JP2004536066A5 - - Google Patents

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Publication number
JP2004536066A5
JP2004536066A5 JP2002591462A JP2002591462A JP2004536066A5 JP 2004536066 A5 JP2004536066 A5 JP 2004536066A5 JP 2002591462 A JP2002591462 A JP 2002591462A JP 2002591462 A JP2002591462 A JP 2002591462A JP 2004536066 A5 JP2004536066 A5 JP 2004536066A5
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JP
Japan
Prior art keywords
methyl
pyrrolidin
alkyl
hydrogen
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2002591462A
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English (en)
Japanese (ja)
Other versions
JP3715280B2 (ja
JP2004536066A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2002/005120 external-priority patent/WO2002094789A1/en
Publication of JP2004536066A publication Critical patent/JP2004536066A/ja
Publication of JP2004536066A5 publication Critical patent/JP2004536066A5/ja
Application granted granted Critical
Publication of JP3715280B2 publication Critical patent/JP3715280B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2002591462A 2001-05-21 2002-05-08 ニューロペプチドｙレセプターのリガンドとしてのキノリン誘導体 Expired - Fee Related JP3715280B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01112370 2001-05-21
PCT/EP2002/005120 WO2002094789A1 (en) 2001-05-21 2002-05-08 Quinoline derivatives as ligands for the neuropeptide y receptor

Publications (3)

Publication Number Publication Date
JP2004536066A JP2004536066A (ja) 2004-12-02
JP2004536066A5 true JP2004536066A5 (https=) 2005-08-25
JP3715280B2 JP3715280B2 (ja) 2005-11-09

Family

ID=8177497

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002591462A Expired - Fee Related JP3715280B2 (ja) 2001-05-21 2002-05-08 ニューロペプチドｙレセプターのリガンドとしてのキノリン誘導体

Country Status (19)

Country Link
US (2) US6818767B2 (https=)
EP (1) EP1395564B1 (https=)
JP (1) JP3715280B2 (https=)
KR (1) KR100621287B1 (https=)
CN (1) CN100376557C (https=)
AR (1) AR035979A1 (https=)
AT (1) ATE387428T1 (https=)
AU (1) AU2002338896B2 (https=)
BR (1) BR0209957A (https=)
CA (1) CA2446324A1 (https=)
DE (1) DE60225274T2 (https=)
ES (1) ES2300478T3 (https=)
GT (1) GT200200090A (https=)
MX (1) MXPA03010565A (https=)
PA (1) PA8545301A1 (https=)
PE (1) PE20021155A1 (https=)
UY (1) UY27300A1 (https=)
WO (1) WO2002094789A1 (https=)
ZA (1) ZA200308783B (https=)

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WO2007024004A1 (ja) 2005-08-24 2007-03-01 Banyu Pharmaceutical Co., Ltd. フェニルピリドン誘導体
WO2007029847A1 (ja) 2005-09-07 2007-03-15 Banyu Pharmaceutical Co., Ltd. 二環性芳香族置換ピリドン誘導体
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CN101679853B (zh) * 2007-06-01 2013-10-30 E.I.内穆尔杜邦公司 用于绿色发光应用的*
US8969514B2 (en) 2007-06-04 2015-03-03 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
MX354786B (es) 2007-06-04 2018-03-21 Synergy Pharmaceuticals Inc Agonistas de guanilato ciclasa utiles para el tratamiento de trastornos gastrointestinales, inflamacion, cancer y otros trastornos.
ATE541841T1 (de) * 2007-11-15 2012-02-15 Boehringer Ingelheim Int Inhibitoren der replikation des human immunodeficiency virus
EA019259B1 (ru) 2007-11-16 2014-02-28 Джилид Сайенсиз, Инк. Ингибиторы репликации вируса иммунодефицита человека
EP2264026A4 (en) 2008-03-06 2012-03-28 Msd Kk ALKYLAMINOPYRIDINDERIVATE
WO2009119726A1 (ja) 2008-03-28 2009-10-01 萬有製薬株式会社 メラニン凝集ホルモン受容体拮抗作用を有するジアリールメチルアミド誘導体
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JPWO2009154132A1 (ja) 2008-06-19 2011-12-01 Ｍｓｄ株式会社 スピロジアミン−ジアリールケトオキシム誘導体
AU2009270833B2 (en) 2008-07-16 2015-02-19 Bausch Health Ireland Limited Agonists of guanylate cyclase useful for the treatment of gastrointestinal, inflammation, cancer and other disorders
EP2319841A1 (en) 2008-07-30 2011-05-11 Msd K.K. (5-membered)-(5-membered) or (5-membered)-(6-membered) fused ring cycloalkylamine derivative
EP2348857B1 (en) 2008-10-22 2016-02-24 Merck Sharp & Dohme Corp. Novel cyclic benzimidazole derivatives useful anti-diabetic agents
US8329914B2 (en) 2008-10-31 2012-12-11 Merck Sharp & Dohme Corp Cyclic benzimidazole derivatives useful as anti-diabetic agents
JP2013520502A (ja) 2010-02-25 2013-06-06 メルク・シャープ・エンド・ドーム・コーポレイション 有用な抗糖尿病薬である新規な環状ベンズイミダゾール誘導体
US9616097B2 (en) 2010-09-15 2017-04-11 Synergy Pharmaceuticals, Inc. Formulations of guanylate cyclase C agonists and methods of use
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RU2015106909A (ru) 2012-08-02 2016-09-27 Мерк Шарп И Доум Корп. Антидиабетические трициклические соединения
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