JP2000513020A - イヌにおける疼痛および炎症治療用ｃｏｘ−２選択性カルプロフェン - Google Patents
イヌにおける疼痛および炎症治療用ｃｏｘ−２選択性カルプロフェンInfo
- Publication number
- JP2000513020A JP2000513020A JP10547869A JP54786998A JP2000513020A JP 2000513020 A JP2000513020 A JP 2000513020A JP 10547869 A JP10547869 A JP 10547869A JP 54786998 A JP54786998 A JP 54786998A JP 2000513020 A JP2000513020 A JP 2000513020A
- Authority
- JP
- Japan
- Prior art keywords
- cox
- inhibitor
- carprofen
- inflammation
- activity
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US4563597P | 1997-05-05 | 1997-05-05 | |
| US60/045,635 | 1997-05-05 | ||
| PCT/IB1998/000662 WO1998050033A1 (fr) | 1997-05-05 | 1998-05-01 | Carprofene inhibant selectivement cox-2 et utilise dans le traitement de la douleur et des inflammations chez les chiens |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JP2000513020A true JP2000513020A (ja) | 2000-10-03 |
Family
ID=21939053
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP10547869A Pending JP2000513020A (ja) | 1997-05-05 | 1998-05-01 | イヌにおける疼痛および炎症治療用ｃｏｘ−２選択性カルプロフェン |
Country Status (32)
| Country | Link |
|---|---|
| EP (1) | EP0988034A1 (fr) |
| JP (1) | JP2000513020A (fr) |
| KR (2) | KR20040004406A (fr) |
| CN (1) | CN1255059A (fr) |
| AP (1) | AP9801234A0 (fr) |
| AR (2) | AR011726A1 (fr) |
| AU (1) | AU6932198A (fr) |
| BG (1) | BG103852A (fr) |
| BR (1) | BR9808720A (fr) |
| CA (1) | CA2288759A1 (fr) |
| DZ (1) | DZ2479A1 (fr) |
| EA (1) | EA003696B1 (fr) |
| GT (1) | GT199800063A (fr) |
| HR (1) | HRP980244A2 (fr) |
| HU (1) | HUP0001286A3 (fr) |
| ID (1) | ID21311A (fr) |
| IL (1) | IL132570A0 (fr) |
| IS (1) | IS5220A (fr) |
| MA (1) | MA26491A1 (fr) |
| NO (1) | NO995389L (fr) |
| NZ (1) | NZ500183A (fr) |
| OA (1) | OA11213A (fr) |
| PA (1) | PA8450601A1 (fr) |
| PE (1) | PE72599A1 (fr) |
| PL (1) | PL337003A1 (fr) |
| SK (1) | SK148199A3 (fr) |
| TN (1) | TNSN98059A1 (fr) |
| TW (1) | TW590773B (fr) |
| UY (1) | UY24989A1 (fr) |
| WO (1) | WO1998050033A1 (fr) |
| YU (1) | YU55899A (fr) |
| ZA (1) | ZA983722B (fr) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6245797B1 (en) | 1997-10-22 | 2001-06-12 | Merck & Co., Inc. | Combination therapy for reducing the risks associated with cardio-and-cerebrovascular disease |
| AU2003204888B2 (en) * | 1998-05-22 | 2005-07-28 | Pfizer Products Inc. | Treating or Preventing the Early Stages of Degeneration of Articular Cartilage or Subchondral Bone in Mammals Using Carprofen and Derivatives |
| US6506785B2 (en) | 1998-05-22 | 2003-01-14 | Pfizer, Inc. | Treating or preventing the early stages of degeneration of articular cartilage or subchondral bone in mammals using carprofen and derivatives |
| AU764872B2 (en) * | 1998-10-23 | 2003-09-04 | Merck Frosst Canada & Co. | Combination product comprising an E-type prostaglandin ligand and a cox-2 selective inhibitor and methods of use |
| WO2000053149A2 (fr) * | 1999-03-10 | 2000-09-14 | G.D. Searle & Co. | Procede et composition se rapportant a l'administration d'un inhibiteur de la cyclo-oxygenase-2 |
| WO2001034204A1 (fr) * | 1999-11-11 | 2001-05-17 | Eli Lilly And Company | Produits composes oncolytiques destines au traitement du cancer |
| JP2004521856A (ja) * | 2000-05-15 | 2004-07-22 | メルク フロスト カナダ アンド カンパニー | Ｃｏｘ−２選択的阻害剤およびトロンボキサン阻害剤を用いる併用療法ならびにそのための組成物 |
| RU2003100874A (ru) | 2000-06-13 | 2004-06-27 | Вайс (Us) | Болеутоляющие и противовоспалительные составы, содержащие ингибиторы циклооксигеназы-2 |
| DE10032132A1 (de) * | 2000-07-01 | 2002-01-17 | Lohmann Therapie Syst Lts | Dermales Therapeutisches System enthaltend nichtsteroidale Antiphlogistika mit selektiver COX-2-Hemmung |
| US7189504B2 (en) | 2000-08-07 | 2007-03-13 | Vanderbilt University | Compositions and methods for detecting and quantifying COX-2 activity and 2-arachidonylglycerol metabolites |
| US20040209959A1 (en) * | 2001-07-16 | 2004-10-21 | Edward Hogestatt | Congeners of acetaminophen and related compounds as substrates for fatty acid conjugation and their use in treatment of pain, fever and inflammation |
| CA2519189C (fr) | 2003-05-07 | 2012-07-17 | Osteologix A/S | Sels de strontium solubles dans l'eau pour le traitement de maladies des cartilages et/ou des os |
| KR100780983B1 (ko) * | 2003-07-31 | 2007-11-30 | 파마시아 앤드 업존 캄파니 엘엘씨 | 소염제의 분산성 제제 |
| WO2006123247A2 (fr) * | 2005-05-20 | 2006-11-23 | Pfizer Limited | Combinaisons synergiques |
| WO2008122967A2 (fr) | 2007-04-04 | 2008-10-16 | Sigmoid Pharma Limited | Composition pharmaceutique orale |
| WO2008132707A1 (fr) | 2007-04-26 | 2008-11-06 | Sigmoid Pharma Limited | Fabrication de minicapsules multiples |
| US9278070B2 (en) | 2009-05-18 | 2016-03-08 | Sigmoid Pharma Limited | Composition comprising oil drops |
| EP2464341B1 (fr) | 2009-08-12 | 2022-07-06 | Sublimity Therapeutics Limited | Compositions immunomodulatrices comprenant une matrice polymère et une phase huileuse |
| GB201020032D0 (en) | 2010-11-25 | 2011-01-12 | Sigmoid Pharma Ltd | Composition |
| GB201212010D0 (en) | 2012-07-05 | 2012-08-22 | Sigmoid Pharma Ltd | Formulations |
| GB201319791D0 (en) | 2013-11-08 | 2013-12-25 | Sigmoid Pharma Ltd | Formulations |
| DK3113774T3 (da) | 2014-03-06 | 2022-03-07 | Elanco Animal Health Incorporated | Sammensætninger af grapiprant og fremgangsmåder til anvendelse deraf |
| EA036036B1 (ru) | 2014-11-07 | 2020-09-16 | Сигмойд Фарма Лимитед | Композиции, содержащие циклоспорин |
| US12109218B2 (en) | 2014-12-09 | 2024-10-08 | Aratana Therapeutics, Inc. | Compositions of grapiprant and methods for using the same |
| MX2017009011A (es) * | 2015-01-09 | 2017-10-02 | Jaguar Animal Health | Metodos para tratar la diarrea en animales de compañia. |
| JP2023520367A (ja) * | 2020-03-25 | 2023-05-17 | エスアールアイ インターナショナル | リポキシゲナーゼ阻害剤 |
| US11116737B1 (en) | 2020-04-10 | 2021-09-14 | University Of Georgia Research Foundation, Inc. | Methods of using probenecid for treatment of coronavirus infections |
| KR102404883B1 (ko) | 2020-11-30 | 2022-06-07 | (주)이노보테라퓨틱스 | 벤즈브로마론을 포함하는 켈로이드 또는 비대흉터 예방 또는 치료용 약학 조성물 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| US3896145A (en) * | 1972-07-24 | 1975-07-22 | Hoffmann La Roche | Carbazoles |
| CA1319886C (fr) * | 1987-02-03 | 1993-07-06 | Alberto Ferro | Solutions de micelles mixtes |
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1998
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