JP2004536066A5 - - Google Patents

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Publication number
JP2004536066A5
JP2004536066A5 JP2002591462A JP2002591462A JP2004536066A5 JP 2004536066 A5 JP2004536066 A5 JP 2004536066A5 JP 2002591462 A JP2002591462 A JP 2002591462A JP 2002591462 A JP2002591462 A JP 2002591462A JP 2004536066 A5 JP2004536066 A5 JP 2004536066A5
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JP
Japan
Prior art keywords
methyl
pyrrolidin
alkyl
hydrogen
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2002591462A
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English (en)
Japanese (ja)
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JP2004536066A (ja
JP3715280B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/EP2002/005120 external-priority patent/WO2002094789A1/en
Publication of JP2004536066A publication Critical patent/JP2004536066A/ja
Publication of JP2004536066A5 publication Critical patent/JP2004536066A5/ja
Application granted granted Critical
Publication of JP3715280B2 publication Critical patent/JP3715280B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2002591462A 2001-05-21 2002-05-08 ニューロペプチドｙレセプターのリガンドとしてのキノリン誘導体 Expired - Fee Related JP3715280B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01112370 2001-05-21
PCT/EP2002/005120 WO2002094789A1 (en) 2001-05-21 2002-05-08 Quinoline derivatives as ligands for the neuropeptide y receptor

Publications (3)

Publication Number Publication Date
JP2004536066A JP2004536066A (ja) 2004-12-02
JP2004536066A5 true JP2004536066A5 (https=) 2005-08-25
JP3715280B2 JP3715280B2 (ja) 2005-11-09

Family

ID=8177497

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002591462A Expired - Fee Related JP3715280B2 (ja) 2001-05-21 2002-05-08 ニューロペプチドｙレセプターのリガンドとしてのキノリン誘導体

Country Status (19)

Country Link
US (2) US6818767B2 (https=)
EP (1) EP1395564B1 (https=)
JP (1) JP3715280B2 (https=)
KR (1) KR100621287B1 (https=)
CN (1) CN100376557C (https=)
AR (1) AR035979A1 (https=)
AT (1) ATE387428T1 (https=)
AU (1) AU2002338896B2 (https=)
BR (1) BR0209957A (https=)
CA (1) CA2446324A1 (https=)
DE (1) DE60225274T2 (https=)
ES (1) ES2300478T3 (https=)
GT (1) GT200200090A (https=)
MX (1) MXPA03010565A (https=)
PA (1) PA8545301A1 (https=)
PE (1) PE20021155A1 (https=)
UY (1) UY27300A1 (https=)
WO (1) WO2002094789A1 (https=)
ZA (1) ZA200308783B (https=)

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EP1921065B1 (en) 2005-08-24 2010-10-20 Banyu Pharmaceutical Co., Ltd. Phenylpyridone derivative
WO2007029847A1 (ja) 2005-09-07 2007-03-15 Banyu Pharmaceutical Co., Ltd. 二環性芳香族置換ピリドン誘導体
AU2006307046A1 (en) 2005-10-27 2007-05-03 Msd K.K. Novel benzoxathiin derivative
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AU2007301126A1 (en) 2006-09-28 2008-04-03 Banyu Pharmaceutical Co., Ltd. Diaryl ketimine derivative
CA2682727C (en) 2007-04-02 2016-03-22 Banyu Pharmaceutical Co., Ltd. Indoledione derivative
WO2008141077A1 (en) * 2007-05-10 2008-11-20 Janssen Pharmaceutica N.V. Process for the preparation of tetrahydroquinolinyl, benzoxazine and benzothiazine derivatives
PL2182950T3 (pl) 2007-05-17 2018-01-31 Helperby Therapeutics Ltd Zastosowanie związków 4-(pirolidyn-1-ylo)chinolinowych do zabijania klinicznie latentnych drobnoustrojów
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US8969514B2 (en) 2007-06-04 2015-03-03 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
EP2527360B1 (en) 2007-06-04 2015-10-28 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
CA2705318C (en) 2007-11-15 2013-12-31 Boehringer Ingelheim International Gmbh Inhibitors of human immunodeficiency virus replication
MX2010005334A (es) 2007-11-16 2010-05-27 Boehringer Ingelheim Int Inhibidores de la replicacion del virus de la inmunodeficiencia humana.
US20110015181A1 (en) 2008-03-06 2011-01-20 Makoto Ando Alkylaminopyridine derivative
EP2272841A1 (en) 2008-03-28 2011-01-12 Banyu Pharmaceutical Co., Ltd. Diarylmethylamide derivative having antagonistic activity on melanin-concentrating hormone receptor
EP2810951B1 (en) 2008-06-04 2017-03-15 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
AU2009261248A1 (en) 2008-06-19 2009-12-23 Banyu Pharmaceutical Co., Ltd. Spirodiamine-diarylketoxime derivative
EP3241839B1 (en) 2008-07-16 2019-09-04 Bausch Health Ireland Limited Agonists of guanylate cyclase useful for the treatment of gastrointestinal, inflammation, cancer and other disorders
WO2010013595A1 (ja) 2008-07-30 2010-02-04 萬有製薬株式会社 ５員－５員又は５員－６員縮環シクロアルキルアミン誘導体
WO2010047982A1 (en) 2008-10-22 2010-04-29 Merck Sharp & Dohme Corp. Novel cyclic benzimidazole derivatives useful anti-diabetic agents
JP5557845B2 (ja) 2008-10-31 2014-07-23 メルク・シャープ・アンド・ドーム・コーポレーション 糖尿病用剤として有用な新規環状ベンゾイミダゾール誘導体
US8895596B2 (en) 2010-02-25 2014-11-25 Merck Sharp & Dohme Corp Cyclic benzimidazole derivatives useful as anti-diabetic agents
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