JP2000508312A5 - - Google Patents
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- Publication number
- JP2000508312A5 JP2000508312A5 JP1997536189A JP53618997A JP2000508312A5 JP 2000508312 A5 JP2000508312 A5 JP 2000508312A5 JP 1997536189 A JP1997536189 A JP 1997536189A JP 53618997 A JP53618997 A JP 53618997A JP 2000508312 A5 JP2000508312 A5 JP 2000508312A5
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US1549996P | 1996-04-11 | 1996-04-11 | |
| US60/015,499 | 1996-04-11 | ||
| PCT/US1997/003458 WO1997037980A1 (en) | 1996-04-11 | 1997-03-28 | Process to prepare oxazolidinones |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008053675A Division JP2008239621A (ja) | 1996-04-11 | 2008-03-04 | オキサゾリジノンの製法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2000508312A JP2000508312A (ja) | 2000-07-04 |
| JP2000508312A5 true JP2000508312A5 (cg-RX-API-DMAC7.html) | 2004-12-02 |
Family
ID=21771765
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP9536189A Ceased JP2000508312A (ja) | 1996-04-11 | 1997-03-28 | オキサゾリジノンの製法 |
| JP2008053675A Withdrawn JP2008239621A (ja) | 1996-04-11 | 2008-03-04 | オキサゾリジノンの製法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008053675A Withdrawn JP2008239621A (ja) | 1996-04-11 | 2008-03-04 | オキサゾリジノンの製法 |
Country Status (24)
Families Citing this family (56)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9601666D0 (en) * | 1996-01-27 | 1996-03-27 | Zeneca Ltd | Chemical compounds |
| GB9702213D0 (en) * | 1996-02-24 | 1997-03-26 | Zeneca Ltd | Chemical compounds |
| GB9609919D0 (en) * | 1996-05-11 | 1996-07-17 | Zeneca Ltd | Chemical compounds |
| GB9717804D0 (en) | 1997-08-22 | 1997-10-29 | Zeneca Ltd | Chemical compounds |
| GB9717807D0 (en) | 1997-08-22 | 1997-10-29 | Zeneca Ltd | Chemical compounds |
| GB9725244D0 (en) | 1997-11-29 | 1998-01-28 | Zeneca Ltd | Chemical compounds |
| TR200003595T2 (tr) * | 1998-06-05 | 2001-07-23 | Astrazeneca Ab | Kimyasal bileşikler |
| US6403804B1 (en) * | 1998-12-07 | 2002-06-11 | Takasago International Corporation | Process for preparing optically active oxazolidinone derivative |
| ATE293616T1 (de) | 1999-02-01 | 2005-05-15 | Upjohn Co | 2-fluoro-(oxido-thiopyran-4-yl)benzol derivate |
| US6608081B2 (en) * | 1999-08-12 | 2003-08-19 | Ortho-Mcneil Pharmaceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
| US6413981B1 (en) | 1999-08-12 | 2002-07-02 | Ortho-Mcneil Pharamceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
| US6297242B1 (en) | 1999-08-12 | 2001-10-02 | Ortho-Mcneil Pharmaceutical, Inc. | N-substituted amidine and guanidine oxazolidinone antibacterials and methods of use thereof |
| GB9928568D0 (en) | 1999-12-03 | 2000-02-02 | Zeneca Ltd | Chemical compounds |
| US6518285B2 (en) | 1999-12-21 | 2003-02-11 | Ortho Mcneil Pharmaceutical, Inc. | Piperidinyloxy and pyrrolidinyloxy oxazolidinone antibacterials |
| US6444813B2 (en) | 2000-02-02 | 2002-09-03 | Pharmacia & Upjohn Company | Linezolid-crystal form II |
| AR027261A1 (es) * | 2000-02-02 | 2003-03-19 | Upjohn Co | Linezolid forma cristalina ii |
| MY127336A (en) * | 2000-03-22 | 2006-11-30 | Upjohn Co | Container for linezolid iv solution |
| US6514529B2 (en) | 2000-03-22 | 2003-02-04 | Pharmacia & Upjohn Company | Oxazolidinone tablet formulation |
| GB0009803D0 (en) * | 2000-04-25 | 2000-06-07 | Astrazeneca Ab | Chemical compounds |
| DK1301207T3 (da) | 2000-06-30 | 2005-10-10 | Pharmacia & Upjohn Co Llc | Sammensætninger til behandling af bakterieinfektioner indeholdende en oxazolidinonforbindelse, sulbactam og ampicillin |
| PE20020300A1 (es) * | 2000-08-22 | 2002-05-10 | Pharmacia Corp | Composicion de solucion de un farmaco antibiotico a base de oxazolidinona con mejoramiento de la carga de farmaco |
| US6288239B1 (en) | 2000-09-19 | 2001-09-11 | Board Of Trustees Operating Michigan State University | 5-trityloxymethyl-oxazolidinones and process for the preparation thereof |
| AR031135A1 (es) | 2000-10-10 | 2003-09-10 | Upjohn Co | Composiciones de antibiotico topico para el tratamiento de infecciones oculares |
| ATE332299T1 (de) * | 2001-04-07 | 2006-07-15 | Astrazeneca Ab | Eine sulfonimid-gruppe enthaltende oxazolidinone als antibiotika |
| CA2440600A1 (en) * | 2001-04-20 | 2002-10-31 | Pharmacia & Upjohn Company | Process to prepare oxazolidinones |
| ES2186550B2 (es) * | 2001-06-27 | 2003-11-16 | Vita Lab | Nuevos derivados de oxazolidinonas como antibacterianos. |
| EP1578723A4 (en) * | 2001-10-18 | 2006-11-02 | Univ Michigan State | Process for the preparation of oxazolidinones and method of use thereof |
| AR038576A1 (es) * | 2002-02-22 | 2005-01-19 | Pharmacia Corp | Formulaciones de drogas antibioticas oftalmicas que contienen un compuesto de ciclodextrina y cloruro de cetil piridinio |
| AU2003213210A1 (en) * | 2002-02-22 | 2003-09-09 | Pharmacia Corporation | Ophthalmic formulation with gum system |
| HUE051230T2 (hu) | 2003-10-16 | 2021-03-01 | Symed Labs Ltd | Linezolid kristályos formája |
| ES2294494T3 (es) * | 2004-04-19 | 2008-04-01 | Symed Labs Limited | Un nuevo procedimiento para la preparacion de linezolid y compuestos relacionados. |
| US7429661B2 (en) * | 2004-07-20 | 2008-09-30 | Symed Labs Limited | Intermediates for linezolid and related compounds |
| RU2008139612A (ru) * | 2006-04-07 | 2010-04-20 | Пфайзер Продактс Инк. (Us) | Способ получения линезолида |
| CN100395270C (zh) * | 2006-05-25 | 2008-06-18 | 湖北大学 | 线型聚苯乙烯支载的(4s)-5,5-二取代基噁唑烷酮及其制备方法和用途 |
| EP2033960A3 (en) * | 2007-09-04 | 2009-04-29 | Dipharma Francis S.r.l. | Linezolid crystalline hydrate form and linezolid salts |
| US20090093631A1 (en) * | 2007-09-06 | 2009-04-09 | Ben-Zion Dolitzky | Processes for the preparation of a linezolid intermediate, linezolid hydroxide |
| EP2163547A1 (en) | 2008-09-16 | 2010-03-17 | Unión Químico Farmacéutica, S.A. (UQUIFA) | Process for the preparation of an oxazolidinone antibacterial agent and intermediates thereof |
| JP5561462B2 (ja) * | 2009-09-17 | 2014-07-30 | 日東化成株式会社 | 漁網防汚塗料組成物、該組成物を用いて形成される防汚塗膜、該塗膜の形成方法、および該塗膜を表面に有する漁網、漁網用具又は水中構造物 |
| CA2785620A1 (en) | 2009-12-26 | 2011-06-30 | Alembic Pharmaceuticals Limited | Process for the preparation of linezolid |
| EP2521723A1 (en) | 2010-01-04 | 2012-11-14 | Enantia, S.L. | Process for the preparation of rivaroxaban and intermediates thereof |
| EP2603505A1 (en) | 2010-08-11 | 2013-06-19 | Synthon BV | Process for making linezolid |
| EP2690100A1 (en) | 2010-08-11 | 2014-01-29 | Synhton B.V. | Process for making linezolid |
| WO2012059823A1 (en) | 2010-11-03 | 2012-05-10 | Wockhardt Limited | Process for the preparation of phosphoric acid mono- (l-{4- [(s) -5- (acetylaminomethyl) - 2 - oxo - oxazolidin- 3 - yl] - 2, 6 - difluorophenyl} - 4 -methoxymethylpiperidin- 4 - yl) ester |
| WO2012094622A2 (en) * | 2011-01-07 | 2012-07-12 | The Regents Of The University Of California | Amination of aryl alcohol derivatives |
| CN102153521B (zh) * | 2011-01-31 | 2012-09-12 | 宁波市鄞州百特佳医药科技有限公司 | 一种用于制备利奈唑胺的中间体及其制备方法 |
| WO2012114354A1 (en) | 2011-02-24 | 2012-08-30 | Lee Pharma Limited | Anhydrous linezolid crystalline form-ii |
| SI2595968T1 (sl) | 2011-02-24 | 2016-01-29 | Lee Pharma Limited | Novi postopek za pripravo linezolida in njegovih novih intermediatov |
| CN102311402B (zh) * | 2011-07-18 | 2013-08-21 | 苏州敬业医药化工有限公司 | 3-取代苯基-5-羟甲基噁唑烷-2-酮的制备方法 |
| CN102321042B (zh) * | 2011-07-18 | 2013-12-04 | 苏州敬业医药化工有限公司 | 3-取代苯基-5-羟甲基噁唑烷-2-酮的制备方法 |
| WO2013072923A1 (en) | 2011-09-19 | 2013-05-23 | Cadila Healthcare Limited | Process for the preparation of crystalline linezolid |
| WO2013111048A1 (en) | 2012-01-24 | 2013-08-01 | Jubilant Life Sciences Limited | Improved process for the preparation of stable crystalline form-i of linezolid, substantially free of residual solvent |
| CN103626712B (zh) * | 2012-08-23 | 2016-06-01 | 重庆药友制药有限责任公司 | 一种用于制备利奈唑胺的中间体及其制备方法 |
| WO2014071990A1 (en) | 2012-11-09 | 2014-05-15 | Synthon Bv | Process for making linezolid |
| WO2015173664A1 (en) | 2014-05-14 | 2015-11-19 | Wockhardt Limited | Process for the preparation of (5s)-n-{3-[3,5-difluoro-4-(4-hydroxy-4-methoxymethyl-piperidin-1-yl)-phenyl]-2-oxo-oxazolidin-5-ylmethyl}-acetamide |
| WO2021184339A1 (en) | 2020-03-20 | 2021-09-23 | Merck Sharp & Dohme Corp. | Oxazolidinone compound and methods of use thereof as an antibacterial agent |
| CN119119019B (zh) * | 2024-09-11 | 2025-11-11 | 遵义医科大学 | 一种杂环磺酰胺/磺酸酯衍生物及其制备方法、应用 |
Family Cites Families (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA681830A (en) * | 1964-03-10 | X. Markley Francis | Process for 5-(aryloxymethyl)-2-oxazolidinones | |
| US3547951A (en) * | 1969-06-17 | 1970-12-15 | Waldo R Hardie | 1,3-dioxolan-4-yl-alkyl guanidines |
| FR2315925A1 (fr) * | 1975-07-04 | 1977-01-28 | Nippon Chemiphar Co | Nouveaux derives de 5-benzyle-2-oxazolidone, leur procede de preparation et leur application en therapeutique |
| FR2356422A1 (fr) * | 1976-03-01 | 1978-01-27 | Delalande Sa | Nouveaux hydroxymethyl-5 oxazolidinone-2, leur procede de preparation et leur application en therapeutique |
| LU80081A1 (fr) * | 1977-08-26 | 1979-05-15 | Delalande Sa | Nouvelles hydroxymethyl-5 oxazolidinones-2,leur procede de preparation et leur application therapeutique |
| JPS6014032B2 (ja) * | 1978-01-20 | 1985-04-11 | 日本ケミフア株式会社東京 | ５‐フエネチル‐２‐オキサゾリドン誘導体およびその製法 |
| US4340606A (en) * | 1980-10-23 | 1982-07-20 | E. I. Du Pont De Nemours And Company | 3-(p-Alkylsulfonylphenyl)oxazolidinone derivatives as antibacterial agents |
| FR2500450A1 (fr) * | 1981-02-25 | 1982-08-27 | Delalande Sa | Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique |
| US4461773A (en) * | 1982-09-15 | 1984-07-24 | E. I. Dupont De Nemours And Company | P-Oxooxazolidinylbenzene compounds as antibacterial agents |
| US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
| US5225565A (en) * | 1988-09-15 | 1993-07-06 | The Upjohn Company | Antibacterial 3-(fused-ring substituted)phenyl-5β-amidomethyloxazolidin-2-ones |
| US5182403A (en) * | 1988-09-15 | 1993-01-26 | The Upjohn Company | Substituted 3(5'indazolyl) oxazolidin-2-ones |
| US5164510A (en) * | 1988-09-15 | 1992-11-17 | The Upjohn Company | 5'Indolinyl-5β-amidomethyloxazolidin-2-ones |
| US5231188A (en) * | 1989-11-17 | 1993-07-27 | The Upjohn Company | Tricyclic [6.5.51]-fused oxazolidinone antibacterial agents |
| JP2908510B2 (ja) * | 1990-04-20 | 1999-06-21 | イハラケミカル工業株式会社 | ベンジルアミン類の製造方法 |
| EP0530812B1 (en) * | 1991-09-05 | 1996-05-22 | Nippon Paint Co., Ltd. | Thermosetting resinous composition containing polyfunctional oxazolidinone component and polyamine component |
| CA2119556C (en) * | 1991-11-01 | 2004-07-06 | Michael Robert Barbachyn | Substituted aryl- and heteroaryl-phenyloxazolidinones |
| SK283420B6 (sk) * | 1992-05-08 | 2003-07-01 | Pharmacia & Upjohn Company | Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny |
| MY115155A (en) * | 1993-09-09 | 2003-04-30 | Upjohn Co | Substituted oxazine and thiazine oxazolidinone antimicrobials. |
| JPH0873455A (ja) * | 1994-03-15 | 1996-03-19 | Upjohn Co:The | オキサゾリジノン誘導体及びこれを有効成分とする医薬組成物 |
| PT788498E (pt) * | 1994-10-26 | 2002-02-28 | Upjohn Co | Compostos antimicrobianos de feniloxazolidinona |
| ES2193201T3 (es) * | 1994-11-15 | 2003-11-01 | Upjohn Co | Agentes antibacterianos tipo oxazolidonas sustituidas con oxazina y tiazina biciclica. |
| CN1068328C (zh) * | 1995-05-11 | 2001-07-11 | 法玛西雅厄普约翰美国公司 | 螺环和双环二嗪基和咔嗪基噁唑烷酮类 |
-
1997
- 1997-03-28 RU RU98120398/04A patent/RU2176643C2/ru not_active IP Right Cessation
- 1997-03-28 ES ES01302264T patent/ES2298198T3/es not_active Expired - Lifetime
- 1997-03-28 SG SG9905133A patent/SG85683A1/en unknown
- 1997-03-28 NZ NZ332278A patent/NZ332278A/xx unknown
- 1997-03-28 CN CNB031594743A patent/CN1319952C/zh not_active Expired - Fee Related
- 1997-03-28 SI SI9730273T patent/SI0892792T1/xx unknown
- 1997-03-28 JP JP9536189A patent/JP2000508312A/ja not_active Ceased
- 1997-03-28 DK DK97915865T patent/DK0892792T3/da active
- 1997-03-28 PT PT01302264T patent/PT1114819E/pt unknown
- 1997-03-28 DK DK01302264T patent/DK1114819T3/da active
- 1997-03-28 AU AU23182/97A patent/AU706117B2/en not_active Ceased
- 1997-03-28 ES ES97915865T patent/ES2166073T3/es not_active Expired - Lifetime
- 1997-03-28 AT AT01302264T patent/ATE383347T1/de not_active IP Right Cessation
- 1997-03-28 EP EP01302264A patent/EP1114819B1/en not_active Expired - Lifetime
- 1997-03-28 CZ CZ0287198A patent/CZ298060B6/cs not_active IP Right Cessation
- 1997-03-28 DE DE69738457T patent/DE69738457T2/de not_active Expired - Fee Related
- 1997-03-28 DE DE69709718T patent/DE69709718T2/de not_active Expired - Fee Related
- 1997-03-28 CZ CZ2007-88A patent/CZ200788A3/cs unknown
- 1997-03-28 KR KR10-2004-7009934A patent/KR100530297B1/ko not_active Expired - Fee Related
- 1997-03-28 US US08/828,923 patent/US5837870A/en not_active Expired - Fee Related
- 1997-03-28 SK SK1336-98A patent/SK284703B6/sk unknown
- 1997-03-28 PT PT97915865T patent/PT892792E/pt unknown
- 1997-03-28 CA CA002248143A patent/CA2248143C/en not_active Expired - Fee Related
- 1997-03-28 WO PCT/US1997/003458 patent/WO1997037980A1/en not_active Ceased
- 1997-03-28 CN CNB011330031A patent/CN1167701C/zh not_active Expired - Fee Related
- 1997-03-28 CN CN97193658A patent/CN1082953C/zh not_active Expired - Fee Related
- 1997-03-28 AT AT97915865T patent/ATE209193T1/de not_active IP Right Cessation
- 1997-03-28 PL PL329295A patent/PL192691B1/pl not_active IP Right Cessation
- 1997-03-28 HU HU0500044A patent/HUP0500044A3/hu unknown
- 1997-03-28 EP EP97915865A patent/EP0892792B1/en not_active Expired - Lifetime
- 1997-04-02 TW TW086104216A patent/TW449593B/zh not_active IP Right Cessation
- 1997-04-08 ZA ZA972983A patent/ZA972983B/xx unknown
-
1998
- 1998-10-09 NO NO19984737A patent/NO311837B1/no unknown
-
2001
- 2001-10-26 NO NO20015253A patent/NO312728B1/no unknown
-
2008
- 2008-03-04 JP JP2008053675A patent/JP2008239621A/ja not_active Withdrawn