JP2002508364A5 - - Google Patents

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Publication number
JP2002508364A5
JP2002508364A5 JP2000539004A JP2000539004A JP2002508364A5 JP 2002508364 A5 JP2002508364 A5 JP 2002508364A5 JP 2000539004 A JP2000539004 A JP 2000539004A JP 2000539004 A JP2000539004 A JP 2000539004A JP 2002508364 A5 JP2002508364 A5 JP 2002508364A5
Authority
JP
Japan
Prior art keywords
hydrogen
cycloalkyl
alkoxy
alkylthio
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2000539004A
Other languages
English (en)
Japanese (ja)
Other versions
JP2002508364A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US1998/026008 external-priority patent/WO1999031077A1/en
Publication of JP2002508364A publication Critical patent/JP2002508364A/ja
Publication of JP2002508364A5 publication Critical patent/JP2002508364A5/ja
Withdrawn legal-status Critical Current

Links

JP2000539004A 1997-12-16 1998-12-08 セロトニン１ａ受容体に対して活性を有するアリールピペラジン Withdrawn JP2002508364A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US6972297P 1997-12-16 1997-12-16
US6979197P 1997-12-16 1997-12-16
US60/069,791 1997-12-16
US60/069,722 1997-12-16
US8958998P 1998-06-17 1998-06-17
US60/089,589 1998-06-17
PCT/US1998/026008 WO1999031077A1 (en) 1997-12-16 1998-12-08 Arylpiperazines having activity at the serotonin 1a receptor

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2008120430A Division JP2008266337A (ja) 1997-12-16 2008-05-02 セロトニン１ａ受容体に対して活性を有するアリールピペラジン

Publications (2)

Publication Number Publication Date
JP2002508364A JP2002508364A (ja) 2002-03-19
JP2002508364A5 true JP2002508364A5 (enExample) 2005-09-15

Family

ID=27371593

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2000539004A Withdrawn JP2002508364A (ja) 1997-12-16 1998-12-08 セロトニン１ａ受容体に対して活性を有するアリールピペラジン
JP2008120430A Pending JP2008266337A (ja) 1997-12-16 2008-05-02 セロトニン１ａ受容体に対して活性を有するアリールピペラジン

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2008120430A Pending JP2008266337A (ja) 1997-12-16 2008-05-02 セロトニン１ａ受容体に対して活性を有するアリールピペラジン

Country Status (32)

Country Link
US (9) US6239135B1 (enExample)
EP (2) EP0924205B1 (enExample)
JP (2) JP2002508364A (enExample)
KR (1) KR100539651B1 (enExample)
CN (2) CN100355714C (enExample)
AR (1) AR017864A1 (enExample)
AT (1) ATE296296T1 (enExample)
AU (1) AU747040B2 (enExample)
BR (1) BR9814280A (enExample)
CA (2) CA2315227C (enExample)
CO (1) CO4980859A1 (enExample)
DE (1) DE69830297T2 (enExample)
DK (1) DK0924205T3 (enExample)
EA (1) EA003703B1 (enExample)
EG (1) EG23983A (enExample)
ES (1) ES2244036T3 (enExample)
HR (1) HRP20000406B1 (enExample)
HU (1) HU226409B1 (enExample)
ID (1) ID26930A (enExample)
IL (3) IL136723A0 (enExample)
MY (1) MY125868A (enExample)
NO (1) NO317098B1 (enExample)
NZ (1) NZ505220A (enExample)
PE (1) PE20000134A1 (enExample)
PL (1) PL193428B1 (enExample)
PT (1) PT924205E (enExample)
SV (1) SV1998000148A (enExample)
TR (1) TR200001727T2 (enExample)
TW (1) TW520366B (enExample)
UA (1) UA66370C2 (enExample)
WO (1) WO1999031077A1 (enExample)
ZA (1) ZA9811473B (enExample)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA66370C2 (en) * 1997-12-16 2004-05-17 Lilly Co Eli Arylpiperazines having activity to setotonin 1 receptors
CZ299712B6 (cs) 1999-09-03 2008-10-29 Apbi Holdings, Llc Použití dapoxetinu pro zvládnutí sexuální dysfunkce podáváním zpusobem podle potreby
EP1286980A2 (en) * 2000-03-24 2003-03-05 Eli Lilly And Company Enantioselective process for preparing arylated lactones and derivatives
WO2002069973A1 (en) 2001-03-02 2002-09-12 Sepracor, Inc. Piperidine-piperazine ligand for neurotransmitter receptors
DE10161809A1 (de) * 2001-12-14 2003-06-26 Gruenenthal Gmbh Arzneimittel enthaltend N,N'-disubstituierte Piperazin-Verbindungen
DE10161644A1 (de) * 2001-12-14 2003-06-26 Gruenenthal Gmbh N,N'-disubstituierte Piperazin-Verbindungen
DE10205721A1 (de) * 2002-02-12 2003-08-21 Biotronik Mess & Therapieg Führungsdraht und implantierbare Elektrodenleitung
US20030189215A1 (en) 2002-04-09 2003-10-09 Jong-Lam Lee Method of fabricating vertical structure leds
ITMI20021328A1 (it) * 2002-06-14 2003-12-15 Recordati Ind Chimica E Farma Nuove piperazine 1,4 - disostituite
US20040072839A1 (en) * 2002-06-14 2004-04-15 Amedeo Leonardi 1-Phenylalkylpiperazines
ITMI20021329A1 (it) * 2002-06-14 2003-12-15 Recordati Chem Pharm Nuove ossialchilammine sostituite
US7071197B2 (en) 2002-06-14 2006-07-04 Recordati S.A. N,N-disubstituted diazocycloalkanes
ITMI20021327A1 (it) * 2002-06-14 2003-12-15 Recordati Chem Pharm Nuove ossialchilpiperazine
US20040197397A1 (en) * 2002-08-30 2004-10-07 Watson Pharmaceuticals, Inc. Drug delivery system for treatment of urinary incontinence
HRP20050533A2 (en) * 2002-12-12 2006-11-30 Aventis Pharma S.A. Aminoindazole derivatives and use thereof as kinase inhibitors
GB0317370D0 (en) * 2003-07-24 2003-08-27 Synaptics Uk Ltd Magnetic calibration array
US20050165025A1 (en) * 2004-01-22 2005-07-28 Recordati Ireland Ltd. Combination therapy with 5HT 1A and 5HT 1B-receptor antagonists
AU2005289808B2 (en) * 2004-09-24 2011-11-03 The Government Of The United States As Represented By The Secretary Of The Army, U.S. Army Medical Research Institute Of Chemical Defense Method of treating organophosphorous poisoning
US9132135B2 (en) * 2004-09-24 2015-09-15 University Of Maryland, Baltimore Method of treating organophosphorous poisoning
US20070202140A1 (en) * 2005-12-22 2007-08-30 Veltri Enrico P Thrombin receptor antagonists as prophylaxis to complications from cardiopulmonary surgery
US20080081067A1 (en) * 2006-10-03 2008-04-03 Gupta Manishkumar Sustained release pharmaceutical compositions of venlafaxine and process for preparation thereof
MX2011005801A (es) * 2008-12-01 2011-06-20 Procter & Gamble Sistemas de perfume.
ES2424122T3 (es) * 2009-11-06 2013-09-27 Aerpio Therapeutics Inc. Inhibidores de la prolilhidroxilasa
WO2012078934A2 (en) 2010-12-08 2012-06-14 Expression Pathology, Inc. Truncated her2 srm/mrm assay
CN110713442A (zh) * 2018-07-11 2020-01-21 程先波 一种邻硝基苯甲醛的制备方法

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB230303A (enExample) * 1900-01-01
US1013907A (en) * 1910-08-22 1912-01-09 David M Neuberger Engine.
BE637389A (enExample) * 1962-09-13
GB1013907A (en) * 1962-09-13 1965-12-22 Ici Ltd Alkene derivatives
GB8909209D0 (en) 1989-04-22 1989-06-07 Wyeth John & Brother Ltd Piperazine derivatives
US5340812A (en) 1989-04-22 1994-08-23 John Wyeth & Brother, Limited Piperazine derivatives
US5382583A (en) 1989-04-22 1995-01-17 John Wyeth & Brother, Limited Piperazine derivatives
GB9021535D0 (en) 1990-10-03 1990-11-14 Wyeth John & Brother Ltd Piperazine derivatives
GB2248499A (en) 1990-10-05 1992-04-08 Richard Branson Seismic data interpretation digitising scanner
IL101722A (en) 1991-05-02 1996-05-14 Wyeth John & Brother Ltd Piperazine derivatives their preparation and pharmaceutical compositions containing them
TW224974B (enExample) 1991-07-02 1994-06-11 Hoffmann La Roche
CN1036395C (zh) 1992-03-19 1997-11-12 约翰韦恩兄弟有限公司 哌嗪衍生物的制备方法
GB9306103D0 (en) 1993-03-24 1993-05-12 Wyeth John & Brother Ltd Piperazine derivatives
JPH06293803A (ja) 1993-11-26 1994-10-21 Loctite Corp 光硬化性組成物
EP0661266A1 (en) 1993-12-27 1995-07-05 Toa Eiyo Ltd. Substituted cyclic amine compounds as 5HT2 antagonists
US5614523A (en) * 1995-01-17 1997-03-25 Eli Lilly And Company Compounds having effects on serotonin-related systems
GB9514384D0 (en) * 1995-07-13 1995-09-13 American Home Prod Medical treatment
UA66370C2 (en) * 1997-12-16 2004-05-17 Lilly Co Eli Arylpiperazines having activity to setotonin 1 receptors
EP1286980A2 (en) * 2000-03-24 2003-03-05 Eli Lilly And Company Enantioselective process for preparing arylated lactones and derivatives

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