|
US1349418A
(en)
*
|
1919-08-05 |
1920-08-10 |
George F Flynn |
Motor-support
|
|
US3590036A
(en)
*
|
1968-11-18 |
1971-06-29 |
George Y Lesher |
Naphthyridine-3-carboxylic acids,their derivatives and preparation thereof
|
|
DE2011970A1
(en)
|
1970-03-13 |
1971-11-18 |
CH. Boehringer Sohn, 6507 Ingelheim |
Imidazo-(1, 2-a)- pyrimidines prepn
|
|
US3635667A
(en)
|
1970-07-23 |
1972-01-18 |
Fmc Corp |
Drycleaning with hydrogen peroxide
|
|
GB1322318A
(en)
*
|
1971-05-19 |
1973-07-04 |
Sterling Drug Inc |
1-alkyl-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acids and esters
|
|
BE786028A
(fr)
|
1971-07-08 |
1973-01-08 |
Boehringer Sohn Ingelheim |
2,3-dihydro-oxo-imidazo(1,2-a)-pyrimidines, leurs sels d'addition avec des acides et procedes pour les fabriquer
|
|
DE2356005A1
(de)
|
1973-11-09 |
1975-05-22 |
Boehringer Sohn Ingelheim |
Neue 7-amino-imidazo eckige klammer auf 1,2-a eckige klammer zu pyrimidine, diese enthaltende arzneimittel sowie verfahren zu deren herstellung
|
|
AU577105B2
(en)
|
1985-04-02 |
1988-09-15 |
T.P.O. :Pharmachim: |
Acylaminic penicillin derivatives
|
|
US6117940A
(en)
|
1997-10-17 |
2000-09-12 |
Mjalli; Adnan M. M. |
Amino-ketone solid support templates
|
|
IL152848A0
(en)
*
|
2000-06-12 |
2003-06-24 |
Eisai Co Ltd |
1,2-dihydropyridine derivatives, pharmaceutical compositions containing the same and methods for the production thereof
|
|
GB0129260D0
(en)
*
|
2001-12-06 |
2002-01-23 |
Eisai London Res Lab Ltd |
Pharmaceutical compositions and their uses
|
|
BR0314759A
(pt)
|
2002-09-26 |
2005-07-26 |
Pfizer |
Derivados de pirazol
|
|
JP2005089352A
(ja)
|
2003-09-16 |
2005-04-07 |
Kissei Pharmaceut Co Ltd |
新規なイミダゾ[1,5−a]ピラジン誘導体、それを含有する医薬組成物およびそれらの用途
|
|
WO2005030791A2
(en)
|
2003-09-23 |
2005-04-07 |
Merck & Co., Inc. |
Isoquinolinone potassium channel inhibitors
|
|
EP1667981A4
(en)
*
|
2003-09-23 |
2008-08-13 |
Merck & Co Inc |
ISOCHINOLINE AS KALIUM CHANNEL INHIBITORS
|
|
KR100703068B1
(ko)
|
2003-12-30 |
2007-04-05 |
에스케이케미칼주식회사 |
피리딘 유도체와 이의 제조방법, 및 이를 포함하는약제조성물
|
|
TW200536830A
(en)
*
|
2004-02-06 |
2005-11-16 |
Chugai Pharmaceutical Co Ltd |
1-(2H)-isoquinolone derivative
|
|
CN1938296A
(zh)
|
2004-04-01 |
2007-03-28 |
安斯泰来制药有限公司 |
作为腺苷拮抗剂的吡嗪衍生物及其制药用途
|
|
GB0420722D0
(en)
|
2004-09-17 |
2004-10-20 |
Addex Pharmaceuticals Sa |
Novel allosteric modulators
|
|
KR100781704B1
(ko)
|
2005-04-20 |
2007-12-03 |
에스케이케미칼주식회사 |
피리딘 유도체와 이의 제조방법, 및 이를 포함하는약제조성물
|
|
US7452892B2
(en)
|
2005-06-17 |
2008-11-18 |
Bristol-Myers Squibb Company |
Triazolopyrimidine cannabinoid receptor 1 antagonists
|
|
KR101373535B1
(ko)
|
2005-07-26 |
2014-03-12 |
사노피 |
Rho-키나제 억제제로서의 피페리디닐-치환된 이소퀴놀론유도체
|
|
JP5049970B2
(ja)
|
2005-07-26 |
2012-10-17 |
サノフイ |
Rho−キナーゼ阻害剤としてのシクロヘキシルアミンイソキノロン誘導体
|
|
US20070099911A1
(en)
|
2005-10-28 |
2007-05-03 |
Wyeth |
Pyrroloquinolinone derivatives as 5-hydroxytryptamine-6 ligands
|
|
CA2646023A1
(en)
*
|
2006-03-10 |
2007-09-20 |
Neurogen Corporation |
Piperazinyl oxoalkyl tetrahydroisoquinolines and related analogues
|
|
GB0612428D0
(en)
|
2006-06-22 |
2006-08-02 |
Prolysis Ltd |
Antibacterial agents
|
|
RU2455302C2
(ru)
|
2006-12-27 |
2012-07-10 |
Санофи-Авентис |
ЗАМЕЩЕННЫЕ ИЗОХИНОЛИНОВЫЕ И ИЗОХИНОЛИНОНОВЫЕ ПРОИЗВОДНЫЕ В КАЧЕСТВЕ ИНГИБИТОРОВ Rho-КИНАЗЫ
|
|
RU2468011C2
(ru)
|
2006-12-27 |
2012-11-27 |
Санофи-Авентис |
Замещенные циклоалкиламином производные изохинолина и изохинолинона
|
|
NZ577980A
(en)
|
2006-12-27 |
2012-01-12 |
Sanofi Aventis |
Cycloalkylamine substituted isoquinolone derivatives
|
|
WO2009029214A1
(en)
*
|
2007-08-23 |
2009-03-05 |
Amgen Inc. |
Isoquinolone derivatives as phosphodiesterase 10 inhibitors
|
|
MX2010008375A
(es)
|
2008-01-30 |
2011-03-04 |
Cephalon Inc Star |
Derivados de piperidina espirocíclicos substituidos como ligandos de receptores de histamina-3 (h3).
|
|
JP5433691B2
(ja)
|
2008-06-25 |
2014-03-05 |
ブリストル−マイヤーズ スクイブ カンパニー |
Hiv結合阻害剤としてのジケトピペリジン誘導体
|
|
WO2010039186A2
(en)
*
|
2008-09-23 |
2010-04-08 |
Renovis, Inc. |
Compounds useful as faah modulators and uses thereof
|
|
EP2196465A1
(en)
|
2008-12-15 |
2010-06-16 |
Almirall, S.A. |
(3-oxo)pyridazin-4-ylurea derivatives as PDE4 inhibitors
|
|
EP2379564A1
(en)
*
|
2008-12-19 |
2011-10-26 |
Schering Corporation |
Bicyclic heterocyclic derivatives and methods of use thereof
|
|
HRP20160967T1
(hr)
|
2009-10-06 |
2016-10-07 |
Millennium Pharmaceuticals, Inc. |
Heterociklički spojevi korisni kao pdk1 inhibitori
|
|
CN102753545A
(zh)
|
2009-12-15 |
2012-10-24 |
盐野义制药株式会社 |
具有血管内皮脂酶抑制活性的噁二唑衍生物
|
|
JP5826261B2
(ja)
|
2010-06-28 |
2015-12-02 |
メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung |
癌に対する使用のためのキナーゼ阻害剤としての2,4−ジアリール置換[1,8]ナフチリジン
|
|
WO2012086735A1
(ja)
*
|
2010-12-22 |
2012-06-28 |
大正製薬株式会社 |
縮合複素環化合物
|
|
AU2012258977A1
(en)
|
2011-05-23 |
2014-01-16 |
Imago Pharmaceuticals, Inc. |
Inhibitors of LRRK2 kinase activity
|
|
RU2477723C2
(ru)
*
|
2011-06-16 |
2013-03-20 |
Общество С Ограниченной Ответственностью "Фьюжн Фарма" |
Ингибиторы протеинкиназ (варианты), их применение для лечения онкологических заболеваний и фармацевтическая композиция на их основе
|
|
CN102827073A
(zh)
|
2011-06-17 |
2012-12-19 |
安吉奥斯医药品有限公司 |
治疗活性组合物和它们的使用方法
|
|
JP6014155B2
(ja)
|
2011-10-31 |
2016-10-25 |
ゼノン・ファーマシューティカルズ・インコーポレイテッドXenon Pharmaceuticals Inc. |
ビアリールエーテルスルホンアミドおよび治療剤としてのそれらの使用
|
|
CN103183675A
(zh)
|
2011-12-27 |
2013-07-03 |
山东轩竹医药科技有限公司 |
磷酸二酯酶-4抑制剂
|
|
WO2013130855A1
(en)
*
|
2012-03-02 |
2013-09-06 |
Takeda Pharmaceutical Company Limited |
Indazole derivatives
|
|
US9550737B2
(en)
|
2012-06-11 |
2017-01-24 |
Ucb Biopharma Sprl |
TNF -α modulating benzimidazoles
|
|
JP2014024838A
(ja)
*
|
2012-06-21 |
2014-02-06 |
Taisho Pharmaceutical Co Ltd |
縮合複素環化合物を有効成分として含有する血糖低下作用薬
|
|
WO2014015088A1
(en)
*
|
2012-07-19 |
2014-01-23 |
Bristol-Myers Squibb Company |
Amide, urea or sulfone amide linked benzothiazole inhibitors of endothelial lipase
|
|
US9765039B2
(en)
*
|
2012-11-21 |
2017-09-19 |
Zenith Epigenetics Ltd. |
Biaryl derivatives as bromodomain inhibitors
|
|
RU2655604C2
(ru)
|
2013-01-11 |
2018-05-29 |
Фуджифилм Корпорэйшн |
Азотсодержащее гетероциклическое соединение или его соль
|
|
EP2970312B1
(en)
*
|
2013-03-11 |
2017-11-15 |
The Regents of The University of Michigan |
Bet bromodomain inhibitors and therapeutic methods using the same
|
|
SG11201506687RA
(en)
*
|
2013-03-15 |
2015-09-29 |
Plexxikon Inc |
Heterocyclic compounds and uses thereof
|
|
MX2015016344A
(es)
*
|
2013-05-27 |
2016-03-01 |
Novartis Ag |
Derivados de imidazo-pirrolidinona y su uso en el tratamiento de enfermedades.
|
|
EP3010918B1
(en)
*
|
2013-06-21 |
2018-08-15 |
Zenith Epigenetics Ltd. |
Novel substituted bicyclic compounds as bromodomain inhibitors
|
|
WO2014205594A1
(en)
*
|
2013-06-24 |
2014-12-31 |
Merck Sharp & Dohme Corp. |
Substituted benzofuran compounds and methods of use thereof for treatment of viral diseases
|
|
JP6509838B2
(ja)
*
|
2013-06-26 |
2019-05-08 |
アッヴィ・インコーポレイテッド |
Btk阻害薬としての一級カルボキサミド類
|
|
EP3290407B1
(en)
*
|
2013-10-18 |
2020-01-01 |
Celgene Quanticel Research, Inc |
Bromodomain inhibitors
|
|
WO2015081189A1
(en)
*
|
2013-11-26 |
2015-06-04 |
Incyte Corporation |
Bicyclic heterocycles as bet protein inhibitors
|
|
US9920052B2
(en)
*
|
2013-12-09 |
2018-03-20 |
Ucb Biopharma Sprl |
Imidazopyridine derivatives as modulators of TNF activity
|
|
US10173991B2
(en)
*
|
2014-01-07 |
2019-01-08 |
Bristol-Myers Squibb Company |
Sulfone amide linked benzothiazole inhibitors of endothelial lipase
|
|
US9499551B2
(en)
|
2014-01-24 |
2016-11-22 |
Confluence Life Sciences, Inc. |
Substituted pyrrolo[2,3-b]pyridines for treating cancer or inflammatory diseases
|
|
EA034972B1
(ru)
*
|
2014-04-23 |
2020-04-13 |
Инсайт Корпорейшн |
1h-пирроло[2,3-c]пиридин-7(6h)-оны в качестве ингибиторов белков bet
|
|
MA40940A
(fr)
|
2014-11-10 |
2017-09-19 |
Constellation Pharmaceuticals Inc |
Pyrrolopyridines substituées utilisées en tant qu'inhibiteurs de bromodomaines
|
|
MA40943A
(fr)
*
|
2014-11-10 |
2017-09-19 |
Constellation Pharmaceuticals Inc |
Pyrrolopyridines substituées utilisées en tant qu'inhibiteurs de bromodomaines
|
|
US9763922B2
(en)
*
|
2014-11-27 |
2017-09-19 |
Genentech, Inc. |
Therapeutic compounds and uses thereof
|
|
EP3265453B1
(en)
*
|
2015-03-05 |
2022-06-29 |
Boehringer Ingelheim International GmbH |
New pyridinones and isoquinolinones as inhibitors of the bromodomain brd9
|
|
AR104259A1
(es)
*
|
2015-04-15 |
2017-07-05 |
Celgene Quanticel Res Inc |
Inhibidores de bromodominio
|
|
TW201642860A
(zh)
*
|
2015-04-22 |
2016-12-16 |
塞爾基因定量細胞研究公司 |
布羅莫結構域抑制劑
|