JP2002543109A - 経口投与の発泡性薬剤配給系 - Google Patents
経口投与の発泡性薬剤配給系Info
- Publication number
- JP2002543109A JP2002543109A JP2000614975A JP2000614975A JP2002543109A JP 2002543109 A JP2002543109 A JP 2002543109A JP 2000614975 A JP2000614975 A JP 2000614975A JP 2000614975 A JP2000614975 A JP 2000614975A JP 2002543109 A JP2002543109 A JP 2002543109A
- Authority
- JP
- Japan
- Prior art keywords
- dosage form
- drug
- effervescent
- amount
- gastrointestinal tract
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
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- BNIILDVGGAEEIG-UHFFFAOYSA-L disodium hydrogen phosphate Chemical compound [Na+].[Na+].OP([O-])([O-])=O BNIILDVGGAEEIG-UHFFFAOYSA-L 0.000 description 1
- ODQWQRRAPPTVAG-GZTJUZNOSA-N doxepin Chemical compound C1OC2=CC=CC=C2C(=C/CCN(C)C)/C2=CC=CC=C21 ODQWQRRAPPTVAG-GZTJUZNOSA-N 0.000 description 1
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- PJMPHNIQZUBGLI-UHFFFAOYSA-N fentanyl Chemical compound C=1C=CC=CC=1N(C(=O)CC)C(CC1)CCN1CCC1=CC=CC=C1 PJMPHNIQZUBGLI-UHFFFAOYSA-N 0.000 description 1
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- TYJJADVDDVDEDZ-UHFFFAOYSA-M potassium hydrogencarbonate Chemical compound [K+].OC([O-])=O TYJJADVDDVDEDZ-UHFFFAOYSA-M 0.000 description 1
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- 229940010747 sodium hyaluronate Drugs 0.000 description 1
- YWIVKILSMZOHHF-QJZPQSOGSA-N sodium;(2s,3s,4s,5r,6r)-6-[(2s,3r,4r,5s,6r)-3-acetamido-2-[(2s,3s,4r,5r,6r)-6-[(2r,3r,4r,5s,6r)-3-acetamido-2,5-dihydroxy-6-(hydroxymethyl)oxan-4-yl]oxy-2-carboxy-4,5-dihydroxyoxan-3-yl]oxy-5-hydroxy-6-(hydroxymethyl)oxan-4-yl]oxy-3,4,5-trihydroxyoxane-2- Chemical compound [Na+].CC(=O)N[C@H]1[C@H](O)O[C@H](CO)[C@@H](O)[C@@H]1O[C@H]1[C@H](O)[C@@H](O)[C@H](O[C@H]2[C@@H]([C@@H](O[C@H]3[C@@H]([C@@H](O)[C@H](O)[C@H](O3)C(O)=O)O)[C@H](O)[C@@H](CO)O2)NC(C)=O)[C@@H](C(O)=O)O1 YWIVKILSMZOHHF-QJZPQSOGSA-N 0.000 description 1
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- VMYFZRTXGLUXMZ-UHFFFAOYSA-N triethyl citrate Natural products CCOC(=O)C(O)(C(=O)OCC)C(=O)OCC VMYFZRTXGLUXMZ-UHFFFAOYSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0007—Effervescent
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/302,105 | 1999-04-29 | ||
| US09/302,105 US6350470B1 (en) | 1998-04-29 | 1999-04-29 | Effervescent drug delivery system for oral administration |
| PCT/US2000/011053 WO2000066089A1 (en) | 1999-04-29 | 2000-04-25 | Effervescent drug delivery system for oral administration |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2002543109A true JP2002543109A (ja) | 2002-12-17 |
| JP2002543109A5 JP2002543109A5 (https=) | 2011-02-24 |
Family
ID=23166279
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000614975A Pending JP2002543109A (ja) | 1999-04-29 | 2000-04-25 | 経口投与の発泡性薬剤配給系 |
Country Status (6)
| Country | Link |
|---|---|
| US (5) | US6350470B1 (https=) |
| EP (1) | EP1091732A4 (https=) |
| JP (1) | JP2002543109A (https=) |
| AU (1) | AU4488700A (https=) |
| CA (1) | CA2335566C (https=) |
| WO (1) | WO2000066089A1 (https=) |
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| JP2007530530A (ja) * | 2004-03-25 | 2007-11-01 | サン・ファーマシューティカル・インダストリーズ・リミテッド | 胃貯留系 |
| JP2008516893A (ja) * | 2004-08-27 | 2008-05-22 | スフェリックス，インク． | 多層錠剤および生体接着性剤形 |
| JP2008533015A (ja) * | 2005-03-07 | 2008-08-21 | ボストン サイエンティフィック リミティッド | 腔内組織工学のためのマイクロカプセル化された組成物 |
| WO2011118453A1 (ja) * | 2010-03-23 | 2011-09-29 | リンテック株式会社 | 固形製剤 |
| JP2012001542A (ja) * | 2004-06-09 | 2012-01-05 | Glaxosmithkline Llc | 薬剤を製造するための装置及び方法 |
| JP2012162581A (ja) * | 2004-05-28 | 2012-08-30 | Imaginot Pty Ltd | 経口治療用化合物の供給系 |
| JP2013103879A (ja) * | 2011-11-10 | 2013-05-30 | Nakanihon Capsule Co Ltd | ハードカプセル |
| JP2022073316A (ja) * | 2020-10-30 | 2022-05-17 | 株式会社ファンケル | 固体製剤 |
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| US20010055613A1 (en) * | 1998-10-21 | 2001-12-27 | Beth A. Burnside | Oral pulsed dose drug delivery system |
| US6716453B1 (en) * | 1999-05-20 | 2004-04-06 | Verion, Inc. | Method for increasing the active loading of compressible composition forms |
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| DE10120092B4 (de) * | 2001-04-25 | 2008-03-20 | Lts Lohmann Therapie-Systeme Ag | Magensaftresistente Vorrichtung zur Freisetzung von mukoadhäsiven Wirkstoffträgern und Verfahren zur Herstellung der magensaftresistenten Vorrichtung |
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| DE10141650C1 (de) | 2001-08-24 | 2002-11-28 | Lohmann Therapie Syst Lts | Transdermales Therapeutisches System mit Fentanyl bzw. verwandten Substanzen |
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| CN102811712A (zh) * | 2010-03-23 | 2012-12-05 | 琳得科株式会社 | 固体制剂 |
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Also Published As
| Publication number | Publication date |
|---|---|
| CA2335566A1 (en) | 2000-11-09 |
| US20020076439A1 (en) | 2002-06-20 |
| US20030133976A1 (en) | 2003-07-17 |
| US20020071809A1 (en) | 2002-06-13 |
| US6509036B2 (en) | 2003-01-21 |
| US6641838B2 (en) | 2003-11-04 |
| US6391335B1 (en) | 2002-05-21 |
| EP1091732A4 (en) | 2006-01-18 |
| EP1091732A1 (en) | 2001-04-18 |
| AU4488700A (en) | 2000-11-17 |
| US6350470B1 (en) | 2002-02-26 |
| US6764696B2 (en) | 2004-07-20 |
| CA2335566C (en) | 2010-07-06 |
| WO2000066089A1 (en) | 2000-11-09 |
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