BR0207509A - Pirazolilpirimidinas - Google Patents
PirazolilpirimidinasInfo
- Publication number
- BR0207509A BR0207509A BR0207509-1A BR0207509A BR0207509A BR 0207509 A BR0207509 A BR 0207509A BR 0207509 A BR0207509 A BR 0207509A BR 0207509 A BR0207509 A BR 0207509A
- Authority
- BR
- Brazil
- Prior art keywords
- pyrazolylpyrimidines
- pirazolylpyrimidines
- substances
- novel
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/34—One oxygen atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/42—One nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
Abstract
"PIRAZOLILPIRIMIDINAS". Novas pirazolilpirimidinas da fórmula (I), na qual R1, R2, X, n, Y, Z e R têm os significados indicados na descrição, vários processos para a preparação dessas substâncias e sua aplicação para combater pragas.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10108480A DE10108480A1 (de) | 2001-02-22 | 2001-02-22 | Pyrazolylpyrimidine |
PCT/EP2002/001400 WO2002068413A1 (de) | 2001-02-22 | 2002-02-11 | Pyrazolylpyrimidine |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0207509A true BR0207509A (pt) | 2004-03-09 |
Family
ID=7675081
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0207509-1A BR0207509A (pt) | 2001-02-22 | 2002-02-11 | Pirazolilpirimidinas |
Country Status (13)
Country | Link |
---|---|
US (1) | US7087616B2 (pt) |
EP (1) | EP1363905A1 (pt) |
JP (1) | JP2004524315A (pt) |
KR (1) | KR100854583B1 (pt) |
CN (1) | CN1301992C (pt) |
BR (1) | BR0207509A (pt) |
DE (1) | DE10108480A1 (pt) |
HU (1) | HUP0303241A2 (pt) |
IL (1) | IL157298A0 (pt) |
MX (1) | MXPA03007433A (pt) |
TW (1) | TWI236475B (pt) |
WO (1) | WO2002068413A1 (pt) |
ZA (1) | ZA200306468B (pt) |
Families Citing this family (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI372050B (en) * | 2003-07-03 | 2012-09-11 | Astex Therapeutics Ltd | (morpholin-4-ylmethyl-1h-benzimidazol-2-yl)-1h-pyrazoles |
US8110573B2 (en) | 2004-12-30 | 2012-02-07 | Astex Therapeutics Limited | Pyrazole compounds that modulate the activity of CDK, GSK and aurora kinases |
DE102005058418A1 (de) * | 2005-12-07 | 2007-06-21 | Bayer Cropscience Gmbh | Verfahren zur Herstellung von Haloalkyl(thio)vinimidiniumsalzen und 4-(Haloalkyl(thio))-pyrazolen und deren Umsetzung zu Pflanzenschutzmitteln |
EP1968579A1 (en) * | 2005-12-30 | 2008-09-17 | Astex Therapeutics Limited | Pharmaceutical compounds |
WO2008001115A2 (en) * | 2006-06-29 | 2008-01-03 | Astex Therapeutics Limited | Pharmaceutical combinations of 1-cyclopropyl-3- [3- (5-m0rphoolin-4-ylmethyl-1h-benzoimidazol-2-yl) -lh-1-pyrazol- 4-yl] -urea |
US20110159111A1 (en) * | 2006-06-29 | 2011-06-30 | Astex Therapeutics Limited | Pharmaceutical combinations |
DE102007003036A1 (de) * | 2006-12-20 | 2008-06-26 | Bayer Cropscience Ag | Pyrimidinylpyrazole |
DE102007044032A1 (de) | 2007-09-14 | 2009-03-19 | Bayer Healthcare Ag | Substituierte heterocyclische Verbindungen und ihre Verwendung |
DE102007048447A1 (de) | 2007-10-10 | 2009-04-16 | Bayer Healthcare Ag | Substituierte Dihydropyrazolthione und ihre Verwendung |
EP2135865A1 (de) * | 2008-06-17 | 2009-12-23 | Bayer CropScience AG | Substituierte 1-(Diazinyl) pyrazol-4-yl-essigsäuren, Verfahren zu deren Herstellung und deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren |
BRPI0918430A2 (pt) * | 2008-08-14 | 2015-11-24 | Bayer Cropscience Ag | 4-fenil-1h-pirazóis inseticidas. |
US8604199B2 (en) * | 2009-04-27 | 2013-12-10 | Dow Agrosciences, Llc. | Insecticidal pyridine compounds |
CN102573478B (zh) * | 2009-10-12 | 2015-12-16 | 拜尔农作物科学股份公司 | 作为杀虫剂的1-(吡啶-3-基)-吡唑和1-(嘧啶-5-基)-吡唑 |
JP2013510815A (ja) | 2009-11-11 | 2013-03-28 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | 新規なジアジニルピラゾリル化合物 |
JP2012116796A (ja) * | 2010-12-01 | 2012-06-21 | Sumitomo Chemical Co Ltd | ヘテロ芳香環化合物およびその有害生物防除用途 |
US9365556B2 (en) | 2012-03-16 | 2016-06-14 | Axikin Pharmaceuticals, Inc. | 3,5-diaminopyrazole kinase inhibitors |
NZ631142A (en) | 2013-09-18 | 2016-03-31 | Axikin Pharmaceuticals Inc | Pharmaceutically acceptable salts of 3,5-diaminopyrazole kinase inhibitors |
PE20170684A1 (es) | 2014-08-04 | 2017-06-15 | Nuevolution As | Derivados de heterociclilo opcionalmente condensados de pirimidina utiles para el tratamiento de enfermedades inflamatorias, metabolicas, oncologicas y autoinmunitarias |
US10118890B2 (en) | 2014-10-10 | 2018-11-06 | The Research Foundation For The State University Of New York | Trifluoromethoxylation of arenes via intramolecular trifluoromethoxy group migration |
US9546163B2 (en) | 2014-12-23 | 2017-01-17 | Axikin Pharmaceuticals, Inc. | 3,5-diaminopyrazole kinase inhibitors |
US11447479B2 (en) | 2019-12-20 | 2022-09-20 | Nuevolution A/S | Compounds active towards nuclear receptors |
JP2023519603A (ja) | 2020-03-31 | 2023-05-11 | ヌエヴォリューション・アクティーゼルスカブ | 核内受容体に対して活性な化合物 |
AU2021249530A1 (en) | 2020-03-31 | 2022-12-01 | Nuevolution A/S | Compounds active towards nuclear receptors |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3910910A (en) * | 1972-03-31 | 1975-10-07 | American Home Prod | (2-Pyrimidinylthio) alkanoic acids, esters, amides and hydrazides |
US4663327A (en) * | 1984-05-23 | 1987-05-05 | Bayer Aktiengesellschaft | 1-heteroaryl-4-aryl-pyrazolin-5-ones |
WO1994029268A1 (de) | 1993-06-07 | 1994-12-22 | Bayer Aktiengesellschaft | Iodpropargylcarbamate und ihre verwendung als biozide im pflanzen- und materialschutz |
CN1153779A (zh) * | 1995-09-28 | 1997-07-09 | 山道士有限公司 | 2-(4-吡唑基氧基-嘧啶-5-基)乙酸衍生物 |
EP0967212A4 (en) * | 1996-12-16 | 2002-01-09 | Sumitomo Chemical Co | PYRAZOLINE COMPOUNDS AND THEIR USE AS PLANT DISEASE CONTROL AGENTS |
-
2001
- 2001-02-22 DE DE10108480A patent/DE10108480A1/de not_active Withdrawn
-
2002
- 2002-02-11 KR KR1020037010576A patent/KR100854583B1/ko not_active IP Right Cessation
- 2002-02-11 BR BR0207509-1A patent/BR0207509A/pt not_active IP Right Cessation
- 2002-02-11 JP JP2002567926A patent/JP2004524315A/ja active Pending
- 2002-02-11 IL IL15729802A patent/IL157298A0/xx unknown
- 2002-02-11 HU HU0303241A patent/HUP0303241A2/hu unknown
- 2002-02-11 US US10/468,371 patent/US7087616B2/en not_active Expired - Fee Related
- 2002-02-11 EP EP02711857A patent/EP1363905A1/de not_active Withdrawn
- 2002-02-11 WO PCT/EP2002/001400 patent/WO2002068413A1/de active Application Filing
- 2002-02-11 MX MXPA03007433A patent/MXPA03007433A/es active IP Right Grant
- 2002-02-11 CN CNB028054326A patent/CN1301992C/zh not_active Expired - Fee Related
- 2002-02-21 TW TW091102971A patent/TWI236475B/zh not_active IP Right Cessation
-
2003
- 2003-08-20 ZA ZA200306468A patent/ZA200306468B/en unknown
Also Published As
Publication number | Publication date |
---|---|
ZA200306468B (en) | 2005-02-04 |
MXPA03007433A (es) | 2003-11-18 |
CN1301992C (zh) | 2007-02-28 |
HUP0303241A2 (hu) | 2004-01-28 |
TWI236475B (en) | 2005-07-21 |
IL157298A0 (en) | 2004-02-19 |
JP2004524315A (ja) | 2004-08-12 |
KR20030075188A (ko) | 2003-09-22 |
KR100854583B1 (ko) | 2008-08-27 |
CN1492864A (zh) | 2004-04-28 |
WO2002068413A1 (de) | 2002-09-06 |
US20040102465A1 (en) | 2004-05-27 |
DE10108480A1 (de) | 2002-09-05 |
US7087616B2 (en) | 2006-08-08 |
EP1363905A1 (de) | 2003-11-26 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BR0207509A (pt) | Pirazolilpirimidinas | |
BR0309873A (pt) | Pirazolo-pirimidin-4-onas substituìdas | |
BR9714377A (pt) | Derivados de 3-tiocarbamoilpirazol como pesticidas | |
BR9611175B1 (pt) | compostos e composiÇÕes farmacÊuticas. | |
BR9714470A (pt) | Fenilcetoenóis substituìdos e sua utilização como agente para o combate de pragas | |
BR0314087A (pt) | Cetoenóis spirocìclicos substituìdos | |
DK0804421T3 (da) | 2-((Dihydro)pyrazolyl-3'-oxymethylen)-anilider som skadedyrsbekæmpelsesmidler og fungicider | |
SE9802729D0 (sv) | Novel Compounds | |
BR9808184A (pt) | 2-arilciclopentano-1, 3-dionas | |
SV2002000776A (es) | Nuevas imidazotriazinonas sustituidas ref.lea 34 985-sv | |
BR0212075A (pt) | Combinações de substâncias ativas fungicidas | |
ES2107284T3 (es) | Nuevas n-piridil-carboxamidas, su procedimiento de preparacion y composiciones farmaceuticas que las contienen. | |
BR0115968A (pt) | Delta1-pirrolinas | |
BR9911978A (pt) | Feniluracilas substituìdas | |
BRPI0410236A (pt) | oxiarenos substituìdos | |
BR0110180A (pt) | 4-hidróxi-tetrahidropiridonas fenil-substituìdas | |
BR0309568A (pt) | Triazolopirimidinas | |
BR0112927A (pt) | Pirazolilbifenilcarboxamidas e sua aplicação para combater microorganismos indesejados | |
BR0109054A (pt) | Benzoilciclohexenonas substituìdas | |
BR0110632A (pt) | 2-enamino-cetonitrilas substituìdas | |
BR0111625A (pt) | Heterociclos substituìdos por hetarila | |
BR0209082A (pt) | 1,3-dionas carbocìclicas substituìdas com tiazolila como pesticidas | |
BR0313751A (pt) | Heterociclilpirimidinas substituìdas | |
ATE222896T1 (de) | Substituierte thiazoline und ihre verwendung zur bekämpfung von tierischen schädlingen | |
BR0012980A (pt) | Tieni (amino) sulfoniluréias substituìdas |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 8A E 9A ANUIDADE(S). |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2103 DE 26/04/2011. |