JP2004502663A - (r)−2−アルキル−3−フェニルプロピオン酸の調製 - Google Patents
(r)−2−アルキル−3−フェニルプロピオン酸の調製 Download PDFInfo
- Publication number
- JP2004502663A JP2004502663A JP2002507758A JP2002507758A JP2004502663A JP 2004502663 A JP2004502663 A JP 2004502663A JP 2002507758 A JP2002507758 A JP 2002507758A JP 2002507758 A JP2002507758 A JP 2002507758A JP 2004502663 A JP2004502663 A JP 2004502663A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- alkyl
- compound
- alkoxy
- methoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 0 COC1=C(*)C[C@](C=C(*)C(O)=O)C=C1 Chemical compound COC1=C(*)C[C@](C=C(*)C(O)=O)C=C1 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/40—Unsaturated compounds
- C07C59/58—Unsaturated compounds containing ether groups, groups, groups, or groups
- C07C59/64—Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings
- C07C59/66—Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings the non-carboxylic part of the ether containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/347—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups
- C07C51/36—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups by hydrogenation of carbon-to-carbon unsaturated bonds
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Catalysts (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH13172000 | 2000-07-03 | ||
| PCT/CH2001/000397 WO2002002500A1 (en) | 2000-07-03 | 2001-06-26 | Preparation of (r)-2-alkyl-3-phenylpropionic acids |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2004502663A true JP2004502663A (ja) | 2004-01-29 |
| JP2004502663A5 JP2004502663A5 (enExample) | 2005-02-03 |
Family
ID=4565374
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002507758A Pending JP2004502663A (ja) | 2000-07-03 | 2001-06-26 | (r)−2−アルキル−3−フェニルプロピオン酸の調製 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US6683206B2 (enExample) |
| EP (1) | EP1296927B1 (enExample) |
| JP (1) | JP2004502663A (enExample) |
| CN (1) | CN100482632C (enExample) |
| AR (1) | AR028783A1 (enExample) |
| AT (1) | ATE546425T1 (enExample) |
| AU (1) | AU2001273761A1 (enExample) |
| BR (1) | BR0112146A (enExample) |
| CA (1) | CA2414839C (enExample) |
| TW (1) | TWI271398B (enExample) |
| WO (1) | WO2002002500A1 (enExample) |
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2004502656A (ja) * | 2000-07-03 | 2004-01-29 | シュペーデル・ファルマ・アーゲー | (r)−2−アルキル−3−フェニル−1−プロパノールの調製方法 |
| JP2004502700A (ja) * | 2000-07-03 | 2004-01-29 | ソルヴィーアス アクチェンゲゼルシャフト | フェロセニルジホスフィンおよびその使用 |
| JP2008525506A (ja) * | 2004-12-27 | 2008-07-17 | ディーエスエム ファイン ケミカルズ オーストリア エヌエフジー ゲーエムベーハー ウント ツェーオー カーゲー | アクリル酸誘導体の遷移金属触媒不斉水素化方法および不斉遷移金属触媒反応用の新規な触媒系 |
| JP2008534448A (ja) * | 2005-03-17 | 2008-08-28 | ビーエーエスエフ ソシエタス・ヨーロピア | 光学活性3−フェニルプロピオン酸誘導体を生成する方法、およびその誘導体の後続生成物 |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH694251A5 (de) * | 1999-07-14 | 2004-10-15 | Eprova Ag | Herstellung von Tetrahydropterin und Derivaten. |
| GB0500700D0 (en) * | 2005-01-14 | 2005-02-23 | Stylacats Ltd | Process for the manufacture of 2-alkyl-3-phenylpropionic acids and alcohols |
| DE102005012408A1 (de) * | 2005-03-17 | 2006-09-21 | Basf Ag | Verfahren zur Herstellung von optisch aktiven 3-Phenylpropionsäurederivaten und Folgeprodukten davon |
| DE102005052195A1 (de) | 2005-10-28 | 2007-05-03 | Reuter Chemischer Apparatebau Kg | Verfahren zur Herstellung von chiralen Octensäurederivaten |
| US7935841B2 (en) | 2006-04-21 | 2011-05-03 | Dr. Reddy's Laboratories Limited | Bisphospholanes for use as catalysts in asymmetric reactions |
| EP1939182A1 (de) * | 2006-12-22 | 2008-07-02 | Speedel Experimenta AG | Verfahren zur Herstellung von (R oder S)-2-Alkyl-3-heterocyclyl-1-propanolen |
| EP1958666A1 (en) | 2007-02-13 | 2008-08-20 | Speedel Experimenta AG | Heterocyclic-substituted alkanamides as therapeutic compounds |
| EP2178816A1 (en) * | 2007-07-11 | 2010-04-28 | DSM Fine Chemicals Austria Nfg GmbH & Co KG | Alpha-substituted , -unsaturated e- or z-aldehydes, use thereof, and processes for their preparation , |
| EP2173696A1 (en) | 2007-07-11 | 2010-04-14 | DSM IP Assets B.V. | Preparation of a saturated aldehyde |
| DE102007049039A1 (de) | 2007-10-11 | 2009-04-16 | Reuter Chemischer Apparatebau Kg | Verfahren zur Herstellung von 8-Hydrazino-8-Aryl-Octanoylderivaten und deren Verwendung |
| US8203005B2 (en) | 2009-10-29 | 2012-06-19 | Carbo Design Llc | Manufacturing process for enantiomerically pure 8-aryloctanoic acids as Aliskiren |
| TW201202178A (en) | 2010-06-04 | 2012-01-16 | Chemo Iberica Sa | Process for producing Aliskiren |
| US8703976B2 (en) | 2011-10-02 | 2014-04-22 | Milan Soukup | Manufacturing process for 8-aryloctanoic acids such as Aliskiren |
| US9056816B2 (en) | 2011-10-25 | 2015-06-16 | Jubilant Life Sciences Limited | Process for the preparation of aliskiren |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4307232A (en) * | 1980-03-21 | 1981-12-22 | E. I. Du Pont De Nemours And Company | Preparation of dialkyl- and diarylphosphonoalkanoic acids and substituted acrylic acids |
| JPH0827079A (ja) * | 1994-04-18 | 1996-01-30 | Ciba Geigy Ag | アルファ−アミノアルカン酸及還元生成物 |
| JPH09309826A (ja) * | 1996-05-22 | 1997-12-02 | Kissei Pharmaceut Co Ltd | 糸球体疾患の予防および治療剤 |
| JP2003519135A (ja) * | 1999-12-23 | 2003-06-17 | アイコス コーポレイション | 環状amp特異性ホスホジエステラーゼ阻害剤としてのピロリジン誘導体 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2671079B1 (fr) * | 1990-12-28 | 1994-06-03 | Elf Aquitaine | Procede d'hydrogenation de composes organiques et catalyseurs au ruthenium pour sa realisation. |
-
2001
- 2001-06-26 CN CNB018122310A patent/CN100482632C/zh not_active Expired - Fee Related
- 2001-06-26 BR BR0112146-4A patent/BR0112146A/pt not_active Application Discontinuation
- 2001-06-26 AT AT01940045T patent/ATE546425T1/de active
- 2001-06-26 CA CA2414839A patent/CA2414839C/en not_active Expired - Fee Related
- 2001-06-26 WO PCT/CH2001/000397 patent/WO2002002500A1/en not_active Ceased
- 2001-06-26 US US10/312,855 patent/US6683206B2/en not_active Expired - Fee Related
- 2001-06-26 AU AU2001273761A patent/AU2001273761A1/en not_active Abandoned
- 2001-06-26 EP EP01940045A patent/EP1296927B1/en not_active Expired - Lifetime
- 2001-06-26 JP JP2002507758A patent/JP2004502663A/ja active Pending
- 2001-06-27 TW TW090115551A patent/TWI271398B/zh not_active IP Right Cessation
- 2001-07-03 AR ARP010103175A patent/AR028783A1/es active IP Right Grant
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4307232A (en) * | 1980-03-21 | 1981-12-22 | E. I. Du Pont De Nemours And Company | Preparation of dialkyl- and diarylphosphonoalkanoic acids and substituted acrylic acids |
| JPH0827079A (ja) * | 1994-04-18 | 1996-01-30 | Ciba Geigy Ag | アルファ−アミノアルカン酸及還元生成物 |
| JPH09309826A (ja) * | 1996-05-22 | 1997-12-02 | Kissei Pharmaceut Co Ltd | 糸球体疾患の予防および治療剤 |
| JP2003519135A (ja) * | 1999-12-23 | 2003-06-17 | アイコス コーポレイション | 環状amp特異性ホスホジエステラーゼ阻害剤としてのピロリジン誘導体 |
Cited By (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2004502656A (ja) * | 2000-07-03 | 2004-01-29 | シュペーデル・ファルマ・アーゲー | (r)−2−アルキル−3−フェニル−1−プロパノールの調製方法 |
| JP2004502700A (ja) * | 2000-07-03 | 2004-01-29 | ソルヴィーアス アクチェンゲゼルシャフト | フェロセニルジホスフィンおよびその使用 |
| JP2008525506A (ja) * | 2004-12-27 | 2008-07-17 | ディーエスエム ファイン ケミカルズ オーストリア エヌエフジー ゲーエムベーハー ウント ツェーオー カーゲー | アクリル酸誘導体の遷移金属触媒不斉水素化方法および不斉遷移金属触媒反応用の新規な触媒系 |
| JP2008534448A (ja) * | 2005-03-17 | 2008-08-28 | ビーエーエスエフ ソシエタス・ヨーロピア | 光学活性3−フェニルプロピオン酸誘導体を生成する方法、およびその誘導体の後続生成物 |
| JP4763771B2 (ja) * | 2005-03-17 | 2011-08-31 | ビーエーエスエフ ソシエタス・ヨーロピア | 光学活性3−フェニルプロピオン酸誘導体を生成する方法、およびその誘導体の後続生成物 |
Also Published As
| Publication number | Publication date |
|---|---|
| US6683206B2 (en) | 2004-01-27 |
| AU2001273761A1 (en) | 2002-01-14 |
| BR0112146A (pt) | 2003-05-06 |
| AR028783A1 (es) | 2003-05-21 |
| CN100482632C (zh) | 2009-04-29 |
| EP1296927A1 (en) | 2003-04-02 |
| CA2414839A1 (en) | 2002-01-10 |
| CA2414839C (en) | 2010-02-16 |
| US20030139625A1 (en) | 2003-07-24 |
| ATE546425T1 (de) | 2012-03-15 |
| TWI271398B (en) | 2007-01-21 |
| EP1296927B1 (en) | 2012-02-22 |
| CN1440379A (zh) | 2003-09-03 |
| WO2002002500A1 (en) | 2002-01-10 |
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