JP2003531184A5 - - Google Patents

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Publication number
JP2003531184A5
JP2003531184A5 JP2001578384A JP2001578384A JP2003531184A5 JP 2003531184 A5 JP2003531184 A5 JP 2003531184A5 JP 2001578384 A JP2001578384 A JP 2001578384A JP 2001578384 A JP2001578384 A JP 2001578384A JP 2003531184 A5 JP2003531184 A5 JP 2003531184A5
Authority
JP
Japan
Prior art keywords
aryloxy
propan
mixture
trialkylsiloxypropane
regioisomers
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2001578384A
Other languages
English (en)
Japanese (ja)
Other versions
JP2003531184A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2001/012792 external-priority patent/WO2001081286A1/en
Publication of JP2003531184A publication Critical patent/JP2003531184A/ja
Publication of JP2003531184A5 publication Critical patent/JP2003531184A5/ja
Pending legal-status Critical Current

Links

JP2001578384A 2000-04-21 2001-04-20 (r)−1−(アリールオキシ)プロパン−2−オールの製造方法 Pending JP2003531184A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US19894200P 2000-04-21 2000-04-21
US60/198,942 2000-04-21
PCT/US2001/012792 WO2001081286A1 (en) 2000-04-21 2001-04-20 Process for preparation of r-1-(aryloxy)propan-2-ol

Publications (2)

Publication Number Publication Date
JP2003531184A JP2003531184A (ja) 2003-10-21
JP2003531184A5 true JP2003531184A5 (https=) 2008-06-19

Family

ID=22735535

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001578384A Pending JP2003531184A (ja) 2000-04-21 2001-04-20 (r)−1−(アリールオキシ)プロパン−2−オールの製造方法

Country Status (7)

Country Link
US (1) US6448449B2 (https=)
EP (1) EP1280753A1 (https=)
JP (1) JP2003531184A (https=)
KR (1) KR20020097223A (https=)
CN (1) CN1438981A (https=)
CA (1) CA2406215A1 (https=)
WO (1) WO2001081286A1 (https=)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU230030B1 (hu) 1999-10-08 2015-05-28 Debiopharm International Sa Fab I inhibitorok
US20020013906A1 (en) * 2000-06-14 2002-01-31 Walter Wallach Secure medical test and result delivery system
EP1560584B1 (en) * 2001-04-06 2009-01-14 Affinium Pharmaceuticals, Inc. Fab i inhibitors
EP1575951B1 (en) * 2002-12-06 2014-06-25 Debiopharm International SA Heterocyclic compounds, methods of making them and their use in therapy
WO2004082586A2 (en) 2003-03-17 2004-09-30 Affinium Pharmaceuticals, Inc. Phamaceutical compositions comprising inhibitors of fab i and further antibiotics
DK1828167T3 (da) * 2004-06-04 2014-10-20 Debiopharm Int Sa Acrylamidderivater som antibiotiske midler
KR20080075027A (ko) * 2005-12-05 2008-08-13 아피늄 파마슈티컬스, 인크. Fabi 억제제 및 항박테리아제로서의헤테로시클릴아크릴아미드 화합물
JP5468899B2 (ja) 2006-07-20 2014-04-09 アフィニウム ファーマシューティカルズ, インク. Fabiインヒビターとしてのアクリルアミド誘導体
EP2125802A4 (en) 2007-02-16 2014-08-20 Debiopharm Int Sa SALTS, PRODRUGS AND POLYMORPHES OF FAB I INHIBITORS
KR101503745B1 (ko) * 2010-02-25 2015-03-19 에스케이이노베이션 주식회사 나이트레이트 음이온의 이산화탄소/에폭사이드 공중합 촉매 시스템
AU2013279021C1 (en) 2012-06-19 2017-03-16 Debiopharm International Sa Prodrug derivatives of (E)-N-methyl-N-((3-methylbenzofuran-2-yl)methyl)-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)acrylamide
RS61312B1 (sr) 2016-02-26 2021-02-26 Debiopharm Int Sa Lek za lečenje infekcija dijabetskog stopala
TN2021000159A1 (en) 2019-02-14 2023-04-04 Debiopharm Int Sa Afabicin formulation, method for making the same and uses thereof
CN112079958A (zh) * 2019-06-12 2020-12-15 中国石化扬子石油化工有限公司 一种碳五共聚石油树脂的制备方法
SG11202113174SA (en) 2019-06-14 2021-12-30 Debiopharm Int Sa Medicament and use thereof for treating bacterial infections involving biofilm

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8525954D0 (en) * 1985-10-21 1985-11-27 Mcneilab Inc Chlorination of carbohydrates &c alcohols
GB8525953D0 (en) * 1985-10-21 1985-11-27 Mcneilab Inc Preparation of galactopyranoside
JP2620290B2 (ja) * 1988-03-11 1997-06-11 旭電化工業株式会社 シリルオキシ基を有するアリールエーテル化合物の製造法
AU4376589A (en) * 1988-11-07 1990-05-10 Gist-Brocades N.V. Optically active benzoxazines and benzothiazines
US5637739A (en) 1990-03-21 1997-06-10 Research Corporation Technologies, Inc. Chiral catalysts and catalytic epoxidation catalyzed thereby
US5559222A (en) * 1995-02-03 1996-09-24 Eli Lilly And Company Preparation of 1-(2'-deoxy-2',2'-difluoro-D-ribo-pentofuranosyl)-cytosine from 2-deoxy-2,2-difluoro-β-D-ribo-pentopyranose
US5665890A (en) 1995-03-14 1997-09-09 President And Fellows Of Harvard College Stereoselective ring opening reactions
DE69818057D1 (de) * 1997-07-10 2003-10-16 Du Pont Herstellung von optisch aktiven halohydrintrialkylsilylethern
JPH11269131A (ja) 1998-03-20 1999-10-05 Asahi Glass Co Ltd 1−アシルオキシ−2−プロパノールの製造方法
JPH11279100A (ja) 1998-03-25 1999-10-12 Asahi Glass Co Ltd 光学活性な1−置換−2−プロパノールの製造方法
JP2000063314A (ja) 1998-08-14 2000-02-29 Asahi Glass Co Ltd 光学活性な1−置換−2−プロパノールの製造方法

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