JP2002509858A5 - - Google Patents

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Publication number
JP2002509858A5
JP2002509858A5 JP2000526506A JP2000526506A JP2002509858A5 JP 2002509858 A5 JP2002509858 A5 JP 2002509858A5 JP 2000526506 A JP2000526506 A JP 2000526506A JP 2000526506 A JP2000526506 A JP 2000526506A JP 2002509858 A5 JP2002509858 A5 JP 2002509858A5
Authority
JP
Japan
Prior art keywords
alkyl
halo
compound
hydroxy
cycloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2000526506A
Other languages
English (en)
Japanese (ja)
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JP2002509858A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US1998/027822 external-priority patent/WO1999033824A1/en
Publication of JP2002509858A publication Critical patent/JP2002509858A/ja
Publication of JP2002509858A5 publication Critical patent/JP2002509858A5/ja
Pending legal-status Critical Current

Links

JP2000526506A 1997-12-31 1998-12-30 複素環式トポイソメラーゼ毒化合物 Pending JP2002509858A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US7028797P 1997-12-31 1997-12-31
US60/070,287 1997-12-31
PCT/US1998/027822 WO1999033824A1 (en) 1997-12-31 1998-12-30 Heterocyclic topoisomerase poisons

Publications (2)

Publication Number Publication Date
JP2002509858A JP2002509858A (ja) 2002-04-02
JP2002509858A5 true JP2002509858A5 (enExample) 2006-02-16

Family

ID=22094368

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000526506A Pending JP2002509858A (ja) 1997-12-31 1998-12-30 複素環式トポイソメラーゼ毒化合物

Country Status (11)

Country Link
US (3) US6667302B2 (enExample)
EP (1) EP1044199B1 (enExample)
JP (1) JP2002509858A (enExample)
CN (1) CN1299358A (enExample)
AT (1) ATE402168T1 (enExample)
AU (1) AU753268B2 (enExample)
CA (1) CA2316221A1 (enExample)
DE (1) DE69839781D1 (enExample)
IL (1) IL136911A0 (enExample)
PL (1) PL341539A1 (enExample)
WO (1) WO1999033824A1 (enExample)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL136911A0 (en) * 1997-12-31 2001-06-14 Univ Rutgers Heterocyclic topoisomerase poisons
TW200517381A (en) * 2003-08-01 2005-06-01 Genelabs Tech Inc Bicyclic heteroaryl derivatives
RU2007130896A (ru) * 2005-01-14 2009-02-20 Дженелэбс Текнолоджиз, Инк. (Us) Индольные производные для лечения вирусных инфекций
US7998974B2 (en) 2005-03-03 2011-08-16 Sirtris Pharmaceuticals, Inc. Fused heterocyclic compounds and their use as sirtuin modulators
ES2431050T3 (es) 2005-08-04 2013-11-22 Sirtris Pharmaceuticals, Inc. Benzotiazoles y tiazolopiridinas como moduladores de la sirtuína
US8093401B2 (en) 2005-08-04 2012-01-10 Sirtris Pharmaceuticals, Inc. Sirtuin modulating compounds
US7855289B2 (en) 2005-08-04 2010-12-21 Sirtris Pharmaceuticals, Inc. Sirtuin modulating compounds
US8088928B2 (en) 2005-08-04 2012-01-03 Sirtris Pharmaceuticals, Inc. Sirtuin modulating compounds
WO2008073451A2 (en) * 2006-12-11 2008-06-19 Sirtris Pharmaceuticals, Inc. Benzoimidazole derivatives as sirtuin (sir) modulating compounds
CL2008001822A1 (es) 2007-06-20 2009-03-13 Sirtris Pharmaceuticals Inc Compuestos derivados de tiazolo[5,4-b]piridina; composicion farmaceutica que comprende a dichos compuestos; y uso del compuesto en el tratamiento de la resistencia a la insulina, sindrome metabolico, diabetes, entre otras.
BRPI0922435A2 (pt) 2008-12-19 2018-09-11 Sirtris Pharmaceuticals Inc "composto de tiazolopiridina moduladores de sirtuina, composição farmacêutica compreendendo o mesmo e seu uso."
JP6959145B2 (ja) 2015-05-28 2021-11-02 エコラボ ユーエスエー インコーポレイティド プリン系腐食抑制剤及びこれを使用する方法
US10519116B2 (en) 2015-05-28 2019-12-31 Ecolab Usa Inc. Water-soluble pyrazole derivatives as corrosion inhibitors
JP6849608B2 (ja) * 2015-05-28 2021-03-24 エコラボ ユーエスエー インコーポレイティド 新規腐食抑制剤
WO2016191672A1 (en) 2015-05-28 2016-12-01 Ecolab Usa Inc. 2-substituted imidazole and benzimidazole corrosion inhibitors

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US26065A (en) 1859-11-08 Improvement in cotton-gins
USRE26065E (en) 1966-07-19 Folybenzimidazoles and their preparation
US2985661A (en) 1956-02-06 1961-05-23 American Cyanamid Co Preparation of 2(omicron-aminophenyl)-benzimidazole
CH420045A (de) 1964-09-01 1967-03-15 Ciba Geigy Verwendung von neuen Poly-azolen als optische Aufhellmittel für textile organische Materialien
DE1670684A1 (de) * 1966-04-01 1970-12-03 Hoechst Ag Verfahren zur Herstellung von basisch substituierten Bis-benzimidazol-derivaten
SU1530628A1 (ru) 1987-11-20 1989-12-23 Ленинградский Технологический Институт Им.Ленсовета Тригидрохлорид 2-[2-фенил-5(6)-бензимидазолил]-N-(3-диметиламинопропил)-5(6)-бензимидазолкарбоксамида в качестве флуоресцентного красител дл исследовани ДНК
JP2700475B2 (ja) 1988-07-30 1998-01-21 コニカ株式会社 非線形光学材料および非線形光学素子
US5106863A (en) 1990-03-26 1992-04-21 Ortho Pharmaceutical Corporation Substituted imidazole and pyridine derivatives
US5807874A (en) 1995-05-17 1998-09-15 Rutgers, The State University Of New Jersey Trisbenzimidazoles useful as topoisomerase I inhibitors
US5767142A (en) 1996-03-20 1998-06-16 Rutgers, The State University Of New Jersey Trisbenzimidazoles useful as topoisomerase I inhibitors
NZ307959A (en) * 1995-05-17 1998-08-26 Univ Rutgers Substituted tribenzimidazole derivatives where the substituent can be aryl or heteroaryl and medicaments
US5770617A (en) * 1996-03-20 1998-06-23 Rutgers, The State University Of New Jersey Terbenzimidazoles useful as antifungal agents
IL136911A0 (en) * 1997-12-31 2001-06-14 Univ Rutgers Heterocyclic topoisomerase poisons
IL137351A0 (en) * 1998-02-12 2001-07-24 Univ Rutgers Heterocyclic topoisomerase poisons

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