JP2001507708A - 炎症の局所治療用製剤を調製する為のジクロロベンジルアルコールの使用及びジクロロベンジルアルコールを含有する製剤 - Google Patents
炎症の局所治療用製剤を調製する為のジクロロベンジルアルコールの使用及びジクロロベンジルアルコールを含有する製剤Info
- Publication number
- JP2001507708A JP2001507708A JP53047998A JP53047998A JP2001507708A JP 2001507708 A JP2001507708 A JP 2001507708A JP 53047998 A JP53047998 A JP 53047998A JP 53047998 A JP53047998 A JP 53047998A JP 2001507708 A JP2001507708 A JP 2001507708A
- Authority
- JP
- Japan
- Prior art keywords
- dichlorobenzyl alcohol
- inflammation
- formulation
- weight
- treatment
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q11/00—Preparations for care of the teeth, of the oral cavity or of dentures; Dentifrices, e.g. toothpastes; Mouth rinses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
- A61K8/34—Alcohols
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q17/00—Barrier preparations; Preparations brought into direct contact with the skin for affording protection against external influences, e.g. sunlight, X-rays or other harmful rays, corrosive materials, bacteria or insect stings
- A61Q17/005—Antimicrobial preparations
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Birds (AREA)
- Oral & Maxillofacial Surgery (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Description
Claims (1)
- 【特許請求の範囲】 1.炎症の局所治療用製剤の調製の為のジクロロベンジルアルコールの使用。 2.ジクロロベンジルアルコールが、2,4−ジクロロベンジルアルコールであ る、請求項1に記載の使用。 3.ジクロロベンジルアルコールが、治療部位において、ジクロロベンジルアル コールの調節された放出及び/又は長期保持を提供する一種以上の物質と組合 される、請求項1に記載の使用。 4.ジクロロベンジルアルコールが、一種以上の生体接着材料と組合される、請 求項3に記載の使用。 5.生体接着材料が、ナトリウムカルボキシセルロース、カルボポール、トラガ ント、カラヤゴム、アルギン酸ナトリウム、ゼラチン、メチルセルロース及び アラビヤゴムの様な親水性コロイドの中から選ばれる、請求項3又は4に記載 の使用。 6.製剤が、皮膚又は粘膜上に適用される為に調剤される、請求項1に記載の使 用。 7.製剤が、経口内及び/又は外部使用の為に調剤される、請求項3に記載の使 用。 8.ジクロロベンジルアルコール、好ましくは2,4−ジクロロベンジルアルコ ールを活性成分として含む事を特徴とする、炎症の局所治療用製剤。 9.活性成分に加えて、生体増粘剤及び水を含む、請求項8に記載の製剤。 10.0.05〜2重量%、好ましくは約1重量%のジクロロベンジルアルコール 、0.1〜10重量%、好ましくは約2重量%の生体接着材料及び90〜99 重量%、好ましくは97重量%の水から成る、請求項9に記載の製剤。 11.生体増粘剤が、ナトリウムカルボキシメチルセルロース、カルボポール、ト ラガント、カラヤゴム、アルギン酸ナトリウム、ゼラチン、メチルセルロース 、アラビヤゴムの様な親水性コロイドム、好ましくはナトリウムカルボキシメ チルセルロースから選ばれる、請求項9又は10に記載の製剤。
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DK2697 | 1997-01-09 | ||
DK0026/97 | 1997-01-09 | ||
PCT/DK1998/000011 WO1998030214A1 (en) | 1997-01-09 | 1998-01-09 | Use of dichlorobenzyl alcohol for preparing a preparation for topical treatment of inflammation and a preparation containing dichlorobenzyl alcohol |
Publications (3)
Publication Number | Publication Date |
---|---|
JP2001507708A true JP2001507708A (ja) | 2001-06-12 |
JP2001507708A5 JP2001507708A5 (ja) | 2005-07-14 |
JP4663036B2 JP4663036B2 (ja) | 2011-03-30 |
Family
ID=8088912
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP53047998A Expired - Fee Related JP4663036B2 (ja) | 1997-01-09 | 1998-01-09 | 炎症の局所治療用製剤を調製する為のジクロロベンジルアルコールの使用及びジクロロベンジルアルコールを含有する製剤 |
Country Status (18)
Country | Link |
---|---|
US (1) | US6251371B1 (ja) |
EP (1) | EP0988033B1 (ja) |
JP (1) | JP4663036B2 (ja) |
KR (1) | KR100573206B1 (ja) |
CN (1) | CN1128614C (ja) |
AT (1) | ATE206047T1 (ja) |
AU (1) | AU719836B2 (ja) |
BR (1) | BR9807056A (ja) |
CA (1) | CA2277207C (ja) |
DE (1) | DE69801820T2 (ja) |
DK (1) | DK0988033T3 (ja) |
ES (1) | ES2162410T3 (ja) |
NO (1) | NO328979B1 (ja) |
NZ (1) | NZ336600A (ja) |
PL (1) | PL189398B1 (ja) |
PT (1) | PT988033E (ja) |
RU (1) | RU2184538C2 (ja) |
WO (1) | WO1998030214A1 (ja) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL137891A (en) | 1998-03-19 | 2005-03-20 | Bifodan As | Disinfecting composition |
EP1488797B1 (en) * | 2000-12-08 | 2008-04-23 | Kyowa Hakko Kogyo Co., Ltd. | Oral preprations having itching-relieving or antipruritic activity |
US7887842B2 (en) | 2003-02-07 | 2011-02-15 | Teikoku Pharma Usa, Inc. | Methods of administering a dermatological agent to a subject |
MX2012010769A (es) * | 2010-03-19 | 2013-02-27 | Oxygen Biotherapeutics Inc | Formulaciones perfluorocarbonadas oftalmicas en forma de crema. |
WO2012044963A2 (en) * | 2010-10-01 | 2012-04-05 | Oxygen Biotherapeutics, Inc. | Perfluorocarbons for use in treating pruritus |
CN104173204B (zh) * | 2014-09-17 | 2015-03-11 | 沈广阳 | 一种水包油乳液组合物 |
US20170312211A1 (en) * | 2014-09-26 | 2017-11-02 | Koninklijke Philips N.V. | Applicator for an oral care composition |
US9980975B2 (en) | 2015-01-22 | 2018-05-29 | Ems S.A. | Dosage forms containing fluticasone propionate for the treatment of inflammatory conditions of the esophagus |
CN111297802A (zh) * | 2018-12-12 | 2020-06-19 | 成都一平医药科技发展有限公司 | 一种用于抗炎及抗菌的组合物 |
Citations (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3123528A (en) * | 1964-03-03 | New therapeutic compositions | ||
JPH06172178A (ja) * | 1992-06-29 | 1994-06-21 | Merck & Co Inc | モルホリン及びチオモルホリンタチキニンレセプタ ーアンタゴニスト |
JPH06506919A (ja) * | 1991-04-15 | 1994-08-04 | スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー | 胃炎治療用医薬組成物 |
WO1994018165A1 (en) * | 1993-02-12 | 1994-08-18 | Pfizer Inc. | Sulfonamide compounds as opioid k-receptor agonists |
JPH07242666A (ja) * | 1994-03-08 | 1995-09-19 | Fujisawa Pharmaceut Co Ltd | 複素環化合物 |
WO1995026134A1 (en) * | 1994-03-28 | 1995-10-05 | The Trustees Of Columbia University In The City Of New York | Composition for inactivating irritants in fluids |
WO1995035103A1 (en) * | 1994-06-20 | 1995-12-28 | Kurt Berg | A pharmaceutical composition for the prevention and/or treatment of viral infections and optionally inflammations as well as a method for the treatment thereof |
JPH08225424A (ja) * | 1994-12-13 | 1996-09-03 | San Medical Kk | 象牙質知覚過敏症用歯科用組成物 |
WO1996029867A2 (en) * | 1995-03-31 | 1996-10-03 | Guthery B Eugene | Fast acting and persistent topical antiseptic |
WO1996032934A1 (en) * | 1995-04-18 | 1996-10-24 | The Boots Company Plc | 2,4-dichlorobenzyl alcohol and amylmetacresol against hiv infection |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE750969A (fr) * | 1970-05-26 | 1970-11-03 | Geigy Ag J R | Composition pour combattre les micro-organismes, |
US4167583A (en) * | 1973-07-03 | 1979-09-11 | Bayer Aktiengesellschaft | Microbial composition and formulations |
GB8411731D0 (en) * | 1984-05-09 | 1984-06-13 | Unilever Plc | Oral compositions |
US4663077A (en) * | 1984-06-11 | 1987-05-05 | Morton Thiokol Inc. | Microbiocidal compositions comprising an aryl alkanol and a microbiocidal compound dissolved therein |
CA2165013C (en) * | 1994-12-13 | 2004-01-06 | Nobuo Nakabayashi | Dental composition for relieving dentin hypersensitivity |
IT1275955B1 (it) * | 1995-03-22 | 1997-10-24 | Dompe Spa | Formulazioni farmaceutiche in forma di gel tissotropico |
EP0852941B1 (de) * | 1996-12-13 | 2003-05-14 | Vesifact Ag | Kosmetische Präparate in Form einer Nanodispersion |
US5989527A (en) * | 1998-01-26 | 1999-11-23 | Inolex Investment Corporation | Compositions and methods for improving the performance of chemical exfoliating agents, sunless tanning agents, skin lightening agents and insect repellents |
-
1998
- 1998-01-09 DE DE69801820T patent/DE69801820T2/de not_active Expired - Lifetime
- 1998-01-09 CA CA002277207A patent/CA2277207C/en not_active Expired - Fee Related
- 1998-01-09 CN CN98801761A patent/CN1128614C/zh not_active Expired - Fee Related
- 1998-01-09 BR BR9807056-8A patent/BR9807056A/pt not_active Application Discontinuation
- 1998-01-09 PT PT98900272T patent/PT988033E/pt unknown
- 1998-01-09 PL PL98334679A patent/PL189398B1/pl not_active IP Right Cessation
- 1998-01-09 JP JP53047998A patent/JP4663036B2/ja not_active Expired - Fee Related
- 1998-01-09 DK DK98900272T patent/DK0988033T3/da active
- 1998-01-09 EP EP98900272A patent/EP0988033B1/en not_active Expired - Lifetime
- 1998-01-09 AT AT98900272T patent/ATE206047T1/de active
- 1998-01-09 NZ NZ336600A patent/NZ336600A/xx not_active IP Right Cessation
- 1998-01-09 US US09/341,427 patent/US6251371B1/en not_active Expired - Lifetime
- 1998-01-09 ES ES98900272T patent/ES2162410T3/es not_active Expired - Lifetime
- 1998-01-09 RU RU99117143/14A patent/RU2184538C2/ru active
- 1998-01-09 WO PCT/DK1998/000011 patent/WO1998030214A1/en active IP Right Grant
- 1998-01-09 AU AU54783/98A patent/AU719836B2/en not_active Ceased
- 1998-01-09 KR KR1019997006205A patent/KR100573206B1/ko not_active IP Right Cessation
-
1999
- 1999-07-07 NO NO19993355A patent/NO328979B1/no not_active IP Right Cessation
Patent Citations (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3123528A (en) * | 1964-03-03 | New therapeutic compositions | ||
JPH06506919A (ja) * | 1991-04-15 | 1994-08-04 | スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー | 胃炎治療用医薬組成物 |
JPH06172178A (ja) * | 1992-06-29 | 1994-06-21 | Merck & Co Inc | モルホリン及びチオモルホリンタチキニンレセプタ ーアンタゴニスト |
WO1994018165A1 (en) * | 1993-02-12 | 1994-08-18 | Pfizer Inc. | Sulfonamide compounds as opioid k-receptor agonists |
JPH07242666A (ja) * | 1994-03-08 | 1995-09-19 | Fujisawa Pharmaceut Co Ltd | 複素環化合物 |
WO1995026134A1 (en) * | 1994-03-28 | 1995-10-05 | The Trustees Of Columbia University In The City Of New York | Composition for inactivating irritants in fluids |
WO1995035103A1 (en) * | 1994-06-20 | 1995-12-28 | Kurt Berg | A pharmaceutical composition for the prevention and/or treatment of viral infections and optionally inflammations as well as a method for the treatment thereof |
JPH08225424A (ja) * | 1994-12-13 | 1996-09-03 | San Medical Kk | 象牙質知覚過敏症用歯科用組成物 |
WO1996029867A2 (en) * | 1995-03-31 | 1996-10-03 | Guthery B Eugene | Fast acting and persistent topical antiseptic |
WO1996032934A1 (en) * | 1995-04-18 | 1996-10-24 | The Boots Company Plc | 2,4-dichlorobenzyl alcohol and amylmetacresol against hiv infection |
Also Published As
Publication number | Publication date |
---|---|
BR9807056A (pt) | 2000-05-02 |
CN1128614C (zh) | 2003-11-26 |
KR100573206B1 (ko) | 2006-04-28 |
WO1998030214A1 (en) | 1998-07-16 |
CN1243437A (zh) | 2000-02-02 |
NO328979B1 (no) | 2010-07-05 |
PT988033E (pt) | 2002-02-28 |
PL334679A1 (en) | 2000-03-13 |
ATE206047T1 (de) | 2001-10-15 |
CA2277207A1 (en) | 1998-07-16 |
JP4663036B2 (ja) | 2011-03-30 |
RU2184538C2 (ru) | 2002-07-10 |
EP0988033A1 (en) | 2000-03-29 |
CA2277207C (en) | 2008-02-19 |
AU5478398A (en) | 1998-08-03 |
DE69801820T2 (de) | 2002-04-11 |
NO993355D0 (no) | 1999-07-07 |
ES2162410T3 (es) | 2001-12-16 |
EP0988033B1 (en) | 2001-09-26 |
KR20000069990A (ko) | 2000-11-25 |
DK0988033T3 (da) | 2001-10-22 |
PL189398B1 (pl) | 2005-07-29 |
AU719836B2 (en) | 2000-05-18 |
NO993355L (no) | 1999-08-18 |
DE69801820D1 (de) | 2001-10-31 |
US6251371B1 (en) | 2001-06-26 |
NZ336600A (en) | 2000-07-28 |
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