrada |
| TWI283164B (en) * | 2001-09-21 | 2007-07-01 | Du Pont | Anthranilamide arthropodicide treatment |
| US20040110777A1 (en) * | 2001-12-03 | 2004-06-10 | Annis Gary David | Quinazolinones and pyridinylpyrimidinones for controlling invertebrate pests |
| BR0307178A (pt) * | 2002-01-22 | 2004-12-07 | Du Pont | Composto, composição e método para controle de pragas invertebradas |
| BR0311707A (pt) * | 2002-06-13 | 2005-03-15 | Du Pont | Composto, composição e método de controle de pelo menos uma praga invertebrada |
| TWI326283B (en) * | 2002-07-31 | 2010-06-21 | Du Pont | Method for preparing fused oxazinones |
| MXPA05005025A (es) * | 2002-11-15 | 2005-08-03 | Du Pont | Nuevos insecticidas de antranilamida. |
| ES2424840T3 (es) | 2003-01-28 | 2013-10-09 | E.I. Du Pont De Nemours And Company | Insecticidas tipo ciano antranilamida |
| TWI367882B (en) * | 2003-03-26 | 2012-07-11 | Du Pont | Preparation and use of 2-substituted-5-oxo-3-pyrazolidinecarboxylates |
| EP1631564A1 (en) * | 2003-06-12 | 2006-03-08 | E.I. Dupont De Nemours And Company | Method for preparing fused oxazinones |
| DE102004006075A1 (de) | 2003-11-14 | 2005-06-16 | Bayer Cropscience Ag | Wirkstoffkombinationen mit insektiziden Eigenschaften |
| DE10353281A1 (de) | 2003-11-14 | 2005-06-16 | Bayer Cropscience Ag | Wirkstoffkombination mit insektiziden und akariziden Eigenschaften |
| DE102004021564A1 (de) | 2003-11-14 | 2005-07-07 | Bayer Cropscience Ag | Wirkstoffkombinationen mit insektiziden Eigenschaften |
| DE10356550A1 (de) | 2003-12-04 | 2005-07-07 | Bayer Cropscience Ag | Wirkstoffkombinationen mit insektiziden Eigenschaften |
| US20070142327A1 (en) | 2003-12-04 | 2007-06-21 | Bayer Cropscience Aktiengesellschaft | Active compound combinations having insecticidal properties |
| KR20060135881A (ko) * | 2004-04-13 | 2006-12-29 | 이 아이 듀폰 디 네모아 앤드 캄파니 | 안트라닐아미드 살충제 |
| DE102004031100A1 (de) * | 2004-06-28 | 2006-01-12 | Bayer Cropscience Ag | Anthranilamide |
| GT200500179AA (es) | 2004-07-01 | 2008-10-29 | Mezclas sinergistas de agentes de antranilamida para el control de plagas de invertebrados | |
| JP4920878B2 (ja) * | 2004-07-14 | 2012-04-18 | 日本電気株式会社 | 認証システム、ネットワーク集線装置及びそれらに用いる認証方法並びにそのプログラム |
| DE102004035134A1 (de) | 2004-07-20 | 2006-02-16 | Bayer Cropscience Ag | Selektive Insektizide auf Basis von Halogenalkylnicotinsäurederivaten, Anthranilsäureamiden oder Phthalsäurediamiden und Safenern |
| MY140912A (en) * | 2004-07-26 | 2010-01-29 | Du Pont | Mixtures of anthranilamide invertebrate pest control agents |
| AU2005306363B2 (en) * | 2004-11-18 | 2012-08-09 | E. I. Du Pont De Nemours And Company | Anthranilamide insecticides |
| AU2006283181A1 (en) * | 2005-08-24 | 2007-03-01 | E. I. Du Pont De Nemours And Company | Anthranilamides for controlling invertebrate pests |
| DE102005044108A1 (de) | 2005-09-15 | 2007-03-29 | Bayer Cropscience Ag | Dioxazin- und Oxdiazin-substituierte Arylamide |
| DE102006032168A1 (de) | 2006-06-13 | 2007-12-20 | Bayer Cropscience Ag | Anthranilsäurediamid-Derivate mit heteroaromatischen Substituenten |
| DE102006030710A1 (de) * | 2006-07-03 | 2008-01-10 | Bayer Cropscience Ag | Synergistische insektizide und fungizide Mischungen |
| WO2008031548A1 (en) * | 2006-09-11 | 2008-03-20 | Syngenta Participations Ag | Process for the preparation of anthranilamide derivatives |
| AR064249A1 (es) * | 2006-11-17 | 2009-03-25 | Basf Ag | Metodo para incrementar la biomasa seca de plantas |
| CN104496901B (zh) * | 2006-12-15 | 2016-05-25 | 石原产业株式会社 | 邻氨基苯甲酰胺系化合物的制造方法 |
| JP5507045B2 (ja) * | 2006-12-15 | 2014-05-28 | 石原産業株式会社 | アントラニルアミド系化合物の製造方法 |
| JP2009001541A (ja) * | 2006-12-15 | 2009-01-08 | Ishihara Sangyo Kaisha Ltd | 新規ピラゾール化合物を中間体として用いるアントラニルアミド系化合物の製造方法 |
| TWI415827B (zh) | 2006-12-21 | 2013-11-21 | Du Pont | 製備２-胺基-５-氰基苯甲酸衍生物之方法 |
| RS52042B (sr) * | 2007-04-25 | 2012-04-30 | Syngenta Participations Ag | Fungicidne smeše |
| WO2009010260A2 (en) * | 2007-07-16 | 2009-01-22 | Syngenta Participations Ag | Condensed anthranilamide insecticides |
| EP2100883A1 (de) * | 2008-03-10 | 2009-09-16 | Bayer CropScience AG | Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4carbonsäure-Derivaten |
| MX2011006319A (es) | 2008-12-18 | 2011-06-24 | Bayer Cropscience Ag | Amidas del acido antranilico sustituidas con tetrazol como plaguicidas. |
| EP2243777A1 (de) * | 2009-04-03 | 2010-10-27 | Bayer CropScience AG | Verfahren zum Herstellen von Pyridyl-substituierten Pyrazolen |
| JP5872467B2 (ja) * | 2009-07-23 | 2016-03-01 | バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ ＧｍｂＨ | アリール置換ピラゾールの調製方法 |
| BR112012014683B1 (pt) | 2009-12-15 | 2017-11-07 | Bayer Cropscience Ag | Process for the production of 5-pyrazolcarboxylic acid derivatives 1-alkyl- / 1-aryl-substituted and compound acid |
| BR112012019973B1 (pt) | 2010-02-09 | 2019-02-05 | Bayer Cropscience Ag | Derivados de ácido antranílico hidrazina-substituídos, misturas, compostos precursores,composições agroquímicas, processos para preparação dos referidos compostos e composições, uso dos compostos, das misturas ou das composições, e método para o controle de pragas animais |
| BR112012026523B1 (pt) | 2010-04-16 | 2018-11-27 | Bayer Intellectual Property Gmbh | antranilamidas substituídas com triazol, composições agroquímicas para controlar insetos prejudiciais e composições para controlar insetos prejudiciais as compreendendo, seu processo para preparar composições agroquímicas e uso, bem como método para controlar pragas animais ou fungos fitopatogênicos |
| MX2012014958A (es) | 2010-06-15 | 2013-02-12 | Bayer Ip Gmbh | Derivados de diamida antranilica. |
| CN103068814B (zh) | 2010-06-15 | 2015-11-25 | 拜耳知识产权有限责任公司 | 邻氨基苯甲酸衍生物 |
| CN103068820A (zh) | 2010-06-15 | 2013-04-24 | 拜耳知识产权有限责任公司 | 新的邻位取代的芳基酰胺衍生物 |
| CN103249729B (zh) | 2010-06-15 | 2017-04-05 | 拜耳知识产权有限责任公司 | 具有环状侧链的邻甲酰胺基苯甲酰胺衍生物 |
| BR112013000583B1 (pt) | 2010-07-09 | 2018-06-12 | Bayer Intellectual Property Gmbh | Derivados de antranilamida como pesticidas, misturas dos referidos compostos, processo para preparar os compostos, composições, composições agroquímicas, processo para produzir as composições agroquímicas, uso do composto e método para controlar pragas animais |
| US8871939B2 (en) | 2011-01-28 | 2014-10-28 | E I Du Pont De Nemours And Company | Method for preparing 2-aminobenzamide derivatives |
| WO2013092519A1 (en) | 2011-12-19 | 2013-06-27 | Bayer Cropscience Ag | Use of anthranilic acid diamide derivatives for pest control in transgenic crops |
| EP2606732A1 (en) | 2011-12-19 | 2013-06-26 | Bayer CropScience AG | Use of an anthranilic diamide derivatives with heteroaromatic and heterocyclic substituents in combination with a biological control agent |
| CA2894399A1 (en) | 2012-12-06 | 2014-06-12 | Quanticel Pharmaceuticals, Inc. | Histone demethylase inhibitors |
| BR112015020830A2 (pt) | 2013-03-06 | 2017-07-18 | Bayer Cropscience Ag | diamidas de ácido antranílico substituídas com alcoximino como pesticidas |
| MX2015017640A (es) * | 2013-06-20 | 2016-09-07 | Basf Se | Proceso para preparar compuestos de piridilpirazol y sus derivados de piridilhidrazina. |
| CN103467380B (zh) * | 2013-09-29 | 2015-06-24 | 南开大学 | 一类取代苯基吡唑酰胺衍生物及其制备方法和应用 |
| KR102736869B1 (ko) | 2014-03-07 | 2024-12-02 | 바이오크리스트파마슈티컬즈,인코포레이티드 | 인간 혈장 칼리크레인 저해제 |
| CN109689629B (zh) * | 2016-09-21 | 2022-11-29 | 拜耳作物科学股份公司 | 制备3-氟烷基-5-吡唑羧酸酯和3-氟烷基-5-吡唑羧酸的方法 |
| BR112020012455B1 (pt) | 2017-12-20 | 2024-04-30 | Pi Industries Ltd | Pirazolopiridina-diamidas, seu uso como inseticida e processos para sua preparação |
| WO2019123194A1 (en) | 2017-12-20 | 2019-06-27 | Pi Industries Ltd. | Anthranilamides, their use as insecticide and processes for preparing the same. |
| JP7307079B2 (ja) | 2018-01-30 | 2023-07-11 | ピーアイ インダストリーズ リミテッド | 新規アントラニルアミド、殺虫剤としてのその使用およびその製造方法 |
| MX2020011671A (es) | 2018-05-21 | 2020-12-10 | Pi Industries Ltd | Nuevo proceso para la preparacion de diamidas antranilicas. |
| KR102790425B1 (ko) | 2018-07-20 | 2025-04-04 | 피아이 인더스트리스 엘티디. | 안트라닐산 디아미드의 새로운 제조 방법 |
| CN114206839B (zh) * | 2019-08-06 | 2025-03-07 | 拜奥克里斯特制药公司 | 血浆激肽释放酶抑制剂的生产规模合成 |
| US12010989B2 (en) | 2019-11-07 | 2024-06-18 | S. C. Johnson & Son, Inc. | Roach gel formulations |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL121416C (https=) | 1961-05-31 | |||
| BR8707672A (pt) | 1987-01-05 | 1989-10-03 | Du Pont | Pirazolinas inseticidas |
| US5091405A (en) | 1987-01-05 | 1992-02-25 | E. I. Du Pont De Nemours And Company | Insecticidal pyrazolines |
| DE3808896A1 (de) | 1988-03-17 | 1989-09-28 | Hoechst Ag | Pflanzenschuetzende mittel auf basis von pyrazolcarbonsaeurederivaten |
| NL9202078A (nl) * | 1992-11-30 | 1994-06-16 | Rijkslandbouwhogeschool | Nieuwe N-acyl-antranilzuurverbindingen en toepassing van N-acyl-antranilzuurverbindingen bij de bestrijding van insecten. |
| US5945641A (en) * | 1998-07-15 | 1999-08-31 | Shieh; Woei-Kang | Stethoscope structure |
| MXPA01008142A (es) | 1999-02-10 | 2003-07-21 | Welfide Corp | Compuestos de amida, y uso medicinal de los mismos. |
| DE19951360A1 (de) * | 1999-10-26 | 2001-05-03 | Aventis Pharma Gmbh | Substituierte Indole |
| MY138097A (en) | 2000-03-22 | 2009-04-30 | Du Pont | Insecticidal anthranilamides |
| AU2002227243A1 (en) | 2000-12-11 | 2002-06-24 | E.I. Du Pont De Nemours And Company | Quinazolinones and pyridinopyrimidinones for controlling invertebrate pests |
| JP2004515547A (ja) | 2000-12-11 | 2004-05-27 | イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー | 置換複素環式フタル酸ジアミド殺節足動物剤 |
| AR036872A1 (es) | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| US7038057B2 (en) * | 2001-08-13 | 2006-05-02 | E.I. Du Pont De Nemours And Company | Substituted 1H-dihydropyrazoles, their preparation and use |
| TWI356822B (en) * | 2001-08-13 | 2012-01-21 | Du Pont | Novel substituted dihydro 3-halo-1h-pyrazole-5-car |
| BR0212183B1 (pt) | 2001-08-16 | 2014-10-21 | Du Pont | composto de antranilamida substituída, seus n-óxidos e sais, método para o controle de uma praga invertebrada e composição para o controle de uma praga invertebrada |
| US20040110777A1 (en) * | 2001-12-03 | 2004-06-10 | Annis Gary David | Quinazolinones and pyridinylpyrimidinones for controlling invertebrate pests |
| US20040063738A1 (en) * | 2001-12-05 | 2004-04-01 | Lahm George Philip | Substituted heterocyclic phthalic acid diamide arthropodicides |
| TW200401641A (en) | 2002-07-18 | 2004-02-01 | Wyeth Corp | 1-Heterocyclylalkyl-3-sulfonylindole or-indazole derivatives as 5-hydroxytryptamine-6 ligands |
| TWI343376B (en) * | 2002-07-31 | 2011-06-11 | Du Pont | Method for preparing 3-halo-4, 5-dihydro-1h-pyrazoles |
| GB0409785D0 (en) | 2004-04-30 | 2004-06-09 | Resolution Chemicals Ltd | Preparation of cabergoline |
-
2002
- 2002-08-13 US US10/482,556 patent/US7038057B2/en not_active Expired - Fee Related
- 2002-08-13 JP JP2003521208A patent/JP4448327B2/ja not_active Expired - Fee Related
- 2002-08-13 CA CA002454298A patent/CA2454298A1/en not_active Abandoned
- 2002-08-13 EP EP02750482A patent/EP1417200B1/en not_active Expired - Lifetime
- 2002-08-13 DE DE60236600T patent/DE60236600D1/de not_active Expired - Lifetime
- 2002-08-13 WO PCT/US2002/025612 patent/WO2003016282A2/en not_active Ceased
- 2002-08-13 AT AT02750482T patent/ATE469892T1/de not_active IP Right Cessation
- 2002-08-13 AU AU2002319814A patent/AU2002319814A1/en not_active Abandoned
-
2006
- 2006-02-13 US US11/352,805 patent/US7622595B2/en not_active Expired - Fee Related
-
2009
- 2009-10-13 US US12/578,227 patent/US7932395B2/en not_active Expired - Fee Related
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