JP2000505084A5 - - Google Patents

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Publication number
JP2000505084A5
JP2000505084A5 JP1997530192A JP53019297A JP2000505084A5 JP 2000505084 A5 JP2000505084 A5 JP 2000505084A5 JP 1997530192 A JP1997530192 A JP 1997530192A JP 53019297 A JP53019297 A JP 53019297A JP 2000505084 A5 JP2000505084 A5 JP 2000505084A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP1997530192A
Other languages
English (en)
Japanese (ja)
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JP2000505084A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US1997/001970 external-priority patent/WO1997030981A1/en
Publication of JP2000505084A publication Critical patent/JP2000505084A/ja
Publication of JP2000505084A5 publication Critical patent/JP2000505084A5/ja
Withdrawn legal-status Critical Current

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JP9530192A 1996-02-26 1997-02-18 アゾリルピペラジニルフェニルオキサゾリジノン抗微生物剤 Withdrawn JP2000505084A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US1231696P 1996-02-26 1996-02-26
US60/012,316 1996-02-26
PCT/US1997/001970 WO1997030981A1 (en) 1996-02-26 1997-02-18 Azolyl piperazinyl phenyl oxazolidinone antimicrobials

Publications (2)

Publication Number Publication Date
JP2000505084A JP2000505084A (ja) 2000-04-25
JP2000505084A5 true JP2000505084A5 (cg-RX-API-DMAC7.html) 2004-11-25

Family

ID=21754387

Family Applications (1)

Application Number Title Priority Date Filing Date
JP9530192A Withdrawn JP2000505084A (ja) 1996-02-26 1997-02-18 アゾリルピペラジニルフェニルオキサゾリジノン抗微生物剤

Country Status (18)

Country Link
US (1) US5736545A (cg-RX-API-DMAC7.html)
EP (1) EP0883611B1 (cg-RX-API-DMAC7.html)
JP (1) JP2000505084A (cg-RX-API-DMAC7.html)
KR (1) KR19990087238A (cg-RX-API-DMAC7.html)
CN (1) CN1082952C (cg-RX-API-DMAC7.html)
AT (1) ATE221521T1 (cg-RX-API-DMAC7.html)
AU (1) AU703831B2 (cg-RX-API-DMAC7.html)
DE (1) DE69714418T2 (cg-RX-API-DMAC7.html)
DK (1) DK0883611T3 (cg-RX-API-DMAC7.html)
ES (1) ES2180945T3 (cg-RX-API-DMAC7.html)
ID (1) ID18467A (cg-RX-API-DMAC7.html)
MY (1) MY116093A (cg-RX-API-DMAC7.html)
NZ (1) NZ331011A (cg-RX-API-DMAC7.html)
PE (1) PE55898A1 (cg-RX-API-DMAC7.html)
PT (1) PT883611E (cg-RX-API-DMAC7.html)
TW (1) TW442460B (cg-RX-API-DMAC7.html)
WO (1) WO1997030981A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA971287B (cg-RX-API-DMAC7.html)

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GB9601666D0 (en) * 1996-01-27 1996-03-27 Zeneca Ltd Chemical compounds
GB9702213D0 (en) * 1996-02-24 1997-03-26 Zeneca Ltd Chemical compounds
GB9609919D0 (en) * 1996-05-11 1996-07-17 Zeneca Ltd Chemical compounds
WO1999002525A1 (en) * 1997-07-11 1999-01-21 Pharmacia & Upjohn Company Thiadiazolyl and oxadiazolyl phenyl oxazolidinone antibacterial agents
GB9717804D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
GB9717807D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
GB9725244D0 (en) 1997-11-29 1998-01-28 Zeneca Ltd Chemical compounds
US6562844B2 (en) 1998-01-23 2003-05-13 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
US7002020B1 (en) 1998-01-23 2006-02-21 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
AU764184B2 (en) 1998-01-23 2003-08-14 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
TR200003595T2 (tr) * 1998-06-05 2001-07-23 Astrazeneca Ab Kimyasal bileşikler
ATE238662T1 (de) * 1998-08-04 2003-05-15 Ciba Sc Holding Ag Verwendung von oxathiazolonen als mikrobizide
WO2000045177A1 (en) 1999-01-27 2000-08-03 Pharmacia & Upjohn Company Assays for modulators of elongation factor p activity
GB9928568D0 (en) 1999-12-03 2000-02-02 Zeneca Ltd Chemical compounds
PE20010851A1 (es) * 1999-12-14 2001-08-17 Upjohn Co Esteres del acido benzoico de oxazolidinonas que tienen un substituyente hidroxiacetilpiperazina
GB0009803D0 (en) * 2000-04-25 2000-06-07 Astrazeneca Ab Chemical compounds
WO2003008389A1 (en) * 2001-07-16 2003-01-30 Ranbaxy Laboratories Limited Oxazolidinone derivatives as potential antimicrobials
BR0112826A (pt) * 2000-07-17 2003-06-24 Ranbaxy Lab Ltd Derivados da oxazolidinona como antimicrobianos
JP2005503435A (ja) * 2001-04-17 2005-02-03 メルク アンド カンパニー インコーポレーテッド ビシクロ[3.1.0]ヘキサン含有オキサゾリジノン抗生物質及びその誘導体
KR20040106551A (ko) * 2002-05-15 2004-12-17 랜박시 래보러터리스 리미티드 페닐 옥사졸리디논 유도체의 다형 제제
CN1668308A (zh) * 2002-07-29 2005-09-14 兰贝克赛实验室有限公司 作为抗菌剂的噁唑烷酮衍生物
MXPA05001558A (es) 2002-08-12 2005-09-08 Pharmacia & Upjohn Co Llc N-aril-2-oxazolidinonas y sus derivados.
AU2002339721A1 (en) * 2002-09-20 2004-04-08 Lupin Limited Oxazolidinone derivatives, process for their preperation and their use as antimycobacterial agents
EP1565186B1 (en) 2002-11-21 2006-11-02 Pharmacia & Upjohn Company LLC N-(4-(piperazin-1-yl)-phenyl-2-oxazolidinone-5-carboxamide derivates and related compounds as antibacterial agents
CA2529292A1 (en) * 2003-07-02 2005-01-20 Merck & Co., Inc. Oxazolidinone antibiotics and derivatives thereof
AU2004256085B2 (en) * 2003-07-02 2007-12-06 Kyorin, Pharmaceutical Co., Ltd. Cyclopropyl Group Substituted Oxazolydinone Antibiotics and Derivatives Thereof
KR20060113625A (ko) * 2003-07-02 2006-11-02 머크 앤드 캄파니 인코포레이티드 시클로프로필기 치환된 옥사졸리디논 항생제 및 그의유도체
US20070293493A1 (en) * 2003-07-02 2007-12-20 Milton Hammond Oxazolidinone antibiotics and derivatives thereof
WO2005051933A1 (en) * 2003-11-28 2005-06-09 Ranbaxy Laboratories Limited An improved process for the synthesis of 4-(4-benzyloxy-carbonylamino-2-fluorophenyl)-piperazine-1-carboxylic acid tert-butyl ester, a key intermediate for oxazolidinone antimicrobials and compounds prepared thereby
WO2005082899A1 (en) * 2004-01-28 2005-09-09 Ranbaxy Laboratories Limited Oxazolidinone derivatives as antimicrobials
US8686011B2 (en) 2004-05-24 2014-04-01 Amgen Inc. Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1
AR049344A1 (es) * 2004-05-24 2006-07-19 Amgen Inc Inhibidores de la 11-beta-hidroxi esteroide deshidrogenasa de tipo 1
WO2006035283A1 (en) * 2004-09-27 2006-04-06 Ranbaxy Laboratories Limited Oxazolidinone derivatives as antimicrobials
WO2006043121A1 (en) * 2004-10-20 2006-04-27 Ranbaxy Laboratories Limited Oxazolidinone derivatives as antimicrobials
WO2006051408A1 (en) * 2004-11-11 2006-05-18 Ranbaxy Laboratories Limited Oxazolidinone derivatives as antimicrobials
EP1912980A2 (en) * 2005-06-20 2008-04-23 Wockhardt Limited Oxazolidinones bearing antimicrobial activity composition and methods of preparation
JO2769B1 (en) 2005-10-26 2014-03-15 جانسين فارماسوتيكا ان. في Rapid decomposition of physiologically antagonistic agents of the 2-dopamine receptor
CN100406455C (zh) * 2006-02-20 2008-07-30 中国科学院上海药物研究所 含三氮唑基的噁唑烷酮类化合物及其制备方法和用途
JO2642B1 (en) * 2006-12-08 2012-06-17 جانسين فارماسوتيكا ان. في Dopamine 2 receptor antagonists are rapidly hydrolyzed
JO2849B1 (en) 2007-02-13 2015-03-15 جانسين فارماسوتيكا ان. في Dopamine 2 receptor antagonists are rapidly hydrolyzed
RU2489431C2 (ru) * 2007-04-23 2013-08-10 Янссен Фармацевтика Н.В. Тиа(диа)золы как быстро диссоциирующие антагонисты рецептора допамина 2
JP5431305B2 (ja) * 2007-04-23 2014-03-05 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 高速解離性ドパミン2受容体アンタゴニストとしての4−アルコキシピリダジン誘導体
JP2010525013A (ja) * 2007-04-23 2010-07-22 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 高速解離性ドパミン2受容体アンタゴニストとしてのピリジン誘導体
CA2712613C (en) * 2008-03-26 2017-02-28 Global Alliance For Tb Drug Development Bicyclic nitroimidazoles covalently linked to substituted phenyl oxazolidinones
CN102159554B (zh) * 2008-07-03 2014-09-24 詹森药业有限公司 作为5-ht6受体拮抗剂的取代的6-(1-哌嗪基)-哒嗪
KR101609218B1 (ko) * 2008-07-31 2016-04-05 얀센 파마슈티카 엔.브이. 속해리성 도파민 2 수용체 길항제로서의 피페라진-1-일-트리플루오로메틸-치환된-피리딘
WO2011152442A1 (ja) * 2010-06-03 2011-12-08 塩野義製薬株式会社 2-クロロ-6-フルオロベンゾオキサゾールの製造方法
CN102079730B (zh) * 2010-09-06 2013-10-16 贵州大学 一类含2,5-取代杂环基砜类衍生物及其合成方法和应用
CN103450173B (zh) * 2013-09-07 2015-06-03 吉首大学 吡咯酮-苯基-噁唑烷酮型化合物及其制法和用途
CN103709119B (zh) * 2013-12-04 2015-05-20 上海应用技术学院 一种制备5-氨基噻唑-4-甲酰胺的方法
CN104202835A (zh) * 2014-09-03 2014-12-10 苏州微站通信科技有限公司 Ue进入静默期时让基站及时释放时频资源的方法
US11548882B2 (en) 2018-04-27 2023-01-10 Osaka University Benzisoxazole compound
US12479816B2 (en) 2019-02-08 2025-11-25 University of Pittsburgh—of the Commonwealth System of Higher Education 20-HETE formation inhibitors

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US4921869A (en) * 1987-10-09 1990-05-01 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4801600A (en) * 1987-10-09 1989-01-31 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4977173A (en) * 1987-10-21 1990-12-11 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl ethenylbenzene derivatives useful as antibacterial agents
US4948801A (en) * 1988-07-29 1990-08-14 E. I. Du Pont De Nemours And Company Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
US5254577A (en) * 1988-07-29 1993-10-19 The Du Pont Merck Pharmaceutical Company Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
SK283420B6 (sk) * 1992-05-08 2003-07-01 Pharmacia & Upjohn Company Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny
MY115155A (en) * 1993-09-09 2003-04-30 Upjohn Co Substituted oxazine and thiazine oxazolidinone antimicrobials.
ATE182142T1 (de) * 1993-11-22 1999-07-15 Upjohn Co Substituierte hydroxyacetyl piperazine phenyl oxazolidinonsäureester

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