JP2004524315A5 - - Google Patents

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Publication number
JP2004524315A5
JP2004524315A5 JP2002567926A JP2002567926A JP2004524315A5 JP 2004524315 A5 JP2004524315 A5 JP 2004524315A5 JP 2002567926 A JP2002567926 A JP 2002567926A JP 2002567926 A JP2002567926 A JP 2002567926A JP 2004524315 A5 JP2004524315 A5 JP 2004524315A5
Authority
JP
Japan
Prior art keywords
alkyl
group
halogenoalkyl
optionally
aryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2002567926A
Other languages
English (en)
Japanese (ja)
Other versions
JP2004524315A (ja
Filing date
Publication date
Priority claimed from DE10108480A external-priority patent/DE10108480A1/de
Application filed filed Critical
Publication of JP2004524315A publication Critical patent/JP2004524315A/ja
Publication of JP2004524315A5 publication Critical patent/JP2004524315A5/ja
Pending legal-status Critical Current

Links

JP2002567926A 2001-02-22 2002-02-11 ピラゾリルピリミジン Pending JP2004524315A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10108480A DE10108480A1 (de) 2001-02-22 2001-02-22 Pyrazolylpyrimidine
PCT/EP2002/001400 WO2002068413A1 (de) 2001-02-22 2002-02-11 Pyrazolylpyrimidine

Publications (2)

Publication Number Publication Date
JP2004524315A JP2004524315A (ja) 2004-08-12
JP2004524315A5 true JP2004524315A5 (https=) 2005-12-22

Family

ID=7675081

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002567926A Pending JP2004524315A (ja) 2001-02-22 2002-02-11 ピラゾリルピリミジン

Country Status (13)

Country Link
US (1) US7087616B2 (https=)
EP (1) EP1363905A1 (https=)
JP (1) JP2004524315A (https=)
KR (1) KR100854583B1 (https=)
CN (1) CN1301992C (https=)
BR (1) BR0207509A (https=)
DE (1) DE10108480A1 (https=)
HU (1) HUP0303241A2 (https=)
IL (1) IL157298A0 (https=)
MX (1) MXPA03007433A (https=)
TW (1) TWI236475B (https=)
WO (1) WO2002068413A1 (https=)
ZA (1) ZA200306468B (https=)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI372050B (en) * 2003-07-03 2012-09-11 Astex Therapeutics Ltd (morpholin-4-ylmethyl-1h-benzimidazol-2-yl)-1h-pyrazoles
MX2007008008A (es) * 2004-12-30 2007-11-12 Astex Therapeutics Ltd Compuestos de pirazol que modulan la actividad de las cinasas cdk, gsk y aurora.
DE102005058418A1 (de) * 2005-12-07 2007-06-21 Bayer Cropscience Gmbh Verfahren zur Herstellung von Haloalkyl(thio)vinimidiniumsalzen und 4-(Haloalkyl(thio))-pyrazolen und deren Umsetzung zu Pflanzenschutzmitteln
US8399442B2 (en) * 2005-12-30 2013-03-19 Astex Therapeutics Limited Pharmaceutical compounds
JP5523829B2 (ja) * 2006-06-29 2014-06-18 アステックス、セラピューティックス、リミテッド 複合薬剤
EP2043635A2 (en) * 2006-06-29 2009-04-08 Astex Therapeutics Limited Pharmaceutical combinations
DE102007003036A1 (de) * 2006-12-20 2008-06-26 Bayer Cropscience Ag Pyrimidinylpyrazole
DE102007044032A1 (de) 2007-09-14 2009-03-19 Bayer Healthcare Ag Substituierte heterocyclische Verbindungen und ihre Verwendung
DE102007048447A1 (de) 2007-10-10 2009-04-16 Bayer Healthcare Ag Substituierte Dihydropyrazolthione und ihre Verwendung
EP2135865A1 (de) * 2008-06-17 2009-12-23 Bayer CropScience AG Substituierte 1-(Diazinyl) pyrazol-4-yl-essigsäuren, Verfahren zu deren Herstellung und deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren
AU2009281457A1 (en) * 2008-08-14 2010-02-18 Bayer Cropscience Ag Insecticidal 4-phenyl-1H-pyrazoles
CN102414197B (zh) 2009-04-27 2015-11-25 美国陶氏益农公司 杀虫剂吡啶化合物
BR112012006956A2 (pt) * 2009-10-12 2015-09-15 Bayer Cropscience Ag 1- (pirida-3-il) -pirazóisol e 1- (pirimida-5-il) - pirazóisol como pesticidas
EP2499130A1 (de) 2009-11-11 2012-09-19 Bayer CropScience AG Neue diazinyl-pyrazolylverbindungen
JP2012116796A (ja) * 2010-12-01 2012-06-21 Sumitomo Chemical Co Ltd ヘテロ芳香環化合物およびその有害生物防除用途
WO2013138617A1 (en) 2012-03-16 2013-09-19 Axikin Pharmaceuticals, Inc. 3,5-diaminopyrazole kinase inhibitors
NZ631142A (en) 2013-09-18 2016-03-31 Axikin Pharmaceuticals Inc Pharmaceutically acceptable salts of 3,5-diaminopyrazole kinase inhibitors
CR20170077A (es) 2014-08-04 2017-06-26 Nuevolution As Derivados de heterociclilo opcionalmente condensados de pirimidina útiles para el tratamiento de enfermedades inflamatorias, metabólicas, oncológicas y autoinmunitarias
US10118890B2 (en) 2014-10-10 2018-11-06 The Research Foundation For The State University Of New York Trifluoromethoxylation of arenes via intramolecular trifluoromethoxy group migration
TWI703133B (zh) 2014-12-23 2020-09-01 美商艾克斯基製藥公司 3,5-二胺基吡唑激酶抑制劑
UY38994A (es) 2019-12-20 2021-07-30 Nuevolution As Compuestos activos frente a receptores nucleares
MX2022007265A (es) 2019-12-20 2022-09-09 Nuevolution As Compuestos activos frente a receptores nucleares.
WO2021198956A1 (en) 2020-03-31 2021-10-07 Nuevolution A/S Compounds active towards nuclear receptors
AU2021245397A1 (en) 2020-03-31 2022-10-20 Nuevolution A/S Compounds active towards nuclear receptors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3910910A (en) * 1972-03-31 1975-10-07 American Home Prod (2-Pyrimidinylthio) alkanoic acids, esters, amides and hydrazides
US4663327A (en) * 1984-05-23 1987-05-05 Bayer Aktiengesellschaft 1-heteroaryl-4-aryl-pyrazolin-5-ones
WO1994029268A1 (de) 1993-06-07 1994-12-22 Bayer Aktiengesellschaft Iodpropargylcarbamate und ihre verwendung als biozide im pflanzen- und materialschutz
CN1153779A (zh) * 1995-09-28 1997-07-09 山道士有限公司 2-(4-吡唑基氧基-嘧啶-5-基)乙酸衍生物
EP0967212A4 (en) * 1996-12-16 2002-01-09 Sumitomo Chemical Co PYRAZOLINE COMPOUNDS AND THEIR USE AS A MEANS FOR CONTROLLING PLANT DISEASES

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