JP2001515895A5 - - Google Patents
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- Publication number
- JP2001515895A5 JP2001515895A5 JP2000510727A JP2000510727A JP2001515895A5 JP 2001515895 A5 JP2001515895 A5 JP 2001515895A5 JP 2000510727 A JP2000510727 A JP 2000510727A JP 2000510727 A JP2000510727 A JP 2000510727A JP 2001515895 A5 JP2001515895 A5 JP 2001515895A5
- Authority
- JP
- Japan
- Prior art keywords
- acid
- cvi
- formula
- hydroxylactone
- producing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US5861897P | 1997-09-11 | 1997-09-11 | |
| US60/058,618 | 1997-09-11 | ||
| PCT/US1998/017993 WO1999012919A1 (en) | 1997-09-11 | 1998-09-03 | Process to produce 4-hydroxy-2-oxo-pyrane derivates useful as protease inhibitors |
Related Child Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009022289A Division JP5016621B2 (ja) | 1997-09-11 | 2009-02-03 | プロテアーゼインヒビターとして有用な４−ヒドロキシ−２−オキソ−ピラン誘導体の製法 |
| JP2009280318A Division JP5266194B2 (ja) | 1997-09-11 | 2009-12-10 | プロテアーゼインヒビターとして有用な４−ヒドロキシ−２−オキソ−ピラン誘導体の製法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2001515895A JP2001515895A (ja) | 2001-09-25 |
| JP2001515895A5 true JP2001515895A5 (https=) | 2006-01-05 |
| JP4462760B2 JP4462760B2 (ja) | 2010-05-12 |
Family
ID=22017924
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000510727A Expired - Lifetime JP4462760B2 (ja) | 1997-09-11 | 1998-09-03 | プロテアーゼインヒビターとして有用な４−ヒドロキシ−２−オキソ−ピラン誘導体の製法 |
| JP2009022289A Expired - Lifetime JP5016621B2 (ja) | 1997-09-11 | 2009-02-03 | プロテアーゼインヒビターとして有用な４−ヒドロキシ−２−オキソ−ピラン誘導体の製法 |
| JP2009280318A Expired - Lifetime JP5266194B2 (ja) | 1997-09-11 | 2009-12-10 | プロテアーゼインヒビターとして有用な４−ヒドロキシ−２−オキソ−ピラン誘導体の製法 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009022289A Expired - Lifetime JP5016621B2 (ja) | 1997-09-11 | 2009-02-03 | プロテアーゼインヒビターとして有用な４−ヒドロキシ−２−オキソ−ピラン誘導体の製法 |
| JP2009280318A Expired - Lifetime JP5266194B2 (ja) | 1997-09-11 | 2009-12-10 | プロテアーゼインヒビターとして有用な４−ヒドロキシ−２−オキソ−ピラン誘導体の製法 |
Country Status (20)
| Country | Link |
|---|---|
| US (2) | US6077963A (https=) |
| EP (1) | EP1015441B1 (https=) |
| JP (3) | JP4462760B2 (https=) |
| KR (1) | KR100569771B1 (https=) |
| CN (3) | CN1284763C (https=) |
| AT (1) | ATE266654T1 (https=) |
| CA (1) | CA2300204C (https=) |
| CZ (1) | CZ298847B6 (https=) |
| DE (1) | DE69823844T2 (https=) |
| DK (1) | DK1015441T3 (https=) |
| ES (1) | ES2221199T3 (https=) |
| FI (1) | FI120973B (https=) |
| HU (1) | HU228986B1 (https=) |
| NO (1) | NO321835B1 (https=) |
| NZ (1) | NZ503338A (https=) |
| PL (1) | PL193240B1 (https=) |
| PT (1) | PT1015441E (https=) |
| RU (2) | RU2223958C2 (https=) |
| SK (1) | SK284974B6 (https=) |
| WO (1) | WO1999012919A1 (https=) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU3699100A (en) | 1999-03-18 | 2000-10-04 | Pharmacia & Upjohn Company | Improved process for asymmetric hydrogenation |
| US6552204B1 (en) * | 2000-02-04 | 2003-04-22 | Roche Colorado Corporation | Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-pyran-2-one |
| US6500963B2 (en) | 2001-02-22 | 2002-12-31 | Boehringer Ingelheim Pharma Kg | Process for preparing optically active dihydropyrones |
| DE10108470A1 (de) * | 2001-02-22 | 2002-09-05 | Boehringer Ingelheim Pharma | Verfahren zur Herstellung optisch aktiver Dihydropyrone |
| US6987123B2 (en) | 2001-07-26 | 2006-01-17 | Cadila Healthcare Limited | Heterocyclic compounds, their preparation, pharmaceutical compositions containing them and their use in medicine |
| DE60234537D1 (de) | 2002-02-07 | 2010-01-07 | Sumitomo Chemical Co | Verfahren zur herstellung von (r)-3-hydroxy-3-(2-phenylethyl) hexansäure und dessen zwischenprodukt |
| DE10313118A1 (de) | 2003-03-24 | 2004-10-07 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Enantioselektive Hydrierung von Intermediaten bei der Tipranavir-Synthese |
| US7512945B2 (en) * | 2003-12-29 | 2009-03-31 | Intel Corporation | Method and apparatus for scheduling the processing of commands for execution by cryptographic algorithm cores in a programmable network processor |
| CN100448836C (zh) * | 2005-06-03 | 2009-01-07 | 浙江中贝化工有限公司 | 一种抗艾滋病药物关键中间体的制备方法 |
| CN102336758A (zh) * | 2005-08-24 | 2012-02-01 | 辉瑞有限公司 | 作为hcv聚合酶抑制剂的化合物及组合物 |
| KR101548306B1 (ko) * | 2007-11-30 | 2015-08-28 | 가부시키가이샤 한도오따이 에네루기 켄큐쇼 | 발광 소자, 발광 장치 및 전자기기 |
| US8853393B2 (en) * | 2011-07-29 | 2014-10-07 | Anhui New Star Pharmaceutical Development Co., Ltd. | Intermediate for preparing tapentadol or analogues thereof |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1355667A (fr) * | 1963-02-05 | 1964-03-20 | Meci Materiel Elect Contr | Gaine tubulaire pour électrode servant à la mesure du ph |
| FR1355668A (fr) * | 1963-02-05 | 1964-03-20 | Moteur rotatif à combustion interne perfectionné | |
| FR2096877B1 (https=) * | 1970-07-09 | 1973-08-10 | Hexachimie | |
| JPH0665657B2 (ja) * | 1984-11-08 | 1994-08-24 | 日本化薬株式会社 | 光学活性マンデル酸の製法 |
| JPH072677B2 (ja) * | 1988-02-19 | 1995-01-18 | 株式会社クラレ | （±）―２―ヒドロキシ―４―フェニルブタン酸の光学分割法 |
| JPH01221345A (ja) * | 1988-02-27 | 1989-09-04 | Ajinomoto Co Inc | マンデル酸誘導体の光学分割方法 |
| JP3084577B2 (ja) * | 1991-09-27 | 2000-09-04 | 山川薬品工業株式会社 | 光学活性なアトロラクチン酸の製造方法および製造の中間体 |
| JP3178086B2 (ja) * | 1992-06-17 | 2001-06-18 | 山川薬品工業株式会社 | 光学活性α−メチルベンジルアミンの製造方法 |
| ZA938019B (en) * | 1992-11-13 | 1995-04-28 | Upjohn Co | Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating HIV and other retroviruses |
| DE69433705T2 (de) * | 1993-11-19 | 2005-03-10 | Parke, Davis & Company | 5,6-Dihydropyronderivate als Proteaseinhibitoren und Antiviralmittel |
| IL129871A (en) * | 1994-05-06 | 2003-11-23 | Pharmacia & Upjohn Inc | Process for preparing 4-phenyl-substituted octanoyl-oxazolidin-2-one intermediates that are useful for preparing pyran-2-ones useful for treating retroviral infections |
| RU2074169C1 (ru) * | 1995-05-10 | 1997-02-27 | Акционерное общество открытого типа "Химпром" | Способ получения этилового эфира п-нитробензойной кислоты |
-
1998
- 1998-09-03 JP JP2000510727A patent/JP4462760B2/ja not_active Expired - Lifetime
- 1998-09-03 DE DE69823844T patent/DE69823844T2/de not_active Expired - Lifetime
- 1998-09-03 PT PT98945806T patent/PT1015441E/pt unknown
- 1998-09-03 EP EP98945806A patent/EP1015441B1/en not_active Expired - Lifetime
- 1998-09-03 RU RU2000109277/04A patent/RU2223958C2/ru active
- 1998-09-03 CA CA002300204A patent/CA2300204C/en not_active Expired - Lifetime
- 1998-09-03 WO PCT/US1998/017993 patent/WO1999012919A1/en not_active Ceased
- 1998-09-03 CN CNB031594735A patent/CN1284763C/zh not_active Expired - Lifetime
- 1998-09-03 CZ CZ20000804A patent/CZ298847B6/cs not_active IP Right Cessation
- 1998-09-03 HU HU0003593A patent/HU228986B1/hu unknown
- 1998-09-03 KR KR1020007002546A patent/KR100569771B1/ko not_active Expired - Lifetime
- 1998-09-03 ES ES98945806T patent/ES2221199T3/es not_active Expired - Lifetime
- 1998-09-03 SK SK226-2000A patent/SK284974B6/sk not_active IP Right Cessation
- 1998-09-03 DK DK98945806T patent/DK1015441T3/da active
- 1998-09-03 CN CNB2007100079776A patent/CN100471832C/zh not_active Expired - Lifetime
- 1998-09-03 NZ NZ503338A patent/NZ503338A/en not_active IP Right Cessation
- 1998-09-03 PL PL339138A patent/PL193240B1/pl unknown
- 1998-09-03 AT AT98945806T patent/ATE266654T1/de active
- 1998-09-03 CN CNB988087111A patent/CN1298714C/zh not_active Expired - Lifetime
- 1998-12-17 US US09/213,887 patent/US6077963A/en not_active Expired - Lifetime
-
2000
- 2000-02-28 US US09/514,087 patent/US6265604B1/en not_active Expired - Lifetime
- 2000-03-10 NO NO20001274A patent/NO321835B1/no not_active IP Right Cessation
- 2000-03-10 FI FI20000553A patent/FI120973B/fi not_active IP Right Cessation
-
2003
- 2003-10-21 RU RU2003131081/04A patent/RU2263106C2/ru active
-
2009
- 2009-02-03 JP JP2009022289A patent/JP5016621B2/ja not_active Expired - Lifetime
- 2009-12-10 JP JP2009280318A patent/JP5266194B2/ja not_active Expired - Lifetime
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